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Direct Synthesis of Diverse 2-Aminobenzo[<i>b</i>]thiophenes via Palladium-Catalyzed Carbon–Sulfur Bond Formation Using Na<sub>2</sub>S<sub>2</sub>O<sub>3</sub>as the Sulfur Source

https://doi.org/10.1021/ol502381e
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Every reference with a DOI in the deposited reference list resolved to a known work in Crossref or DataCite at the dated check, and none carried a retraction, withdrawal, or removal notice.

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The 25 checked references that resolve
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Synthesis and binding affinities of fluoroalkylated raloxifenes
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Structure−Activity Relationships of Selective Estrogen Receptor Modulators:  Modifications to the 2-Arylbenzothiophene Core of Raloxifene
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Synthesis and Pharmacology of Conformationally Restricted Raloxifene Analogues:  Highly Potent Selective Estrogen Receptor Modulators
resolves10.1016/j.bmcl.2004.12.074
Benzothiophenes containing a piperazine side chain as selective ligands for the estrogen receptor α and their bioactivities in vivo
resolves10.1016/j.bmcl.2012.04.047
Design, synthesis, and structure–activity relationships of novel spiro-piperidines as acetyl-CoA carboxylase inhibitors
resolves10.1016/j.bmc.2011.01.041
Discovery of novel (4-piperidinyl)-piperazines as potent and orally active acetyl-CoA carboxylase 1/2 non-selective inhibitors: F-Boc and triF-Boc groups are acid-stable bioisosteres for the Boc group
resolves10.1016/j.bmcl.2006.02.049
New HIV-1 reverse transcriptase inhibitors based on a tricyclic benzothiophene scaffold: Synthesis, resolution, and inhibitory activity
resolves10.1021/jm2000773
Novel Benzo[<i>b</i>]thiophene Derivatives as New Potential Antidepressants with Rapid Onset of Action
resolves10.1021/jm070050f
Synthesis and Biological Evaluation of 2- and 3-Aminobenzo[<i>b</i>]thiophene Derivatives as Antimitotic Agents and Inhibitors of Tubulin Polymerization
resolves10.1016/j.bmc.2010.05.068
Substituted 2-(3′,4′,5′-trimethoxybenzoyl)-benzo[b]thiophene derivatives as potent tubulin polymerization inhibitors
resolves10.1021/jm4013938
Concise Synthesis and Biological Evaluation of 2-Aroyl-5-Amino Benzo[<i>b</i>]thiophene Derivatives As a Novel Class of Potent Antimitotic Agents
resolves10.1021/cc900172u
Diverse Methyl Sulfone-Containing Benzo[<i>b</i>]thiophene Library via Iodocyclization and Palladium-Catalyzed Coupling
resolves10.1021/ol100816g
One-Pot Synthesis of Amine-Substituted Aryl Sulfides and Benzo[<i>b</i>]thiophene Derivatives
resolves10.1021/jo401353w
Copper-Catalyzed Synthesis of Benzo[<i>b</i>]thiophenes and Benzothiazoles Using Thiocarboxylic Acids as a Coupling Partner
resolves10.1021/ol401981w
A New Synthesis of Benzo[<i>b</i>]thiophene-2-thiolates and Their Derivatives <i>via</i> Base-Promoted Transformation of 4-(2-Mercaptophenyl)-1,2,3-thiadiazoles
resolves10.1021/jo01023a021
2-Aminobenzo[b]thiophene. An Aromatic Ring Tautomer<sup>1,2</sup>
resolves10.1002/anie.200603089
General Preparation of Primary, Secondary, and Tertiary Aryl Amines by the Oxidative Coupling of Polyfunctional Aryl and Heteroaryl Amidocuprates
resolves10.1016/j.tet.2010.01.069
A convenient approach towards 2- and 3-aminobenzo[b]thiophenes
resolves10.1139/v87-302
Destabilized carbocations. Nuclear magnetic resonance detection and reactivities of aryl α-thioformamidyl cations
resolves10.1002/anie.200700619
Highly Selective Thiiranation of 1,2‐Allenyl Sulfones with Br<sub>2</sub> and Na<sub>2</sub>S<sub>2</sub>O<sub>3</sub>: Mechanism and Asymmetric Synthesis of Alkylidenethiiranes
resolves10.1021/ol400618k
Efficient Access to 1,4-Benzothiazine: Palladium-Catalyzed Double C–S Bond Formation Using Na<sub>2</sub>S<sub>2</sub>O<sub>3</sub> as Sulfurating Reagent
resolves10.1021/ol500112y
Direct Cross-Coupling Access to Diverse Aromatic Sulfide: Palladium-Catalyzed Double C–S Bond Construction Using Na<sub>2</sub>S<sub>2</sub>O<sub>3</sub> as a Sulfurating Reagent
resolves10.1021/ol5009747
A Highly Efficient Cu-Catalyzed S-Transfer Reaction: From Amine to Sulfide
resolves10.1002/ejoc.201201061
A Microwave‐Assisted Domino Benzannulation Reaction towards Functionalized Naphthalenes, Quinolines, and Isoquinolines
resolves10.1039/c3ob40103k
Palladium(ii)-catalyzed synthesis of functionalized indenones via oxidation and cyclization of 2-(2-arylethynylphenyl)acetonitriles
The 1 reference without a DOI — listed, not checked
no DOI — not checkedref15/cit15
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