Every reference with a DOI in the deposited reference list resolved to a known
work in Crossref or DataCite at the dated check, and none carried a retraction,
withdrawal, or removal notice.
The 46 checked references that resolve
resolves10.1038/nrd2590The exploration of macrocycles for drug discovery — an underexploited structural class
resolves10.1021/jm1012374Macrocycles Are Great Cycles: Applications, Opportunities, and Challenges of Synthetic Macrocycles in Drug Discovery
resolves10.1002/cmdc.201500450Cyclic and Macrocyclic Peptides as Chemical Tools To Recognise Protein Surfaces and Probe Protein–Protein Interactions
resolves10.1002/anie.201208344Nonproteinogenic Amino Acid Building Blocks for Nonribosomal Peptide and Hybrid Polyketide Scaffolds
resolves10.1039/C4CS00246FPeptide stapling techniques based on different macrocyclisation chemistries
resolves10.1021/jm020017nMolecular Properties That Influence the Oral Bioavailability of Drug Candidates
resolves10.1021/ja400119tA Perfluoroaryl-Cysteine S
<sub>N</sub>
Ar Chemistry Approach to Unprotected Peptide Stapling
resolves10.1038/nature18941Oxidative diversification of amino acids and peptides by small-molecule iron catalysis
resolves10.1038/nprot.2011.324Synthesis of all-hydrocarbon stapled α-helical peptides by ring-closing olefin metathesis
resolves10.1073/pnas.1311706110Template-constrained macrocyclic peptides prepared from native, unprotected precursors
resolves10.1038/nchem.1729A strategy for the diversity-oriented synthesis of macrocyclic scaffolds using multidimensional coupling
resolves10.1038/nchem.1024Regio- and stereodivergent antibiotic oxidative carbocyclizations catalysed by Rieske oxygenase-like enzymes
resolves10.1038/nchem.2237Structure and biosynthesis of a macrocyclic peptide containing an unprecedented lysine-to-tryptophan crosslink
resolves10.1039/c2np20034aStrained cyclophane natural products: Macrocyclization at its limits
resolves10.1039/c2cc36962aPeptidic macrocyclization via palladium-catalyzed chemoselective indole C-2 arylation
resolves10.1038/ncomms8160New peptide architectures through C–H activation stapling between tryptophan–phenylalanine/tyrosine residues
resolves10.1021/ja510233hSite-Selective C(sp<sup>3</sup>)–H Functionalization of Di-, Tri-, and Tetrapeptides at the N-Terminus
resolves10.1039/C6SC05530CSynthesis of bioactive and stabilized cyclic peptides by macrocyclization using C(sp
<sup>3</sup>
)–H activation
resolves10.1002/anie.201201666CH Bond Functionalization: Emerging Synthetic Tools for Natural Products and Pharmaceuticals
resolves10.1039/c1cs15013hRecent developments in natural product synthesis using metal-catalysed C–H bond functionalisation
resolves10.1002/anie.200806273Palladium(II)‐Catalyzed CH Activation/CC Cross‐Coupling Reactions: Versatility and Practicality
resolves10.1021/cr900184ePalladium-Catalyzed Ligand-Directed C−H Functionalization Reactions
resolves10.1021/cr500200xC–H Functionalization in the Synthesis of Amino Acids and Peptides
resolves10.1021/ja054549fHighly Regioselective Arylation of sp<sup>3</sup> C−H Bonds Catalyzed by Palladium Acetate
resolves10.1021/ja910900pAuxiliary-Assisted Palladium-Catalyzed Arylation and Alkylation of sp<sup>2</sup> and sp<sup>3</sup> Carbon−Hydrogen Bonds
resolves10.1021/ar9000058Palladium- and Copper-Catalyzed Arylation of Carbon−Hydrogen Bonds
resolves10.1021/ol061389jNovel Acetoxylation and C−C Coupling Reactions at Unactivated Positions in α-Amino Acid Derivatives
resolves10.1021/acs.accounts.6b00022Syntheses and Transformations of α-Amino Acids via Palladium-Catalyzed Auxiliary-Directed sp<sup>3</sup> C–H Functionalization
resolves10.1021/ol101220xFacile Benzo-Ring Construction via Palladium-Catalyzed Functionalization of Unactivated sp<sup>3</sup> C−H Bonds under Mild Reaction Conditions
resolves10.1002/anie.201305615Use of a Readily Removable Auxiliary Group for the Synthesis of Pyrrolidones by the Palladium‐Catalyzed Intramolecular Amination of Unactivated γ C(sp<sup>3</sup>)H Bonds
resolves10.1246/cl.2010.1118Overview of the Mechanistic Work on the Concerted Metallation–Deprotonation Pathway
resolves10.1039/C4SC01545BPalladium-catalyzed trifluoroacetate-promoted mono-arylation of the β-methyl group of alanine at room temperature: synthesis of β-arylated α-amino acids through sequential C–H functionalization
resolves10.1021/ja512374gThe Mechanism of a Ligand-Promoted C(sp<sup>3</sup>)–H Activation and Arylation Reaction via Palladium Catalysis: Theoretical Demonstration of a Pd(II)/Pd(IV) Redox Manifold
resolves10.1021/jm060230+Parallel Artificial Membrane Permeability Assay: A New Membrane for the Fast Prediction of Passive Human Skin Permeability
The 4 references without a DOI — listed, not checked
no DOI — not checkedRogdan, A. R., Jerome, S. V., Houk, K. N. & James, K. Strained cyclophane macrocycles: impact of progressive ring size reduction on synthesis and structure. J. Am. Chem. Soc. 132, 2127–2138 (2010).
no DOI — not checkedBooker, S. J. Anaerobic functionalization of unactivated C–H bonds. Curr. Opin. Chem. Biol. 13, (58–73 (2009).
no DOI — not checkedFrisch, M. J. et al. Gaussian 09, Revision D.01 (Gaussian, 2009).
no DOI — not checkedMcKeown, M. R. & Bradner, J. E. MYC activation is a hallmark of cancer initiation and maintenance. Cold Spring Harb. Persp. Med. 4, a014241 (2014).
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