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Analysis of Past and Present Synthetic Methodologies on Medicinal Chemistry: Where Have All the New Reactions Gone?

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Outgoing claims: the papers this work cites, builds on, or argues with.

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What points at this work

Incoming claims: where this work appears in other papers’ reference lists and arguments.

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Recent Advances in Chemistry Technologies and Applications to Medicinal Chemistry
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CuI Catalyzed Regio‐ and Stereo‐selective Hydroboration of Ynamides: α‐ and β‐Borylation via Hydro‐Cupration and Borylation
inferred← citeshttps://doi.org/10.1002/ajoc.202300508openalex-snapshot
Assembling of Polyaryls (Terphenyls, Tetraphenyls, Pentaphenyls, and Hexaphenyls) through Pd(II)‐catalyzed C−H Arylation of Biaryl Carboxamides with Iodobiaryls
inferred← citeshttps://doi.org/10.1002/ajoc.202300660openalex-snapshot
Dehydrative Condensation of Carboxylic Acids with Amines Promoted by HBF4/MS 5A
inferred← citeshttps://doi.org/10.1002/ajoc.202400082openalex-snapshot
Synthesis of 3‐Aryl Substituted Triimidazotriazines via Regioselective Direct Arylation
inferred← citeshttps://doi.org/10.1002/ajoc.202400088openalex-snapshot
Photocatalytic (V 2 O 5 /TiO 2 ) Blue LED Mediated Selective Oxidation of Alcohols, Styrene to Aldehydes, and Oxygenation of Alkyl‐Benzene to Ketones
inferred← citeshttps://doi.org/10.1002/ajoc.202400350openalex-snapshot
Efficient Cu‐Based Mixed Oxides Catalyst for α‐Alkylation of Ketones with Alcohols
inferred← citeshttps://doi.org/10.1002/ajoc.202500353openalex-snapshot
Highly Regioselective Butylation of N‐Sulfonyl‐1,2,3‐triazoles by the Formation of Quaternary Carbon‐Centered C(sp3)─N Bonds
inferred← citeshttps://doi.org/10.1002/ajoc.202500559openalex-snapshot
Piano‐Stool Rhodium(V) and Rhodium(IV) Intermediates in C─H Functionalization and B─H Functionalization: Mechanistic Insights and Emerging Reactivity
inferred← citeshttps://doi.org/10.1002/ajoc.202500607openalex-snapshot
Cyclopropenium Ion–Enabled Reductive Amination of Aldehydes With Indolines Without an External Hydride Source
inferred← citeshttps://doi.org/10.1002/ajoc.202500629openalex-snapshot
Mechanochemical Bodroux Reaction: Sustainable Ball Milling Approach for Direct Amidation of Esters
inferred← citeshttps://doi.org/10.1002/ajoc.70271openalex-snapshot
Electrochemical Oxidative N–N Coupling to Construct Benzo[ c ]cinnolines and Azoarenes
inferred← citeshttps://doi.org/10.1002/ajoc.70283openalex-snapshot
Discovery of a Novel Cyclobutanol Scaffold With Anti‐Inflammatory Activity and Its Modular Synthesis
inferred← citeshttps://doi.org/10.1002/ajoc.70371openalex-snapshot
Organocatalyzed Sustainable Annulation to Construct 4‐Amino‐ and 4‐Thioquinoline Scaffolds as Potential Cancer Therapeutics
inferred← citeshttps://doi.org/10.1002/ajoc.70445openalex-snapshot
N ‐Directed Rh‐Catalyzed Regioselective Amidation of Quinoxaline‐2(1 H )‐ones Using Dioxazolones
inferred← citeshttps://doi.org/10.1002/ange.1441281openalex-snapshot
Ligand‐Enabled Stereoselective Coupling of Methylene C(sp 3 )─H Bonds With Alkenyl Bromide via Pd II /Pd 0 /Pd II Catalysis
inferred← citeshttps://doi.org/10.1002/ange.1983055openalex-snapshot
Gold‐Einzelatomkatalysatoren ermöglichen die selektive Shuttle‐Hydrochlorierung von Alkinen
inferred← citeshttps://doi.org/10.1002/ange.201604193openalex-snapshot
Evaluierung neuer Reaktionen zur Steuerung der Wirkstoff‐Forschung: ein Eignungstest
inferred← citeshttps://doi.org/10.1002/ange.201605463openalex-snapshot
Nickel‐Catalyzed Cross‐Coupling of Redox‐Active Esters with Boronic Acids
inferred← citeshttps://doi.org/10.1002/ange.201609394openalex-snapshot
Moderne Strategien zur Synthese funktioneller Fluorophore
inferred← citeshttps://doi.org/10.1002/ange.201705525openalex-snapshot
Mechanistic Insight Leads to a Ligand Which Facilitates the Palladium‐Catalyzed Formation of 2‐(Hetero)Arylaminooxazoles and 4‐(Hetero)Arylaminothiazoles
inferred← citeshttps://doi.org/10.1002/ange.201707906openalex-snapshot
Electrochemically Enabled, Nickel‐Catalyzed Amination
inferred← citeshttps://doi.org/10.1002/ange.201710195openalex-snapshot
Neue Anwendungen der Klick‐Chemie in Zellbiologie und Wirkstoffentwicklung
inferred← citeshttps://doi.org/10.1002/ange.201800364openalex-snapshot
Eisenkatalysierte Kreuzkupplungen in der Synthese von Pharmazeutika: Streben nach Nachhaltigkeit
inferred← citeshttps://doi.org/10.1002/ange.201806271openalex-snapshot
Selective Functionalization of Aminoheterocycles by a Pyrylium Salt
inferred← citeshttps://doi.org/10.1002/ange.201809431openalex-snapshot
Alkyl‐C‐C‐Bindungsbildung durch Nickel/Photoredox‐Kreuzkupplung
inferred← citeshttps://doi.org/10.1002/ange.201812534openalex-snapshot
Hochdurchsatzstrategien zur Entdeckung und Optimierung katalytischer Reaktionen
inferred← citeshttps://doi.org/10.1002/ange.201813233openalex-snapshot
Intermolecular Heck Coupling with Hindered Alkenes Directed by Potassium Carboxylates
inferred← citeshttps://doi.org/10.1002/ange.201900536openalex-snapshot
High‐Throughput Reaction Screening with Nanomoles of Solid Reagents Coated on Glass Beads
inferred← citeshttps://doi.org/10.1002/ange.201901935openalex-snapshot
Evaluierung der Reaktionsbedingungs‐basierten Sensitivität chemischer Transformationen
inferred← citeshttps://doi.org/10.1002/ange.201906130openalex-snapshot
Oxidative Amide Coupling from Functionally Diverse Alcohols and Amines Using Aerobic Copper/Nitroxyl Catalysis
inferred← citeshttps://doi.org/10.1002/ange.201907837openalex-snapshot
N‐Heterocyclic Carbene Catalyzed Concerted Nucleophilic Aromatic Substitution of Aryl Fluorides Bearing α,β‐Unsaturated Amides
inferred← citeshttps://doi.org/10.1002/ange.201909492openalex-snapshot
Exploiting Imine Photochemistry for Masked N‐Centered Radical Reactivity
inferred← citeshttps://doi.org/10.1002/ange.201912043openalex-snapshot
Enantioenriched Methylene‐Bridged Benzazocanes Synthesis by Organocatalytic and Superacid Activations
inferred← citeshttps://doi.org/10.1002/ange.201912518openalex-snapshot
Direct Catalytic Decarboxylative Amination of Aryl Acetic Acids
inferred← citeshttps://doi.org/10.1002/ange.201914315openalex-snapshot
Rational Design of an Iron‐Based Catalyst for Suzuki–Miyaura Cross‐Couplings Involving Heteroaromatic Boronic Esters and Tertiary Alkyl Electrophiles
inferred← citeshttps://doi.org/10.1002/ange.201915837openalex-snapshot
Polarity Umpolung Strategy for the Radical Alkylation of Alkenes
inferred← citeshttps://doi.org/10.1002/ange.201916015openalex-snapshot
Iridium‐Catalyzed Silylation of Five‐Membered Heteroarenes: High Sterically Derived Selectivity from a Pyridyl‐Imidazoline Ligand
inferred← citeshttps://doi.org/10.1002/ange.202000224openalex-snapshot
Amide Synthesis by Nickel/Photoredox‐Catalyzed Direct Carbamoylation of (Hetero)Aryl Bromides
inferred← citeshttps://doi.org/10.1002/ange.202000887openalex-snapshot
Automated, Accelerated Nanoscale Synthesis of Iminopyrrolidines
inferred← citeshttps://doi.org/10.1002/ange.202001520openalex-snapshot
Iridium‐katalysierte C‐H‐Borylierung von Heteroarenen: Eine Balance zwischen sterischer and elektronischer Regiokontrolle
inferred← citeshttps://doi.org/10.1002/ange.202002271openalex-snapshot
Nickel‐Catalyzed Synthesis of Dialkyl Ketones from the Coupling of N‐Alkyl Pyridinium Salts with Activated Carboxylic Acids
inferred← citeshttps://doi.org/10.1002/ange.202004260openalex-snapshot
Deuteriodifluoromethylation and gem‐Difluoroalkenylation of Aldehydes Using ClCF2H in Continuous Flow
inferred← citeshttps://doi.org/10.1002/ange.202006724openalex-snapshot
Palladium‐Catalyzed Electrophilic Functionalization of Pyridine Derivatives through Phosphonium Salts
inferred← citeshttps://doi.org/10.1002/ange.202007251openalex-snapshot
Copper‐Catalyzed Borylative Couplings with C−N Electrophiles
inferred← citeshttps://doi.org/10.1002/ange.202010631openalex-snapshot
The 2‐Pyridyl Problem: Challenging Nucleophiles in Cross‐Coupling Arylations
inferred← citeshttps://doi.org/10.1002/ange.202012459openalex-snapshot
Chemoselective Amide‐Forming Ligation Between Acylsilanes and Hydroxylamines Under Aqueous Conditions
inferred← citeshttps://doi.org/10.1002/ange.202012496openalex-snapshot
Regioselektiver Brom/Magnesium‐Austausch für die selektive Funktionalisierung von polyhalogenierten Arenen und Heterozyklen
inferred← citeshttps://doi.org/10.1002/ange.202012877openalex-snapshot
Light‐Promoted C–N Coupling of Aryl Halides with Nitroarenes
inferred← citeshttps://doi.org/10.1002/ange.202013089openalex-snapshot
Heterocyclization Reagents for Rapid Assembly of N‐Fused Heteroarenes from Alkenes
inferred← citeshttps://doi.org/10.1002/ange.202013499openalex-snapshot
Highly Robust Iron Catalyst System for Intramolecular C(sp 3 )−H Amidation Leading to γ‐Lactams
inferred← citeshttps://doi.org/10.1002/ange.202014239openalex-snapshot
Modifizierte Enzyme ermöglichen die selektive N‐Alkylierung von Pyrazolen unter Verwendung einfacher Halogenalkane
inferred← citeshttps://doi.org/10.1002/ange.202100949openalex-snapshot
Bimetallic Cooperative Catalysis for Decarbonylative Heteroarylation of Carboxylic Acids via C‐O/C‐H Coupling
inferred← citeshttps://doi.org/10.1002/ange.202103910openalex-snapshot
Enantio‐ und diastereoselektive, vollständige Hydrierung von Benzofuranen mittels Kaskadenkatalyse
inferred← citeshttps://doi.org/10.1002/ange.202106412openalex-snapshot
Direct Amidation of Esters by Ball Milling**
inferred← citeshttps://doi.org/10.1002/ange.202107490openalex-snapshot
Gerüst‐Editierung – Stickstoff‐Deletion sekundärer Amine mithilfe anomerer Amid‐Reagenzien
inferred← citeshttps://doi.org/10.1002/ange.202107820openalex-snapshot
Chemoselective, Scalable Nickel‐Electrocatalytic O‐Arylation of Alcohols
inferred← citeshttps://doi.org/10.1002/ange.202108587openalex-snapshot
Chiral Arylated Amines via C−N Coupling of Chiral Amines with Aryl Bromides Promoted by Light
inferred← citeshttps://doi.org/10.1002/ange.202112454openalex-snapshot
The Formal Cross‐Coupling of Amines and Carboxylic Acids to Form sp3–sp3 Carbon–Carbon Bonds
inferred← citeshttps://doi.org/10.1002/ange.202112668openalex-snapshot
Generation of Oxyphosphonium Ions by Photoredox/Cobaloxime Catalysis for Scalable Amide and Peptide Synthesis in Batch and Continuous‐Flow
inferred← citeshttps://doi.org/10.1002/ange.202114235openalex-snapshot
Strain‐Release‐Driven Friedel–Crafts Spirocyclization of Azabicyclo[1.1.0]butanes
inferred← citeshttps://doi.org/10.1002/ange.202114514openalex-snapshot
Stereodivergent Attached‐Ring Synthesis via Non‐Covalent Interactions: A Short Formal Synthesis of Merrilactone A
inferred← citeshttps://doi.org/10.1002/ange.202115626openalex-snapshot
Nitrogen Atom Transfer Catalysis by Metallonitrene C−H Insertion: Photocatalytic Amidation of Aldehydes
inferred← citeshttps://doi.org/10.1002/ange.202116108openalex-snapshot
Digitizing Chemical Synthesis in 3D Printed Reactionware
inferred← citeshttps://doi.org/10.1002/ange.202117738openalex-snapshot
Acridine‐Functionalized Covalent Organic Frameworks (COFs) as Photocatalysts for Metallaphotocatalytic C−N Cross‐Coupling
inferred← citeshttps://doi.org/10.1002/ange.202200144openalex-snapshot
Chemoselective Transamidation of Thioamides by Transition‐Metal‐Free N−C(S) Transacylation
inferred← citeshttps://doi.org/10.1002/ange.202202794openalex-snapshot
Highly Chemoselective Transamidation of Unactivated Tertiary Amides by Electrophilic N−C(O) Activation by Amide‐to‐Acyl Iodide Re‐routing
inferred← citeshttps://doi.org/10.1002/ange.202204647openalex-snapshot
Maschinelles Lernen zur Vorhersage chemischer Reaktivität: Die Bedeutung “gescheiterter” Experimente
inferred← citeshttps://doi.org/10.1002/ange.202206692openalex-snapshot
Enantioselective Hydrocarbamoylation of Alkenes
inferred← citeshttps://doi.org/10.1002/ange.202207829openalex-snapshot
Visible Light‐Mediated Cyclisation Reaction for the Synthesis of Highly‐Substituted Tetrahydroquinolines and Quinolines
inferred← citeshttps://doi.org/10.1002/ange.202209784openalex-snapshot
ppm Pd‐Containing Nanoparticles as Catalysts for Negishi Couplings … in Water
inferred← citeshttps://doi.org/10.1002/ange.202209882openalex-snapshot
Meerwein‐type Bromoarylation with Arylthianthrenium Salts
inferred← citeshttps://doi.org/10.1002/ange.202210312openalex-snapshot
Dearomative Aminocarbonylation of Arenes via Bifunctional Coordination to Chromium
inferred← citeshttps://doi.org/10.1002/ange.202210525openalex-snapshot
Decarboxylative Sulfinylation Enables a Direct, Metal‐Free Access to Sulfoxides from Carboxylic Acids
inferred← citeshttps://doi.org/10.1002/ange.202211080openalex-snapshot
Directing Group‐Free Formal Suzuki–Miyaura Coupling of Simple Ketones Enabled by Activation of Unstrained C−C Bonds
inferred← citeshttps://doi.org/10.1002/ange.202212873openalex-snapshot
Umpolung Synthesis of Pyridyl Ethers by BiV‐Mediated O‐Arylation of Pyridones
inferred← citeshttps://doi.org/10.1002/ange.202213653openalex-snapshot
Gold(I)‐Catalyzed Benzylic C(sp3)−H Functionalizations: Divergent Synthesis of Indole[a]‐ and [b]‐Fused Polycycles**
inferred← citeshttps://doi.org/10.1002/ange.202215422openalex-snapshot
Dearomatization of Biaryls through Polarity Mismatched Radical Spirocyclization
inferred← citeshttps://doi.org/10.1002/ange.202218565openalex-snapshot
Computational Evolution Of New Catalysts For The Morita–Baylis–Hillman Reaction**
inferred← citeshttps://doi.org/10.1002/ange.202302223openalex-snapshot
A General and Practical Route to Functionalized Bicyclo[1.1.1]Pentane‐Heteroaryls Enabled by Photocatalytic Multicomponent Heteroarylation of [1.1.1]Propellane
inferred← citeshttps://doi.org/10.1002/ange.202302908openalex-snapshot
Catalytic S N Ar Hexafluoroisopropoxylation of Aryl Chlorides and Bromides
inferred← citeshttps://doi.org/10.1002/ange.202306191openalex-snapshot
Photoinduced Electron Transfer from Xanthates to Acyl Azoliums: Divergent Ketone Synthesis via N‐Heterocyclic Carbene Catalysis
inferred← citeshttps://doi.org/10.1002/ange.202306659openalex-snapshot
Anwendungen der C−H‐Aktivierung im präparativen Maßstab in der medizinischen Chemie
inferred← citeshttps://doi.org/10.1002/ange.202307258openalex-snapshot
Design and Application of Peptide‐Mimic Phosphonium Salt Catalysts in Asymmetric Synthesis
inferred← citeshttps://doi.org/10.1002/ange.202309993openalex-snapshot
Regioselective and Enantioselective Copper‐Catalyzed Hydroaminocarbonylation of Unactivated Alkenes and Alkynes
inferred← citeshttps://doi.org/10.1002/ange.202310540openalex-snapshot
Eine photochemische Strategie für die Synthese von ortho‐Aminophenolen durch dearomative‐rearomative Kupplung zwischen Arylaziden und Alkoholen
inferred← citeshttps://doi.org/10.1002/ange.202313717openalex-snapshot
Dual Nickel/Photoredox‐Catalyzed Asymmetric Carbamoylation of Benzylic C(sp3)−H Bonds
inferred← citeshttps://doi.org/10.1002/ange.202313848openalex-snapshot
Phenoxythiazoline (FTz)‐Cobalt(II) Precatalysts Enable C(sp2)–C(sp3) Bond‐Formation for Key Intermediates in the Synthesis of Toll‐like Receptor 7/8 Antagonists**
inferred← citeshttps://doi.org/10.1002/ange.202315108openalex-snapshot
The Construction of Highly Substituted Piperidines via Dearomative Functionalization Reaction
inferred← citeshttps://doi.org/10.1002/ange.202316458openalex-snapshot
Exploring Superacid‐Promoted Skeletal Reorganization of Aliphatic Nitrogen‐Containing Compounds
inferred← citeshttps://doi.org/10.1002/ange.202318304openalex-snapshot
Entschützende Funktionalisierung: eine direkte Umwandlung von Nms‐Amiden in Carbonsäureamide
inferred← citeshttps://doi.org/10.1002/ange.202318676openalex-snapshot
The Future of Chemical Sciences is Sustainable
inferred← citeshttps://doi.org/10.1002/ange.202319758openalex-snapshot
Synthesis of N‐Difluoromethyl Carbonyl Compounds from N‐Difluoromethylcarbamoyl Fluorides
inferred← citeshttps://doi.org/10.1002/ange.202319930openalex-snapshot
Overcoming a Radical Polarity Mismatch in Strain‐Release Pentafluorosulfanylation of [1.1.0]Bicyclobutanes: An Entryway to Sulfone‐ and Carbonyl‐Containing SF5‐Cyclobutanes
inferred← citeshttps://doi.org/10.1002/ange.202400333openalex-snapshot
Room‐Temperature Copper‐Catalyzed Etherification of Aryl Bromides
inferred← citeshttps://doi.org/10.1002/ange.202408419openalex-snapshot
A Rationally Designed Iron(II) Catalyst for C(sp 3 )−C(sp 2 ) and C(sp 3 )−C(sp 3 ) Suzuki–Miyaura Cross‐Coupling
inferred← citeshttps://doi.org/10.1002/ange.202408947openalex-snapshot
P,N‐koordinierende Ylid‐funktionalisierte Phosphane (NYPhos): Eine Ligandenplattform für die selektive Monoarylierung kleiner Nukleophile
inferred← citeshttps://doi.org/10.1002/ange.202411295openalex-snapshot
Rapid Aminations of Functionalized Aryl Fluorosulfates in Water
inferred← citeshttps://doi.org/10.1002/ange.202412247openalex-snapshot
Nickel Catalyzed Carbonylative Cross Coupling for Direct Access to Isotopically Labeled Alkyl Aryl Ketones
inferred← citeshttps://doi.org/10.1002/ange.202417107openalex-snapshot
C−H Alkylation of Heterocycles via Light‐Mediated Palladium Catalysis
inferred← citeshttps://doi.org/10.1002/ange.202417414openalex-snapshot
Fe‐Catalyzed α‐C(sp3)−H Amination of N‐Heterocycles
inferred← citeshttps://doi.org/10.1002/ange.202418367openalex-snapshot
Activation and C−C Coupling of Aryl Iodides via Bismuth Photocatalysis
inferred← citeshttps://doi.org/10.1002/ange.202421258openalex-snapshot
Development and Applications of an Amide Linchpin Reagent
inferred← citeshttps://doi.org/10.1002/ange.202421608openalex-snapshot
Arene Ring Expansion by Ruthenium η 6 ‐Arene Complexes
inferred← citeshttps://doi.org/10.1002/ange.202422185openalex-snapshot
Enzymatic Cascades for Stereoselective and Regioselective Amide Bond Assembly
inferred← citeshttps://doi.org/10.1002/ange.202422742openalex-snapshot
Catalytic Reductive Amination and Tandem Amination–Alkylation of Esters Enabled by a Cationic Iridium Complex
inferred← citeshttps://doi.org/10.1002/ange.202423804openalex-snapshot
Photochemische Permutation von Indazolen zu Benzimidazolen
inferred← citeshttps://doi.org/10.1002/ange.202424051openalex-snapshot
“Naked Nickel”‐Catalyzed Heteroaryl–Heteroaryl Suzuki–Miyaura Coupling
inferred← citeshttps://doi.org/10.1002/ange.202425514openalex-snapshot
Z ‐Selektive organophotochemische Alkinsemireduktion
inferred← citeshttps://doi.org/10.1002/ange.202504750openalex-snapshot
Iron‐Catalyzed Reductive Allylic C─H Amination of Olefin with Nitroarenes via Intermolecular Nitroso Ene Reaction
inferred← citeshttps://doi.org/10.1002/ange.202505984openalex-snapshot
Streamlining SuFEx Inhibitor Development: A Unified Approach Using Photolabile and Orthogonal Sulfinate Protecting Groups
inferred← citeshttps://doi.org/10.1002/ange.202508594openalex-snapshot
Synthesis of a Library of N‐monofluoromethyl Compounds from N‐monofluoromethyl Carbamoyl/Thiocarbamoyl Fluorides
inferred← citeshttps://doi.org/10.1002/ange.202509657openalex-snapshot
Nickel‐Catalyzed Suzuki–Miyaura Cross‐Coupling Reaction of Aliphatic Alcohol Derivatives
inferred← citeshttps://doi.org/10.1002/ange.202510300openalex-snapshot
Biocatalytic Alkylation of Ambident Nucleophiles Enables Selective N ‐Functionalization of Heterocycles and Late‐Stage Modifications
inferred← citeshttps://doi.org/10.1002/ange.202512496openalex-snapshot
General Base‐Free Suzuki‐Miyaura Cross‐Coupling Reaction via Electrophilic Substitution Transmetalation
inferred← citeshttps://doi.org/10.1002/ange.202514741openalex-snapshot
Amine‐Ligated Boryl Radicals Enables Direct C─F Borylation and Cross‐Couplings of Polyfluoroarenes
inferred← citeshttps://doi.org/10.1002/ange.202515469openalex-snapshot
Amide and Thioester Synthesis Via Oxidative Coupling of Alcohols with Amines or Thiols Using Alcohol Dehydrogenases
inferred← citeshttps://doi.org/10.1002/ange.202515595openalex-snapshot
Machine Learning‐Driven Automated Synthesis of Polysubstituted Gentisaldehydes
inferred← citeshttps://doi.org/10.1002/ange.202516584openalex-snapshot
Photoredox/Nickel‐Cocatalyzed Asymmetric C–O and C–S Couplings for Atroposelective Synthesis of N ‐Heterobiaryls
inferred← citeshttps://doi.org/10.1002/ange.202517652openalex-snapshot
Ligand‐Enabled Cu‐Catalyzed Deoxyalkynylation of α‐Unfunctionalized Alcohols with Terminal Alkynes
inferred← citeshttps://doi.org/10.1002/ange.202518260openalex-snapshot
Aminative Suzuki–Miyaura Coupling: Tackling Alkyl Nucleophiles and Addressing the Viability of the Electrophile‐First Mechanism
inferred← citeshttps://doi.org/10.1002/ange.202520677openalex-snapshot
Frame‐Shifted Synthesis of Oligoheterocycles as a Platform for Molecular Design
inferred← citeshttps://doi.org/10.1002/ange.202520841openalex-snapshot
Electrochemical Azolation of Electron‐rich Fluoroarenes: A Controlled Redox Chain Unlocks C─N Bond‐forming e ‐S N Ar
inferred← citeshttps://doi.org/10.1002/ange.202521490openalex-snapshot
Engaging Tertiary Benzylic Radicals in Metallaphotoredox Catalysis: A Modular Approach to Access Diaryl Quaternary Centers
inferred← citeshttps://doi.org/10.1002/ange.202521633openalex-snapshot
Novel Sulfonium Reagents for the Modular Synthesis of Spiro[2.3]Hexanes and Heteroatom‐Containing Analogues: Synthesis, Application, and Evaluation as Bioisosteres
inferred← citeshttps://doi.org/10.1002/ange.202524431openalex-snapshot
A Radical Cascade with Double Intramolecular Hydrogen Atom Transfer for the Generation of Bisfunctionalized Cyclopentanes from Linear Alkynes
inferred← citeshttps://doi.org/10.1002/ange.5407928openalex-snapshot
Electrochemical Desilylative Fluorination Enables Access to N ‐Monofluoromethyl Amides and Peptides
inferred← citeshttps://doi.org/10.1002/ange.6908076openalex-snapshot
Photoinduced Copper‐Catalyzed Stereoselective C(sp 3 )‐H Amination Enabled by Preorganized Multiple Noncovalent Interactions
inferred← citeshttps://doi.org/10.1002/ange.6992524openalex-snapshot
Deaminative Allylation of Primary Amines
inferred← citeshttps://doi.org/10.1002/ange.8290035openalex-snapshot
Synthesis of Large‐ and Medium‐Sized Heterobiaryl Atropisomeric Rings and Atropopeptides by Catalytic Intramolecular S N Ar
inferred← citeshttps://doi.org/10.1002/ange.9109858openalex-snapshot
Remapping the Synthetic Landscape of α‐Tertiary Alkylamines via Dual‐Functional Catechol
inferred← citeshttps://doi.org/10.1002/ange.9297515openalex-snapshot
Sustainable Pd‐Catalyzed Aminations “on Dirty Water”
inferred← citeshttps://doi.org/10.1002/anie.1441281openalex-snapshot
Ligand‐Enabled Stereoselective Coupling of Methylene C(sp 3 )─H Bonds With Alkenyl Bromide via Pd II /Pd 0 /Pd II Catalysis
inferred← citeshttps://doi.org/10.1002/anie.1983055openalex-snapshot
Gold Single‐Atom Catalysts Enable Selective Shuttle Hydrochlorination of Alkynes
inferred← citeshttps://doi.org/10.1002/anie.201604193openalex-snapshot
Evaluating New Chemistry to Drive Molecular Discovery: Fit for Purpose?
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