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Chromone as a Privileged Scaffold in Drug Discovery: Recent Advances

https://doi.org/10.1021/acs.jmedchem.6b01720

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Outgoing claims: the papers this work cites, builds on, or argues with.

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Organocatalytic oxa‐Michael/Michael Addition/Deformylation Cascade Reaction of 3‐Formylchromone with p‐Quinol: Synthesis of the Furanochromanone Skeleton

inferred← citeshttps://doi.org/10.1002/adsc.202201154openalex-snapshot

Synthesis of Functionalized 3‐(1H‐Isochromen)‐chromones via Ag2O‐Catalyzed Cascade Cyclization Reaction of o‐Hydroxyarylenaminones with o‐Alkynylbenzaldehydes

inferred← citeshttps://doi.org/10.1002/adsc.202201410openalex-snapshot

Martin Silicates as Partners in Photoredox/Ni Dual Catalysis for the Installation of CH3, CH2D, CD2H, CD3 and 13CH3 Groups onto (Hetero)Arenes

inferred← citeshttps://doi.org/10.1002/adsc.202300207openalex-snapshot

(CF3CO)2O/K2CO3‐Mediated Synthesis of 3‐Sulfonylchromones through Cyclocondensation of β‐Ketosulfones and Carboxylic Acids

inferred← citeshttps://doi.org/10.1002/adsc.202300260openalex-snapshot

Mechanochemical Defluorinative Acylation of ortho‐Hydroxyarylenaminones by CF3‐Compounds: Synthesis of 3‐Acylchromones

inferred← citeshttps://doi.org/10.1002/adsc.202300512openalex-snapshot

Solvent‐Regulated Electrochemical Selenylation and Deuteration of Alkynyl Aryl Ketones: Chemoselective Synthesis of 3‐Selenylated Chromones and Deutero‐Selenylated Chalcones

inferred← citeshttps://doi.org/10.1002/adsc.202301152openalex-snapshot

One‐Pot Access to 3‐Sulfonyl Flavones via K2CO3‐Mediated Annulation of α‐Sulfonyl o‐Hydroxyacetophenones with Substituted Nitriles

inferred← citeshttps://doi.org/10.1002/adsc.202400093openalex-snapshot

Silver‐catalyzed Cascade Bis‐heteroannulation Reaction of Enynones and o‐Hydroxyphenyl Enaminones: Access to Highly Functionalized 3‐Furylmethyl Chromones

inferred← citeshttps://doi.org/10.1002/adsc.202401396openalex-snapshot

Organic Photoredox Catalytic Sulfonylation of Enaminones to Access 3‐Sulfonyl Chromones

inferred← citeshttps://doi.org/10.1002/adsc.202500172openalex-snapshot

AgNO 3 ‐Catalyzed Regio‐selective Bis‐heteroannulation of o ‐Hydroxyphenyl Enaminones and Yne‐enones: A Facile synthesis of Functionalized 3‐(Furan‐3‐ylmethyl) Chromones

inferred← citeshttps://doi.org/10.1002/adsc.70260openalex-snapshot

Switchable Divergent Synthesis of 3‐Dithiocarbamyl and 3‐Carbamothioyl Chromones Through Chromone Annulation Reactions of o ‐Hydroxyenaminones With CS 2

inferred← citeshttps://doi.org/10.1002/advs.202415795openalex-snapshot

Copper‐Catalyzed Carbonylative Cyclization of CO 2 : A Promising Approach for Synthesis of Flavone

inferred← citeshttps://doi.org/10.1002/aic.17748openalex-snapshot

De novo drug design framework based on mathematical programming method and deep learning model

inferred← citeshttps://doi.org/10.1002/ajoc.201800128openalex-snapshot

Site‐Selective C−H Bond Functionalization of Chromones and Coumarins

inferred← citeshttps://doi.org/10.1002/ajoc.202000714openalex-snapshot

Palladium‐Catalyzed Allylic Cycloaddition of Vinylethylene Carbonates with 3‐Nitrochromone

inferred← citeshttps://doi.org/10.1002/ajoc.202100694openalex-snapshot

Tetramethylammonium Iodide (TMAI)‐Promoted Sulfenylation/Annulation of Enaminones with Thiosulfonates

inferred← citeshttps://doi.org/10.1002/ajoc.202300499openalex-snapshot

I2/PPh3‐Mediated Cyclization of Enaminones with Sodium Sulfinates: A Protocol for the Synthesis of 3‐Thiolated Chromones

inferred← citeshttps://doi.org/10.1002/ajoc.202400391openalex-snapshot

Divergent Sc(OTf)3‐Catalyzed Tandem Cyclization of o‐Hydroxyphenyl Enaminones with 1,3,5‐Triazinanes: Access to C3‐Aminomethyl Chromones and Tetrahydropyrimidines

inferred← citeshttps://doi.org/10.1002/ajoc.70254openalex-snapshot

Intermolecular Friedel–Crafts Acylation/Cyclization Reaction of 2‐Methoxybenzoyl Chlorides with 1‐Haloalkynes for the Synthesis of 3‐Halo(thio)Chromenones

inferred← citeshttps://doi.org/10.1002/ange.201806729openalex-snapshot

Enzymology of Anthraquinone‐γ‐Pyrone Ring Formation in Complex Aromatic Polyketide Biosynthesis

inferred← citeshttps://doi.org/10.1002/ange.202310115openalex-snapshot

Precise Recognition in Water by an Endo‐Functionalized Cavity: Tuning the Complementarity of Binding Sites

inferred← citeshttps://doi.org/10.1002/ange.202508335openalex-snapshot

Ternary Aldehyde–Copper–Iridium Catalysis Enables Stereodivergent Allylation via α‐C‐H Functionalization of Primary Amines

inferred← citeshttps://doi.org/10.1002/anie.201806729openalex-snapshot

Enzymology of Anthraquinone‐γ‐Pyrone Ring Formation in Complex Aromatic Polyketide Biosynthesis

inferred← citeshttps://doi.org/10.1002/anie.202310115openalex-snapshot

Precise Recognition in Water by an Endo‐Functionalized Cavity: Tuning the Complementarity of Binding Sites

inferred← citeshttps://doi.org/10.1002/anie.202508335openalex-snapshot

Ternary Aldehyde–Copper–Iridium Catalysis Enables Stereodivergent Allylation via α‐C‐H Functionalization of Primary Amines

inferred← citeshttps://doi.org/10.1002/aoc.70095openalex-snapshot

DNA Binding Affinities and Antimicrobial Activities of Pd(II) Complexes of Chromone Schiff Bases

inferred← citeshttps://doi.org/10.1002/aoc.7192openalex-snapshot

Dual function of new Nd(III) and Gd(III) complexes for cytotoxic and optoelectronic fields: Synthesis, characterization, DFT calculations, and PVA composite films

inferred← citeshttps://doi.org/10.1002/ardp.70224openalex-snapshot

Chromones as Nonclassical Inhibitors of Carbonic Anhydrase IX and XII Isoforms: Probing Chromone‐Based Derivatives

inferred← citeshttps://doi.org/10.1002/asia.202500153openalex-snapshot

The Application of N‐Aryl Glycines and Their Analogues in Visible‐Light‐Promoted Photoredox Catalysis

inferred← citeshttps://doi.org/10.1002/cbdv.202300251openalex-snapshot

Selective Induction of DNA Damage and Cell Cycle Arrest Mediated by Chromone‐Triazole Dyads Derivatives: Effects on Breast and Prostate Cancer Cells

inferred← citeshttps://doi.org/10.1002/chem.202500283openalex-snapshot

Visible‐Light Photocatalysis for Sustainable Chromene Synthesis and Functionalization

inferred← citeshttps://doi.org/10.1002/cjoc.70466openalex-snapshot

Diastereodivergent Asymmetric [3+2] Cyclization of Chromone Derivatives with γ ‐Hydroxyenones †

inferred← citeshttps://doi.org/10.1002/cmdc.202500447openalex-snapshot

Recent Insights in Multi‐Target Drugs in Pharmacology and Medicinal Chemistry

inferred← citeshttps://doi.org/10.1002/cnma.202300641openalex-snapshot

Visible Light Mediated Synthesis of 3‐Indolmethyl Chromones via the Cyclization of o‐Hydroxyaryl Enaminones with 3‐Indoleacetic Acids Catalyzed by Graphitic Carbon Nitride Adorned with Copper Nanoparticles

inferred← citeshttps://doi.org/10.1002/ejoc.201801159openalex-snapshot

Synthesis of Chromone‐Containing Allylmorpholines through a Morita–Baylis–Hillman‐Type Reaction

inferred← citeshttps://doi.org/10.1002/ejoc.201801231openalex-snapshot

New Entries to 3‐Acylchromones: TM‐Catalysed Decarboxylative Cross‐Coupling of α‐Keto Acids with ortho‐Hydroxyarylenaminones, 2,3‐Unsubstituted Chromones and 3‐Iodochromones

inferred← citeshttps://doi.org/10.1002/ejoc.201900519openalex-snapshot

Electroreductive Intermolecular Coupling of Chromones with Benzophenones: Synthesis of 2‐Diarylmethylchromones and Tetrasubstituted Furans

inferred← citeshttps://doi.org/10.1002/ejoc.201901636openalex-snapshot

One‐Step Synthesis of Trifluoroethylated Chromones via Radical Cascade Cyclization–Coupling of 2‐(Allyloxy)arylaldehydes

inferred← citeshttps://doi.org/10.1002/ejoc.202100213openalex-snapshot

Selective Synthesis of 5‐Alkylated and 5‐Alkenylated Chromones via Catalytic C‐H Coupling of Chromones with Allyl Alcohols

inferred← citeshttps://doi.org/10.1002/ejoc.202300456openalex-snapshot

Base‐Promoted Difunctionalization of Alkynes: One‐Pot Synthesis of Polysubstituted Chromones

inferred← citeshttps://doi.org/10.1002/ejoc.202400401openalex-snapshot

Electrochemical Decarboxylative Addition of N‐Aryl Glycines to Enaminones: Access to C3‐Aminomethyl Chromones

inferred← citeshttps://doi.org/10.1002/ejoc.202401061openalex-snapshot

Tetrasubstituted Chromanone Synthesis by a Tandem Oxa‐Michael/Michael Addition Reaction of 2‐Hydroxyacetophenones and Alkynyl Nitriles

inferred← citeshttps://doi.org/10.1002/ejoc.202401247openalex-snapshot

Synthesis of Enantioenriched 2‐((Hetera)Cyclo) Alkylchromanols and their Spirocyclic Analogs through Enzymatic Resolution

inferred← citeshttps://doi.org/10.1002/ejoc.202500107openalex-snapshot

Pd‐catalyzed CH Activation and Oxidative Annulation to Access N‐methoxy‐7H‐Chromenoquinolinones and N‐methoxyphenyl quinolinones

inferred← citeshttps://doi.org/10.1002/ejoc.202500167openalex-snapshot

Recent Advances of Enaminones in Multi‐component Reactions: A Brief Review

inferred← citeshttps://doi.org/10.1002/jhet.3894openalex-snapshot

Synthesis and characterization of novel 2‐(1‐benzyl‐3‐[4‐fluorophenyl]‐1H‐pyrazol‐4‐yl)‐7‐fluoro‐4H‐chromen‐4‐one derivatives

inferred← citeshttps://doi.org/10.1002/jhet.70156openalex-snapshot

Utility of 3‐Formylchromone in the Synthesis of Polyfunctional Nitrogenous Hybrids: Empowered by Anticancer Efficiency and Molecular Simulations

inferred← citeshttps://doi.org/10.1002/jms.4305openalex-snapshot

Gas phase reaction between chromones and solvent in an electrospray ionization source

inferred← citeshttps://doi.org/10.1002/ppsc.201900083openalex-snapshot

Harnessing Calcium‐Oxalate‐ (CaOx‐) Nanocrystal‐Induced Prodeath Autophagy for Attenuating Human Renal Proximal Tubular Epithelial Cell Injury

inferred← citeshttps://doi.org/10.1002/ptr.6419openalex-snapshot

Polyphenols: A concise overview on the chemistry, occurrence, and human health

inferred← citeshttps://doi.org/10.1002/rcm.8567openalex-snapshot

Formation of molecular oxygen‐ and water‐attached fragment ions in the fragmentation of protonated 3‐(phenylthio)chromones

inferred← citeshttps://doi.org/10.1002/slct.201800613openalex-snapshot

Synthesis of Novel Thiophene‐Chalcone Derivatives as Anticancer‐ and Apoptosis‐Inducing Agents

inferred← citeshttps://doi.org/10.1002/slct.201900009openalex-snapshot

Synthesis of a New Series of Furopyranone‐ and Furocoumarin‐Chromone Conjugates Followed by In–Vitro Cytotoxicity Activity Evaluation, and Molecular Docking Study

inferred← citeshttps://doi.org/10.1002/slct.201903001openalex-snapshot

Catalytic Efficiency of Biosynthesized Silver Nanoparticles in Synthesis of Chromones and Reduction of Nitro Aromatics

inferred← citeshttps://doi.org/10.1002/slct.202001749openalex-snapshot

Peroxy‐Benzoic Acid Mediated Domino C[sp 2 ] Hydroxylation /Annulation of Enaminones for the Synthesis of 3‐Hydroxy Chromones

inferred← citeshttps://doi.org/10.1002/slct.202003553openalex-snapshot

A Convenient Synthesis of Iguratimod‐Amine Precursor via NHC‐Catalyzed Aldehyde‐Nitrile Cross Coupling Reaction

inferred← citeshttps://doi.org/10.1002/slct.202104360openalex-snapshot

Solvent‐Free Microwave‐Assisted Multicomponent Synthesis of 4 H ‐Chromenes Using Fe 3 O 4 ‐Based Hydrotalcites as Bifunctional Catalysts

inferred← citeshttps://doi.org/10.1002/slct.202203340openalex-snapshot

Synthesis of Chromone‐Spiroindolinone‐Cyclopentene Derivatives through Phosphine‐Catalyzed (3+2) Annulation of Morita‐Baylis‐Hillman Carbonates with Oxindole‐Chromones

inferred← citeshttps://doi.org/10.1002/slct.202401465openalex-snapshot

Bifunctional Squaramide‐Catalyzed Asymmetric Michael/Cyclization Reactions of 3‐Hydroxychromenones with Isatylidenemalononitriles

inferred← citeshttps://doi.org/10.1002/slct.202405579openalex-snapshot

I 2 ‐Promoted Alkylsulfenylation/Cyclization of Enaminones with S ‐Alkyl Bunte Salts: Synthesis of 3‐Alkylsulfenylated Chromones

inferred← citeshttps://doi.org/10.1002/slct.73878openalex-snapshot

Enantioselective Mannich Reaction of 2‐Aminochromones With Isatin‐Derived N ‐Boc Ketimines

inferred← citeshttps://doi.org/10.1002/tcr.202500073openalex-snapshot

Harnessing Chromone as a Versatile Scaffold for Emerging Biological Applications: Recent Advances and Medicinal Insights

inferred← citeshttps://doi.org/10.1007/978-981-19-9605-4_10openalex-snapshot

Therapeutic Potential of Benzopyrones Against Antiparasitic Diseases

inferred← citeshttps://doi.org/10.1007/s00044-019-02320-wopenalex-snapshot

Synthesis and biological evaluation of novel chromonyl enaminones as α-glucosidase inhibitors

inferred← citeshttps://doi.org/10.1007/s00706-019-02512-5openalex-snapshot

Synthesis and structural study of 2-(haloalkyl)-3-methylchromones

inferred← citeshttps://doi.org/10.1007/s00894-021-04800-6openalex-snapshot

Modeling the structural and reactivity properties of hydrazono methyl-4H-chromen-4-one derivatives—wavefunction-dependent properties, molecular docking, and dynamics simulation studies

inferred← citeshttps://doi.org/10.1007/s00894-026-06887-1openalex-snapshot

Organometallic-enhanced chromone-thiazole hybrid antioxidants: a DFT study of solvent-dependent HAT/SPLET switching

inferred← citeshttps://doi.org/10.1007/s10593-022-03058-xopenalex-snapshot

Unexpected conversion of 4-oxo-4H-chromene-2-carboxylic acid to 2-(1,3-benzothiazol-2-yl)-4H-chromen-4-one and spiro[1,4-benzothiazine-2,2'-chromene]-3,4'(3'H,4H)-dione

inferred← citeshttps://doi.org/10.1007/s10593-023-03219-6openalex-snapshot

Expanding the isoflavone, pyrazole, and oxazole chemical space through 2'-carboxamido-2-hydroxydeoxybenzoin precursors

inferred← citeshttps://doi.org/10.1007/s10593-023-03221-yopenalex-snapshot

Parent 5(7)-azachromones and their partially hydrogenated derivatives: synthesis and physicochemical properties

inferred← citeshttps://doi.org/10.1007/s10593-024-03357-5openalex-snapshot

Progress in the synthesis of 3-fluorochromones (microreview)

inferred← citeshttps://doi.org/10.1007/s10593-025-03406-7openalex-snapshot

Perspective on Biginelli reaction: en route toward the development of biologically and industrially relevant dihydropyrimidone-based frameworks

inferred← citeshttps://doi.org/10.1007/s11030-021-10234-2openalex-snapshot

Rapid synthetic approaches to libraries of diversified 1,2-dihydrochromeno[2,3-c]pyrrole-3,9-diones and 3-(2-hydroxyphenyl)-4,5-dihydropyrrolo[3,4-c]pyrazol-6(1H)-ones

inferred← citeshttps://doi.org/10.1007/s11030-024-11027-zopenalex-snapshot

HFIP-driven Schmidt-type reaction enables chromone-3-carbonitriles and its applications

inferred← citeshttps://doi.org/10.1007/s11030-025-11284-6openalex-snapshot

Synthesis and multi-target evaluation of 2-(2-phenylethyl)/2,3-styrylchromone derivatives as potential anti-Alzheimer’s disease agents

inferred← citeshttps://doi.org/10.1007/s11094-024-03245-4openalex-snapshot

Design, Creation, and Biological Screening of Newer Coumarin-Coupled Heterocyclic Hybrids as Acetylcholinesterase Inhibitors that may be Useful in the Treatment of Alzheimer’s Disease

inferred← citeshttps://doi.org/10.1007/s11172-022-3658-0openalex-snapshot

Synthesis of 2,3-heterofused chromones, hetero analogues of xanthone

inferred← citeshttps://doi.org/10.1007/s12039-026-02484-0openalex-snapshot

A novel synthesis of C3-carbonylated imidazopyridines by the ring opening and closing cascade (ROCC) mechanism

inferred← citeshttps://doi.org/10.1007/s40199-020-00378-1openalex-snapshot

Chromone–lipoic acid conjugate: Neuroprotective agent having acceptable butyrylcholinesterase inhibition, antioxidant and copper-chelation activities

inferred← citeshttps://doi.org/10.1007/s42250-025-01416-8openalex-snapshot

Coumarin-Indole-Triazole Hybrids: Synthesis, Antimicrobial Evaluation, DFT Insights, Molecular Docking, and Dynamics as Potential Antibacterial Agents

inferred← citeshttps://doi.org/10.1007/s42452-021-04188-1openalex-snapshot

Spectroscopic and computational study of chromone derivatives with antitumor activity: detailed DFT, QTAIM and docking investigations

inferred← citeshttps://doi.org/10.1007/s43630-025-00797-6openalex-snapshot

Photochemical access to flavone- and aurone-fused estrone derivatives

inferred← citeshttps://doi.org/10.1016/b978-0-12-816125-8.00013-4openalex-snapshot

Analysis of Chemical Spaces: Implications for Drug Repurposing

inferred← citeshttps://doi.org/10.1016/b978-0-12-820586-0.00013-3openalex-snapshot

Synthesis of biologically relevant heterocyclic skeletons under solvent-free condition

inferred← citeshttps://doi.org/10.1016/b978-0-323-95893-6.00004-9openalex-snapshot

Visible light–driven organic synthesis under iridium (IrIII)-complex photocatalysis

inferred← citeshttps://doi.org/10.1016/b978-0-443-18611-0.00020-6openalex-snapshot

Privileged scaffolds in anti-diabetic drug discovery

inferred← citeshttps://doi.org/10.1016/bs.aihch.2019.01.003openalex-snapshot

The literature of heterocyclic chemistry, part XVII, 2017

inferred← citeshttps://doi.org/10.1016/j.apsb.2021.09.027openalex-snapshot

Free energy perturbation (FEP)-guided scaffold hopping

inferred← citeshttps://doi.org/10.1016/j.bcp.2025.116806openalex-snapshot

Discovery of a novel C2-functionalized chromen-4-one scaffold for the development of p38α MAPK signaling inhibitors to mitigate neutrophilic inflammatory responses

inferred← citeshttps://doi.org/10.1016/j.bioorg.2019.03.042openalex-snapshot

Design, synthesis and evaluation of 2-(indolylmethylidene)-2,3-dihydro-1-benzofuran-3-one and 2-(indolyl)-4H-chromen-4-one derivatives as novel monoamine oxidases inhibitors

inferred← citeshttps://doi.org/10.1016/j.bioorg.2019.103285openalex-snapshot

2-Styrylchromone derivatives as potent and selective monoamine oxidase B inhibitors

inferred← citeshttps://doi.org/10.1016/j.bioorg.2021.104750openalex-snapshot

Chromone derivatives bearing pyridinium moiety as multi-target-directed ligands against Alzheimer’s disease

inferred← citeshttps://doi.org/10.1016/j.bioorg.2022.106049openalex-snapshot

Design, synthesis and biological evaluation of novel chromone-maleimide hybrids as potent anti-inflammatory agents against LPS-induced acute lung injury

inferred← citeshttps://doi.org/10.1016/j.bioorg.2024.107865openalex-snapshot

Chromene-based compounds as drug candidates for renal and bladder cancer therapy – A systematic review

inferred← citeshttps://doi.org/10.1016/j.bioorg.2025.109350openalex-snapshot

Design, synthesis, and multi-target evaluation of Chromone-based derivatives as promising anti-Alzheimer's disease agents

inferred← citeshttps://doi.org/10.1016/j.bioorg.2026.109564openalex-snapshot

Design-led synthesis and multidimensional evaluation of novel thiadiazoles as multitarget anti-Alzheimer agents: kinetics, DFT and in silico mapping

inferred← citeshttps://doi.org/10.1016/j.bmc.2018.08.010openalex-snapshot

Synthesis, molecular docking, and biological activity of 2-vinyl chromones: Toward selective butyrylcholinesterase inhibitors for potential Alzheimer's disease therapeutics

inferred← citeshttps://doi.org/10.1016/j.bmc.2021.116255openalex-snapshot

Synthesis and biological evaluation of 3-styrylchromone derivatives as selective monoamine oxidase B inhibitors

inferred← citeshttps://doi.org/10.1016/j.bmcl.2019.126945openalex-snapshot

Design, synthesis and anti-TMV activities of novel chromone derivatives containing dithioacetal moiety

inferred← citeshttps://doi.org/10.1016/j.cclet.2021.03.071openalex-snapshot

Selective detection of Zn2+ and Cd2+ ions in water using a host-guest complex between chromone and Q[7]

inferred← citeshttps://doi.org/10.1016/j.cclet.2024.110474openalex-snapshot

Forging of silaoxycarbocyclics by interrupted Catellani reaction

inferred← citeshttps://doi.org/10.1016/j.cclet.2024.110784openalex-snapshot

An update on the advances in chromone and the derivatives synthesis based on the key chromone annulation of o-hydroxyaryl enaminones

inferred← citeshttps://doi.org/10.1016/j.ccr.2018.04.008openalex-snapshot

Recent developments in the chemistry of ferrocenyl secondary natural product conjugates

inferred← citeshttps://doi.org/10.1016/j.ccr.2025.217231openalex-snapshot

O-aminobenzamide: An increasingly popular privileged scaffold in drug discovery

inferred← citeshttps://doi.org/10.1016/j.ccr.2026.218084openalex-snapshot

Natural product-conjugated gold(I) complexes: Coordination chemistry and biomedical applications

inferred← citeshttps://doi.org/10.1016/j.chemphys.2018.09.042openalex-snapshot

Specific solvent effect on the photophysical behavior of substituted chromones: A combined fluorescence, DFT and MD study

inferred← citeshttps://doi.org/10.1016/j.dyepig.2026.113952openalex-snapshot

Recent progress in thiol-chromene click regulated functional molecules

inferred← citeshttps://doi.org/10.1016/j.ejmech.2018.01.074openalex-snapshot

The lead optimization of the polyamine conjugate of flavonoid with a naphthalene motif: Synthesis and biological evaluation

inferred← citeshttps://doi.org/10.1016/j.ejmech.2018.07.056openalex-snapshot

Multi-target-directed ligands for Alzheimer's disease: Discovery of chromone-based monoamine oxidase/cholinesterase inhibitors

inferred← citeshttps://doi.org/10.1016/j.ejmech.2018.07.058openalex-snapshot

Exploitation of new chalcones and 4H-chromenes as agents for cancer treatment

inferred← citeshttps://doi.org/10.1016/j.ejmech.2019.04.025openalex-snapshot

Synthetic heterocyclic candidates as promising α-glucosidase inhibitors: An overview

inferred← citeshttps://doi.org/10.1016/j.ejmech.2019.111772openalex-snapshot

Optimization of the chromone scaffold through QSAR and docking studies: Identification of potent inhibitors of ABCG2

inferred← citeshttps://doi.org/10.1016/j.ejmech.2020.112503openalex-snapshot

Chromones bearing amino acid residues: Easily accessible and potent inhibitors of the breast cancer resistance protein ABCG2

inferred← citeshttps://doi.org/10.1016/j.ejmech.2020.112787openalex-snapshot

A comprehensive review of monoamine oxidase inhibitors as Anti-Alzheimer’s disease agents: A review

inferred← citeshttps://doi.org/10.1016/j.ejmech.2020.112958openalex-snapshot

Water-soluble inhibitors of ABCG2 (BCRP) – A fragment-based and computational approach

inferred← citeshttps://doi.org/10.1016/j.ejmech.2022.114507openalex-snapshot

Design and synthesis of chromone-based monoamine oxidase B inhibitors with improved drug-like properties

inferred← citeshttps://doi.org/10.1016/j.ejmech.2023.115308openalex-snapshot

Design, synthesis and evaluation of novel monoamine oxidase B (MAO-B) inhibitors with improved pharmacokinetic properties for Parkinson's disease

inferred← citeshttps://doi.org/10.1016/j.ejmech.2023.115944openalex-snapshot

Discovery of potent chromone-based autotaxin inhibitors inspired by cannabinoids

inferred← citeshttps://doi.org/10.1016/j.ejmech.2024.116759openalex-snapshot

A comprehensive review of new small molecule drugs approved by the FDA in 2022: Advance and prospect

inferred← citeshttps://doi.org/10.1016/j.ejmech.2025.117978openalex-snapshot

Harnessing cell cycle intervention and evading P-glycoprotein efflux: natural product-inspired C2-aminophenyl chromones as dual modulators against multidrug-resistant cancer

inferred← citeshttps://doi.org/10.1016/j.ejmech.2026.118701openalex-snapshot

Multi-target-directed chromone–carboxamide hybrids: Potent AChE/MAO-B inhibitors with anti-Aβ/Tau and neuroprotective activities

inferred← citeshttps://doi.org/10.1016/j.ejmech.2026.119219openalex-snapshot

Discovery of chromone-derived EGFR inhibitors as potent apoptosis inducers in cancer: In vitro and in vivo insights

inferred← citeshttps://doi.org/10.1016/j.fitote.2021.105004openalex-snapshot

A new antibacterial chromone from a marine sponge-associated fungus Aspergillus sp. LS57

inferred← citeshttps://doi.org/10.1016/j.gresc.2022.05.002openalex-snapshot

Multicomponent cascade reaction of 3-formylchromones: Highly regioselective synthesis of functionalized pyridin-2(1H)-ones

inferred← citeshttps://doi.org/10.1016/j.gresc.2022.10.003openalex-snapshot

Cascade reaction of 3-formylchromones: Highly selective synthesis of 4-oxo-3-(1H-pyrrol-3-yl)-4H-chromenes

inferred← citeshttps://doi.org/10.1016/j.gresc.2022.10.014openalex-snapshot

Highly selective synthesis of functionalized morphan derivatives through a multi-component cascade reaction of 3-formylchromones, 2-naphthols, and enaminones

inferred← citeshttps://doi.org/10.1016/j.inoche.2022.110026openalex-snapshot

Binding interactions and sensing applications of chromone derived Schiff base chemosensors via absorption and emission studies: A comprehensive review

inferred← citeshttps://doi.org/10.1016/j.jare.2023.06.014openalex-snapshot

Synergistic effect of cold gas plasma and experimental drug exposure exhibits skin cancer toxicity in vitro and in vivo

inferred← citeshttps://doi.org/10.1016/j.jcat.2025.115993openalex-snapshot

Palladium-catalyzed carbonylative synthesis of 13C-labeled flavones

inferred← citeshttps://doi.org/10.1016/j.jfluchem.2019.109354openalex-snapshot

Transformations of 3-acyl-4H-polyfluorochromen-4-ones under the action of amino acids and biogenic amines

inferred← citeshttps://doi.org/10.1016/j.jfluchem.2020.109717openalex-snapshot

Synthesis, experimental and theoretical study of novel 2-haloalkyl (-CF2H, -CCl2H, -CF2CF3)-, 3-bromo and bromomethyl substituted chromones

inferred← citeshttps://doi.org/10.1016/j.jfluchem.2025.110421openalex-snapshot

Synthesis of fluorinated 4H-chromen-4-ones from 2-hydroxyacetophenones and in vitro evaluation of their anticancer and antiviral activity

inferred← citeshttps://doi.org/10.1016/j.mcat.2022.112320openalex-snapshot

Palladium-catalyzed norbornene-mediated dehydrogenative annulation of 3-iodochromones with trifluoroacetimidoyl chlorides for the construction of trifluoromethyl-substituted chromeno[2,3-c]quinolin-12-ones

inferred← citeshttps://doi.org/10.1016/j.mcat.2024.114443openalex-snapshot

Photocatalytic radical-promoted cyclization of thiomethyl ynones with aldehydes: synthesis of thiochromones

inferred← citeshttps://doi.org/10.1016/j.mencom.2019.03.041openalex-snapshot

Reactions of carbamoylated amino enones with 3-substituted chromones for the preparation of 2-pyridones and chromeno[4,3-b]pyridine-2,5-diones

inferred← citeshttps://doi.org/10.1016/j.microc.2025.113984openalex-snapshot

A reversible fluorescent probe for monitoring sulfur dioxide and formaldehyde in real samples and living cells

inferred← citeshttps://doi.org/10.1016/j.molliq.2025.129019openalex-snapshot

Exploring the anticancer potential of chromene-based thiosemicarbazones through in vitro, molecular docking, molecular dynamics simulation and DFT studies

inferred← citeshttps://doi.org/10.1016/j.molstruc.2021.130618openalex-snapshot

Coumarin linked heterocyclic hybrids: A promising approach to develop multi target drugs for Alzheimer's disease

inferred← citeshttps://doi.org/10.1016/j.molstruc.2021.130706openalex-snapshot

Synthesis, structural characterization, antioxidant and cytotoxic activity towards human cancer cell lines and computational studies of new Ni(II), Co(II) and Pd(II) complexes with 3-[bis(3,5-dimethylpyrazol-1-yl)methyl]chromen-4-one derivatives

inferred← citeshttps://doi.org/10.1016/j.molstruc.2021.131683openalex-snapshot

Synthesis, cytotoxic and antioxidant activities of new n-substituted 3-(benzimidazol-2-yl)-chromones containing 2,6-di-tert-butylphenol fragment

inferred← citeshttps://doi.org/10.1016/j.molstruc.2022.132533openalex-snapshot

A chromone-based colorimetric fluorescence sensor for selective detection of Cu2+ions, and its application for in-situ imaging

inferred← citeshttps://doi.org/10.1016/j.molstruc.2022.133972openalex-snapshot

Theoretical vibrational spectroscopy (FT-IR), PED and DFT calculations of chromones and thiochromones

inferred← citeshttps://doi.org/10.1016/j.molstruc.2023.136205openalex-snapshot

Design, synthesis, in-vitro and in-silico studies of chromone‐isoxazoline conjugates as anti‐bacterial agents

inferred← citeshttps://doi.org/10.1016/j.molstruc.2023.137452openalex-snapshot

Spectroscopic (FT-IR, FT-Raman, NMR and UV–vis), quantum calculation, molecular structure, solvent interaction, ADME and molecular docking investigation on 4-oxo-4h-1-benzopyran-2-carboxylic acid

inferred← citeshttps://doi.org/10.1016/j.molstruc.2024.140739openalex-snapshot

Synthesis, crystal structure, spectroscopic characterization, DFT calculations, Hirshfeld surface analysis, biological activity studies, molecular docking investigation, and ADMET properties evaluation of a novel 3-substituted coumarin derivative

inferred← citeshttps://doi.org/10.1016/j.molstruc.2024.140972openalex-snapshot

Design, synthesis and characterization of new amide-linked Chromone-Isoxazole Hybrids: In Vitro anti-bacterial and antioxidant evaluation, DFT calculations, ADMET profiling, docking and molecular dynamics simulation

inferred← citeshttps://doi.org/10.1016/j.molstruc.2025.141990openalex-snapshot

Molecular structure, spectroscopy, reactivity and biological activity: A collection of selected communications based on thiadiazole linked benzamide derivatives

inferred← citeshttps://doi.org/10.1016/j.molstruc.2025.144474openalex-snapshot

Synthesis of spiropyrrolidine oxindoles from isatin-THβC derived azomethine ylide and 3-arylidene-chroman-4-ones

inferred← citeshttps://doi.org/10.1016/j.molstruc.2025.144950openalex-snapshot

Solvent-free, mechanochemical synthesis of chromone-based Schiff bases: A green approach to bioactive heterocycles

inferred← citeshttps://doi.org/10.1016/j.neuro.2018.02.017openalex-snapshot

Myxobacterial natural products: An under-valued source of products for drug discovery for neurological disorders

inferred← citeshttps://doi.org/10.1016/j.pestbp.2025.106311openalex-snapshot

Design and synthesis of sulfur-containing pseudilin analogs and their biological activity evaluation

inferred← citeshttps://doi.org/10.1016/j.poly.2017.10.027openalex-snapshot

Novel copper(II), cobalt(II) and nickel(II) complexes with 5-(4-oxo-4H-chromen-3-yl)-4,5-dihydro-1,3,4-thiadiazole-2-carboxamide: Synthesis, structure, spectroscopic studies

inferred← citeshttps://doi.org/10.1016/j.poly.2021.115638openalex-snapshot

Comprehensive biological {DNA/RNA binding profile, cleavage &cytotoxicity activity} of structurally well-characterized chromone-appended Cu(II)(L1-3)(phen) potential anticancer drug candidates

inferred← citeshttps://doi.org/10.1016/j.rechem.2025.102601openalex-snapshot

Natural chromones targeting autophagy signalling pathways as potential anticancer interventions: a systematic review

inferred← citeshttps://doi.org/10.1016/j.saa.2019.117193openalex-snapshot

A novel chromone based colorimetric sensor for highly selective detection of copper ions: Synthesis, optical properties and DFT calculations

inferred← citeshttps://doi.org/10.1016/j.saa.2025.126638openalex-snapshot

Credentials of chromone based probe as colorimetric sensor for the detection of Cu2+ ion: design of test paper kit and potential anticancer activity

inferred← citeshttps://doi.org/10.1016/j.talanta.2018.12.014openalex-snapshot

A highly sensitive and responsive fluorescent probe based on 6-azide-chroman dye for detection and imaging of hydrogen sulfide in cells

inferred← citeshttps://doi.org/10.1016/j.tet.2022.133018openalex-snapshot

Electrooxidative tandem cyclization of enaminones to give 3-arylthiochromone derivatives

inferred← citeshttps://doi.org/10.1016/j.tet.2024.133948openalex-snapshot

HFIP promoted cyclization of o-hydroxyaryl enaminones with chlorohydrocarbon for synthesis of chromone-containing triarylmethanes

inferred← citeshttps://doi.org/10.1016/j.tet.2024.134087openalex-snapshot

Divergent synthesis of chromones and chromanones from diketones using an AgOTf/[Si]H system by switching hydrosilanes

inferred← citeshttps://doi.org/10.1016/j.tetlet.2018.11.055openalex-snapshot

Total synthesis of diaportheone A

inferred← citeshttps://doi.org/10.1016/j.tetlet.2020.152602openalex-snapshot

A new multicomponent approach to the synthesis of substituted furan-2(5H)-ones containing 4H-chromen-4-one fragment

inferred← citeshttps://doi.org/10.1016/j.tifs.2021.02.029openalex-snapshot

Fungal glycosides: Structure and biological function

inferred← citeshttps://doi.org/10.1021/acs.cgd.2c01076openalex-snapshot

First Example of Chromone-Based Nickel(II) Coordination Polymers with Tunable Magnetic Properties

inferred← citeshttps://doi.org/10.1021/acs.chemrev.1c00513openalex-snapshot

Site-Selective Cross-Coupling of Polyhalogenated Arenes and Heteroarenes with Identical Halogen Groups

inferred← citeshttps://doi.org/10.1021/acs.jafc.1c03626openalex-snapshot

Discovery of Novel Chromone Derivatives as Potential Anti-TSWV Agents

inferred← citeshttps://doi.org/10.1021/acs.jafc.3c06367openalex-snapshot

Novel 5-Sulfonyl-1,3,4-thiadiazole-Substituted Flavonoids as Potential Bactericides and Fungicides: Design, Synthesis, Three-Dimensional Quantitative Structure–Activity Relationship Studies

inferred← citeshttps://doi.org/10.1021/acs.jafc.6c01634openalex-snapshot

Design and Synthesis of Novel Chroman-4-one Derivatives Containing a Sulfone Moiety as Potential Antibacterial Agents for Kiwifruit Bacterial Canker

inferred← citeshttps://doi.org/10.1021/acs.jmedchem.3c01087openalex-snapshot

Synthesis of Metallo-Chromone Porphyrin Nano-Starch Sensitizers as Photodynamic Therapeutics for the Eradication of Enterococci Dental Pathogens

inferred← citeshttps://doi.org/10.1021/acs.jmedchem.4c02080openalex-snapshot

Discovery of Potent and Selective CDK4/6 Inhibitors for the Treatment of Chemotherapy-Induced Myelosuppression

inferred← citeshttps://doi.org/10.1021/acs.jmedchem.8b00357openalex-snapshot

Tight-Binding Inhibition of Human Monoamine Oxidase B by Chromone Analogs: A Kinetic, Crystallographic, and Biological Analysis

inferred← citeshttps://doi.org/10.1021/acs.jmedchem.8b00876openalex-snapshot

From Oxiranes to Oligomers: Architectures of U.S. FDA Approved Pharmaceuticals Containing Oxygen Heterocycles

inferred← citeshttps://doi.org/10.1021/acs.jnatprod.1c00385openalex-snapshot

Effect of the Chromone Core Substitution of Dirchromone on the Resultant Biological Activities

inferred← citeshttps://doi.org/10.1021/acs.joc.0c00537openalex-snapshot

Photoredox Functionalization of 3-Halogenchromones, 3-Formylchromones, and Chromone-3-carboxylic Acids: Routes to 3-Acylchromones

inferred← citeshttps://doi.org/10.1021/acs.joc.1c00981openalex-snapshot

Michael-Aldol Double Elimination Cascade to Make Pyridines: Use of Chromone for the Synthesis of Indolizines

inferred← citeshttps://doi.org/10.1021/acs.joc.1c02796openalex-snapshot

Photoredox-Catalyzed Cascade of o-Hydroxyarylenaminones to Access 3-Aminated Chromones

inferred← citeshttps://doi.org/10.1021/acs.joc.1c02997openalex-snapshot

Flexible Approach for the Synthesis of Annulated 4H-Pyrans Based on a Cu(I)-Catalyzed C-Allylation/O-Vinylation Reaction of Cyclic 1-Bromoallyl Tosylates with Cyclic and Acyclic 1,3-Dicarbonyls

inferred← citeshttps://doi.org/10.1021/acs.joc.2c00695openalex-snapshot

An Environmentally Benign Multicomponent Cascade Reaction of 3-Formylchromones, 2-Naphthols, and Heterocyclic Ketal Aminals: Site-Selective Synthesis of Functionalized Morphan Derivatives

inferred← citeshttps://doi.org/10.1021/acs.joc.2c01005openalex-snapshot

Copper-Mediated Cyclization of o -Hydroxyaryl Enaminones with 3-Indoleacetic Acids toward the Synthesis of 3-Indolmethyl-Chromones

inferred← citeshttps://doi.org/10.1021/acs.joc.2c01637openalex-snapshot

Transition-Metal-Free Synthesis of 3-Acyl Chromones by the Tandem Reaction of Ynones and Methyl Salicylates

inferred← citeshttps://doi.org/10.1021/acs.joc.2c01719openalex-snapshot

Multicomponent Cascade Reaction of 3-Cyanochromones: Highly Site-Selective Synthesis of 2-(1H-Imidazol-1-yl)-4H-chromen-4-one Derivatives

inferred← citeshttps://doi.org/10.1021/acs.joc.2c02698openalex-snapshot

The Suzuki–Miyaura Cross-Coupling–Claisen Rearrangement–Cross-Metathesis Approach to Prenylated Isoflavones

inferred← citeshttps://doi.org/10.1021/acs.joc.3c00093openalex-snapshot

A Strategy for Accessing Trifluoromethyl Carbinol-Containing Chromones from o-Hydroxyaryl Enaminones and Trifluoroacetaldehyde/Ketone Derivatives

inferred← citeshttps://doi.org/10.1021/acs.joc.3c00407openalex-snapshot

One-Pot Synthesis of Chromone-2-carboxylate Scaffold: An Important Pharmacophore with Diverse Biological Properties

inferred← citeshttps://doi.org/10.1021/acs.joc.3c01339openalex-snapshot

Visible-Light-Induced Synthesis of 3-Alkyl Chromones under Catalyst- and Additive-Free Conditions

inferred← citeshttps://doi.org/10.1021/acs.joc.3c02337openalex-snapshot

Synthesis of Chroman-2,4-diones via Ring-Opening/Ring-Closing Reaction Involving Palladium-Catalyzed Intramolecular Aryloxycarbonylation

inferred← citeshttps://doi.org/10.1021/acs.joc.3c02399openalex-snapshot

Photoredox-Catalyzed Tandem Cyclization of Enaminones with N-Sulfonylaminopyridinium Salts toward the Synthesis of 3-Sulfonaminated Chromones

inferred← citeshttps://doi.org/10.1021/acs.joc.4c01410openalex-snapshot

Lewis Acid-Driven Multicomponent Reactions Enable 2-Alkyl Chromanones with Anticancer Activities

inferred← citeshttps://doi.org/10.1021/acs.joc.4c01591openalex-snapshot

Base-Dependent Divergent Carbodifluoroalkylation and Halodifluoroalkylation of Alkenes under Visible-Light Irradiation

inferred← citeshttps://doi.org/10.1021/acs.joc.5c00206openalex-snapshot

Defluorinative Approach for the Synthesis of Chromones via [4 + 2] Annulation of Difluoro Quinone Methide

inferred← citeshttps://doi.org/10.1021/acs.joc.5c00424openalex-snapshot

Visible-Light-Driven Tandem Cyclization of o-Hydroxyaryl Enaminones: Access to 3-(α-Arylsulfonamido)trifluoroethyl Chromones

inferred← citeshttps://doi.org/10.1021/acs.joc.6c00346openalex-snapshot

Selective O -Acylation of Ketones with Carboxylic Acids for Enol Esters Synthesis

inferred← citeshttps://doi.org/10.1021/acs.joc.6c01078openalex-snapshot

Organocatalytic Asymmetric Michael Addition/Annulation Cascade toward the β-Nitro Chromones

inferred← citeshttps://doi.org/10.1021/acs.joc.6c01871openalex-snapshot

Visible-Light-Induced Synthesis for Sulfonyl (Thio)chromones and 4-Quinolones from 2-Alknyl Benzaldehydes and Sodium Sulfinates via a Cascade Sulfonylation/Cyclization/Isomerization Processes

inferred← citeshttps://doi.org/10.1021/acs.joc.8b00099openalex-snapshot

Three-Component Site-Selective Synthesis of Highly Substituted 5H-Chromeno-[4,3-b]pyridines

inferred← citeshttps://doi.org/10.1021/acs.joc.8b00177openalex-snapshot

Cu(OAc)2Mediated Synthesis of 3-Sulfonyl Chromen-4-ones

inferred← citeshttps://doi.org/10.1021/acs.joc.8b01043openalex-snapshot

Stereocontrolled Synthesis of 3-Sulfonyl Chroman-4-ols

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