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Enantioselective Synthesis of Fluoro–Dihydroquinazolones and −Benzooxazinones by Fluorination-Initiated Asymmetric Cyclization Reactions
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What this work says
Outgoing claims: the papers this work cites, builds on, or argues with.
inferredcites →https://doi.org/10.1002/1521-3773(20011203)40:23<4461::aid-anie4461>3.0.co;2-eopenalex-snapshot
Synthesis of Fluorogypsetin and Fluorobrevianamide E by a Novel Fluorination–Cyclization of cyclo-L-Trp-L-AAs This work was supported by a Grant-in-Aid for Scientific Research from the Ministry of Education, Science, Sports and Culture, Japan. N.S. wishes to thank the Novartis Foundation (Japan)…
inferredcites →https://doi.org/10.1002/9783906390444openalex-snapshot
Hydrolysis in Drug and Prodrug Metabolism
inferredcites →https://doi.org/10.1002/adsc.201100849openalex-snapshot
Catalytic Asymmetric Synthesis of Dihydroquinazolinones from Imines and 2‐Aminobenzamides
inferredcites →https://doi.org/10.1002/anie.200500395openalex-snapshot
Enantioselective Formation of Stereogenic Carbon–Fluorine Centers by a Simple Catalytic Method
inferredcites →https://doi.org/10.1002/anie.200500571openalex-snapshot
Direct Asymmetric α‐Fluorination of Aldehydes
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The Development of Double Axially Chiral Phosphoric Acids and Their Catalytic Transfer Hydrogenation of Quinolines
inferredcites →https://doi.org/10.1002/anie.200804770openalex-snapshot
Asymmetric Brønsted Acid Catalysis: Catalytic Enantioselective Synthesis of Highly Biologically Active Dihydroquinazolinones
inferredcites →https://doi.org/10.1002/anie.200901795openalex-snapshot
Electrophilic Fluorocyclization of Allyl Silanes
inferredcites →https://doi.org/10.1002/anie.201005347openalex-snapshot
N‐Phosphinyl Phosphoramide—A Chiral Brønsted Acid Motif for the Direct Asymmetric N,O‐Acetalization of Aldehydes
inferredcites →https://doi.org/10.1002/anie.201103151openalex-snapshot
Organocatalyzed Enantioselective Fluorocyclizations
inferredcites →https://doi.org/10.1002/anie.201205343openalex-snapshot
Asymmetric Counteranion‐Directed Catalysis: Concept, Definition, and Applications
inferredcites →https://doi.org/10.1002/anie.201205383openalex-snapshot
A Doubly Axially Chiral Phosphoric Acid Catalyst for the Asymmetric Tandem Oxyfluorination of Enamides
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inferredcites →https://doi.org/10.1002/anie.201302002openalex-snapshot
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inferredcites →https://doi.org/10.1002/anie.201303527openalex-snapshot
Enantioselective Organocatalytic Fluorination‐Induced Wagner–Meerwein Rearrangement
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Highly Enantioselective Bromocyclization of Tryptamines and Its Application in the Synthesis of (−)‐Chimonanthine
inferredcites →https://doi.org/10.1002/cbic.200301023openalex-snapshot
Fluorine in Medicinal Chemistry
inferredcites →https://doi.org/10.1002/chem.200600495openalex-snapshot
Non‐Biaryl Atropisomers in Organocatalysis
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Fluoroartemisinins: Metabolically More Stable Antimalarial Artemisinin Derivatives
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inferredcites →https://doi.org/10.1016/b978-0-12-374194-3.00017-2openalex-snapshot
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inferredcites →https://doi.org/10.1016/b978-0-12-744481-9.x5000-4openalex-snapshot
The Practice of Medicinal Chemistry
inferredcites →https://doi.org/10.1016/b978-012744481-9/50035-0openalex-snapshot
BIOTRANSFORMATION REACTIONS
inferredcites →https://doi.org/10.1016/j.bmcl.2008.12.035openalex-snapshot
(−)-Cercosporamide derivatives as novel antihyperglycemic agents
inferredcites →https://doi.org/10.1016/j.bmcl.2011.07.098openalex-snapshot
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inferredcites →https://doi.org/10.1021/cs400591uopenalex-snapshot
Highly Enantioselective Synthesis of Dihydroquinazolinones Catalyzed by SPINOL-Phosphoric Acids
inferredcites →https://doi.org/10.1021/ja01496a020openalex-snapshot
Quinazolinone Sulfonamides. A New Class of Diuretic Agents1
inferredcites →https://doi.org/10.1021/ja051805fopenalex-snapshot
Enantioselective Organocatalytic α-Fluorination of Aldehydes
inferredcites →https://doi.org/10.1021/ja0533085openalex-snapshot
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inferredcites →https://doi.org/10.1021/ja311798qopenalex-snapshot
Chiral Anion Phase-Transfer Catalysis Applied to the Direct Enantioselective Fluorinative Dearomatization of Phenols
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Silver-Catalyzed Radical Aminofluorination of Unactivated Alkenes in Aqueous Media
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Palladium-Catalyzed Intramolecular Aminofluorination of Unactivated Alkenes
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A Novel Synthesis of Fluorinated Pyrazoles via Gold(I)-Catalyzed Tandem Aminofluorination of Alkynes in the Presence of Selectfluor
inferredcites →https://doi.org/10.1038/nchem.1405openalex-snapshot
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inferredcites →https://doi.org/10.1039/b711844aopenalex-snapshot
Understanding organofluorine chemistry. An introduction to the C–F bond
inferredcites →https://doi.org/10.1039/c1md00145kopenalex-snapshot
The synthesis and evaluation of dihydroquinazolin-4-ones and quinazolin-4-ones as thyroid stimulating hormone receptor agonists
inferredcites →https://doi.org/10.1070/mc2002v012n03abeh001564openalex-snapshot
Fluorocyclization of norbornenecarboxylic acids with F-TEDA-BF4
inferredcites →https://doi.org/10.1073/pnas.1304346110openalex-snapshot
A combination of directing groups and chiral anion phase-transfer catalysis for enantioselective fluorination of alkenes
inferredcites →https://doi.org/10.1080/14756360701425014openalex-snapshot
The role of fluorine in medicinal chemistry
inferredcites →https://doi.org/10.1126/science.1213918openalex-snapshot
Asymmetric Electrophilic Fluorination Using an Anionic Chiral Phase-Transfer Catalyst
inferredcites →https://doi.org/10.1146/annurev.pharmtox.41.1.443openalex-snapshot
Metabolism of Fluorine-Containing Drugs
inferredcites →https://doi.org/10.3762/bjoc.6.38openalex-snapshot
The C–F bond as a conformational tool in organic and biological chemistry
What points at this work
Incoming claims: where this work appears in other papers’ reference lists and arguments.
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Homoleptic Pyrazinoic Acid Transition Metal Complex as an Efficient Catalyst Toward Elegant Three-Component Synthesis of 3,4-Dihydro-2h-1,3-Benzoxazines
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phosphate/phosphorus (P) catalysts/phosphoric acid
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Asymmetric Fluorination Reactions
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Recent Developments in Enantioselective Organocatalytic Cascade Reactions for the Construction of Halogenated Ring Systems
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