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PROTAC Degrader of Estrogen Receptor α Targeting DNA-Binding Domain in Breast Cancer
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What this work says
Outgoing claims: the papers this work cites, builds on, or argues with.
inferredcites →https://doi.org/10.1002/0471143030.cb0602s00openalex-snapshot
Immunoblotting and Immunodetection
inferredcites →https://doi.org/10.1002/0471143030.cb0602s52openalex-snapshot
Immunoblotting and Immunodetection
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A Stepwise Huisgen Cycloaddition Process: Copper(I)-Catalyzed Regioselective “Ligation” of Azides and Terminal Alkynes
inferredcites →https://doi.org/10.1002/advs.202102555openalex-snapshot
Destruction of DNA‐Binding Proteins by Programmable Oligonucleotide PROTAC (O'PROTAC): Effective Targeting of LEF1 and ERG
inferredcites →https://doi.org/10.1002/advs.202170136openalex-snapshot
Destruction of DNA‐Binding Proteins by Programmable Oligonucleotide PROTAC (O'PROTAC): Effective Targeting of LEF1 and ERG (Adv. Sci. 20/2021)
inferredcites →https://doi.org/10.1002/ange.202012330openalex-snapshot
RNA‐PROTACs: Degraders of RNA‐Binding Proteins
inferredcites →https://doi.org/10.1002/anie.201101817openalex-snapshot
Increasing the Efficacy of Bioorthogonal Click Reactions for Bioconjugation: A Comparative Study
inferredcites →https://doi.org/10.1002/anie.201206231openalex-snapshot
Small‐Molecule Inhibitors of the Interaction between the E3 Ligase VHL and HIF1α
inferredcites →https://doi.org/10.1002/anie.202012330openalex-snapshot
RNA‐PROTACs: Degraders of RNA‐Binding Proteins
inferredcites →https://doi.org/10.1002/anie.202107347openalex-snapshot
Aptamer‐PROTAC Conjugates (APCs) for Tumor‐Specific Targeting in Breast Cancer
inferredcites →https://doi.org/10.1002/j.1460-2075.1987.tb02706.xopenalex-snapshot
The estrogen‐responsive element as an inducible enhancer: DNA sequence requirements and conversion to a glucocorticoid‐responsive element.
inferredcites →https://doi.org/10.1007/978-1-60327-575-0_1openalex-snapshot
Nuclear Receptors: One Big Family
inferredcites →https://doi.org/10.1007/s12032-009-9397-3openalex-snapshot
Inhibition of autophagy by 3-MA potentiates cisplatin-induced apoptosis in esophageal squamous cell carcinoma cells
inferredcites →https://doi.org/10.1016/0022-1759(83)90303-4openalex-snapshot
Rapid colorimetric assay for cellular growth and survival: Application to proliferation and cytotoxicity assays
inferredcites →https://doi.org/10.1016/0022-1759(91)90198-oopenalex-snapshot
A rapid and simple method for measuring thymocyte apoptosis by propidium iodide staining and flow cytometry
inferredcites →https://doi.org/10.1016/0092-8674(87)90581-2openalex-snapshot
Functional domains of the human estrogen receptor
inferredcites →https://doi.org/10.1016/0092-8674(88)90017-7openalex-snapshot
The estrogen receptor binds tightly to its responsive element as a ligand-induced homodimer
inferredcites →https://doi.org/10.1016/0092-8674(93)90485-9openalex-snapshot
The C. elegans cell death gene ced-3 encodes a protein similar to mammalian interleukin-1β-converting enzyme
inferredcites →https://doi.org/10.1016/0092-8674(95)90199-xopenalex-snapshot
The nuclear receptor superfamily: The second decade
inferredcites →https://doi.org/10.1016/b978-0-12-418687-3.00006-9openalex-snapshot
Purification of DNA Oligos by Denaturing Polyacrylamide Gel Electrophoresis (PAGE)
inferredcites →https://doi.org/10.1016/j.bios.2017.07.043openalex-snapshot
Fully disposable microfluidic electrochemical device for detection of estrogen receptor alpha breast cancer biomarker
inferredcites →https://doi.org/10.1016/j.bmcl.2019.03.035openalex-snapshot
Selective degradation of CDK6 by a palbociclib based PROTAC
inferredcites →https://doi.org/10.1016/j.ccell.2020.03.009openalex-snapshot
Overcoming Endocrine Resistance in Breast Cancer
inferredcites →https://doi.org/10.1016/j.cell.2008.08.037openalex-snapshot
Sgs1 Helicase and Two Nucleases Dna2 and Exo1 Resect DNA Double-Strand Break Ends
inferredcites →https://doi.org/10.1016/j.cell.2019.11.031openalex-snapshot
Proteolysis-Targeting Chimeras as Therapeutics and Tools for Biological Discovery
inferredcites →https://doi.org/10.1016/j.chembiol.2017.09.009openalex-snapshot
The Advantages of Targeted Protein Degradation Over Inhibition: An RTK Case Study
inferredcites →https://doi.org/10.1016/j.chembiol.2021.03.011openalex-snapshot
Targeted degradation of transcription factors by TRAFTACs: TRAnscription Factor TArgeting Chimeras
inferredcites →https://doi.org/10.1016/j.chembiol.2021.04.011openalex-snapshot
Targeted protein degradation: A promise for undruggable proteins
inferredcites →https://doi.org/10.1016/j.ejmech.2020.112689openalex-snapshot
Targeting estrogen receptor α for degradation with PROTACs: A promising approach to overcome endocrine resistance
inferredcites →https://doi.org/10.1016/j.ymthe.2005.03.038openalex-snapshot
Role of clathrin- and caveolae-mediated endocytosis in gene transfer mediated by lipo- and polyplexes
inferredcites →https://doi.org/10.1016/s0039-128x(99)00014-8openalex-snapshot
The structure of the nuclear hormone receptors
inferredcites →https://doi.org/10.1016/s0140-6736(13)62422-8openalex-snapshot
Pathological complete response and long-term clinical benefit in breast cancer: the CTNeoBC pooled analysis
inferredcites →https://doi.org/10.1021/ac9026498openalex-snapshot
Gold-Nanoparticle-Based Assay for Instantaneous Detection of Nuclear Hormone Receptor−Response Elements Interactions
inferredcites →https://doi.org/10.1021/acs.biochem.8b00391openalex-snapshot
Targeting the C481S Ibrutinib-Resistance Mutation in Bruton’s Tyrosine Kinase Using PROTAC-Mediated Degradation
inferredcites →https://doi.org/10.1021/acs.jmedchem.6b01781openalex-snapshot
A “Click Chemistry Platform” for the Rapid Synthesis of Bispecific Molecules for Inducing Protein Degradation
inferredcites →https://doi.org/10.1021/acs.jmedchem.7b00635openalex-snapshot
Identification and Characterization of Von Hippel-Lindau-Recruiting Proteolysis Targeting Chimeras (PROTACs) of TANK-Binding Kinase 1
inferredcites →https://doi.org/10.1021/acschembio.7b00985openalex-snapshot
Development of Stabilized Peptide-Based PROTACs against Estrogen Receptor α
inferredcites →https://doi.org/10.1021/acsmedchemlett.1c00629openalex-snapshot
Development of Chimeric Molecules That Degrade the Estrogen Receptor Using Decoy Oligonucleotide Ligands
inferredcites →https://doi.org/10.1021/ja202946kopenalex-snapshot
Design and Structure of Stapled Peptides Binding to Estrogen Receptors
inferredcites →https://doi.org/10.1021/ja209924vopenalex-snapshot
Targeting the von Hippel–Lindau E3 Ubiquitin Ligase Using Small Molecules To Disrupt the VHL/HIF-1α Interaction
inferredcites →https://doi.org/10.1021/jacs.1c03852openalex-snapshot
TF-PROTACs Enable Targeted Degradation of Transcription Factors
inferredcites →https://doi.org/10.1021/jo011148jopenalex-snapshot
Peptidotriazoles on Solid Phase: [1,2,3]-Triazoles by Regiospecific Copper(I)-Catalyzed 1,3-Dipolar Cycloadditions of Terminal Alkynes to Azides
inferredcites →https://doi.org/10.1038/bjc.1972.33openalex-snapshot
Apoptosis: A Basic Biological Phenomenon with Wideranging Implications in Tissue Kinetics
inferredcites →https://doi.org/10.1038/d41573-021-00052-4openalex-snapshot
Targeted protein degraders crowd into the clinic
inferredcites →https://doi.org/10.1038/s41392-019-0101-6openalex-snapshot
PROTACs: great opportunities for academia and industry
inferredcites →https://doi.org/10.1038/s41467-018-08027-7openalex-snapshot
Differential PROTAC substrate specificity dictated by orientation of recruited E3 ligase
inferredcites →https://doi.org/10.1038/s41591-019-0668-zopenalex-snapshot
A selective BCL-XL PROTAC degrader achieves safe and potent antitumor activity
inferredcites →https://doi.org/10.1039/d1cc05025gopenalex-snapshot
G4-PROTAC: targeted degradation of a G-quadruplex binding protein
inferredcites →https://doi.org/10.1073/pnas.141230798openalex-snapshot
Protacs: Chimeric molecules that target proteins to the Skp1–Cullin–F box complex for ubiquitination and degradation
inferredcites →https://doi.org/10.1073/pnas.96.15.8461openalex-snapshot
Characterization of lipid bilayer phases by confocal microscopy and fluorescence correlation spectroscopy
inferredcites →https://doi.org/10.1093/jnci/88.19.1361openalex-snapshot
Human Papillomavirus Type 18: Association With Poor Prognosis in Early Stage Cervical Cancer
inferredcites →https://doi.org/10.1093/jnci/djh166openalex-snapshot
Mechanisms of Tamoxifen Resistance: Increased Estrogen Receptor-HER2/neu Cross-Talk in ER/HER2-Positive Breast Cancer
inferredcites →https://doi.org/10.1093/nar/29.14.2905openalex-snapshot
Estrogen receptor interaction with estrogen response elements
inferredcites →https://doi.org/10.1093/nar/9.23.6505openalex-snapshot
Equilibria and kinetics of lac repressor-operator interactions by polyacrylamide gel electrophoresis
inferredcites →https://doi.org/10.1093/nar/gkm935openalex-snapshot
A versatile method for the preparation of conjugates of peptides with DNA/PNA/analog by employing chemo-selective click reaction in water
inferredcites →https://doi.org/10.1097/00008390-200112000-00011openalex-snapshot
Angiopoietin-1, angiopoietin-2 and Tie-2 in tumour and non-tumour tissues during growth of experimental melanoma
inferredcites →https://doi.org/10.1097/mjt.0b013e31817c941fopenalex-snapshot
Methods in Molecular Biology
inferredcites →https://doi.org/10.1101/gad.316646.118openalex-snapshot
Signaling pathways and steroid receptors modulating estrogen receptor α function in breast cancer
inferredcites →https://doi.org/10.1111/j.1365-2818.1993.tb03315.xopenalex-snapshot
Aberrations in confocal fluorescence microscopy induced by mismatches in refractive index
inferredcites →https://doi.org/10.1126/science.2667136openalex-snapshot
Transcriptional Regulation in Mammalian Cells by Sequence-Specific DNA Binding Proteins
inferredcites →https://doi.org/10.1126/science.274.5285.246openalex-snapshot
Identification of a Human Mitotic Checkpoint Gene: hsMAD2
inferredcites →https://doi.org/10.1126/science.aar6245openalex-snapshot
CRISPR-Cas12a target binding unleashes indiscriminate single-stranded DNase activity
inferredcites →https://doi.org/10.1186/s12943-016-0575-6openalex-snapshot
Long non-coding RNA TUG1 is involved in cell growth and chemoresistance of small cell lung cancer by regulating LIMK2b via EZH2
inferredcites →https://doi.org/10.1186/s13045-020-00885-3openalex-snapshot
Proteolysis-targeting chimera (PROTAC) for targeted protein degradation and cancer therapy
inferredcites →https://doi.org/10.2174/156802612799436641openalex-snapshot
General Molecular Biology and Architecture of Nuclear Receptors
inferredcites →https://doi.org/10.2217/fon.13.82openalex-snapshot
Preparation and Characterization of Gelatin Nanoparticles Containing pDNA Encoding IL-12 anD Their Expression in CT-26 Carcinoma Cells
inferredcites →https://doi.org/10.3322/caac.21492openalex-snapshot
Global cancer statistics 2018: GLOBOCAN estimates of incidence and mortality worldwide for 36 cancers in 185 countries
inferredcites →https://doi.org/10.3322/caac.21660openalex-snapshot
Global Cancer Statistics 2020: GLOBOCAN Estimates of Incidence and Mortality Worldwide for 36 Cancers in 185 Countries
What points at this work
Incoming claims: where this work appears in other papers’ reference lists and arguments.
inferred← citeshttps://doi.org/10.1002/chem.202503641openalex-snapshot
Accelerating the Discovery of Targeted Protein Degraders: Advances in Synthetic Methodologies and Screening Tactics
inferred← citeshttps://doi.org/10.1002/cmdc.202300422openalex-snapshot
Click Chemistry and Targeted Degradation: A Winning Combination for Medicinal Chemists?
inferred← citeshttps://doi.org/10.1002/cmdc.202400267openalex-snapshot
Proteolysis Targeting Chimeras (PROTACs) in Breast Cancer Therapy
inferred← citeshttps://doi.org/10.1002/mco2.290openalex-snapshot
PROTACs: A novel strategy for cancer drug discovery and development
inferred← citeshttps://doi.org/10.1002/mco2.478openalex-snapshot
mRNA PROTACs: engineering PROTACs for high‐efficiency targeted protein degradation
inferred← citeshttps://doi.org/10.1002/mco2.694openalex-snapshot
Mechanisms of resistance to tyrosine kinase inhibitor‐targeted therapy and overcoming strategies
inferred← citeshttps://doi.org/10.1002/smll.202302525openalex-snapshot
Selective Proteolysis of Activated Transcriptional Factor by NIR‐Responsive Palindromic DNA Thalidomide Conjugate Inhibits the Canonical Smad Pathway
inferred← citeshttps://doi.org/10.1007/s10549-023-07136-2openalex-snapshot
Complete elimination of estrogen receptor α by PROTAC estrogen receptor α degrader ERD-148 in breast cancer cells
inferred← citeshttps://doi.org/10.1007/s11426-024-2246-0openalex-snapshot
ZIF-90-loaded DNAzyme-responsive PROTAC for the self-powered degradation of NF-κB
inferred← citeshttps://doi.org/10.1007/s12272-025-01583-9openalex-snapshot
Advances and challenges of estrogen receptor-targeted agents in breast cancer
inferred← citeshttps://doi.org/10.1016/b978-0-443-21816-3.00005-1openalex-snapshot
Degraders of proteins involved in transcription nuclear hormone receptors
inferred← citeshttps://doi.org/10.1016/j.addr.2026.115819openalex-snapshot
Bridged PROTAC, DNA-based PROTAC and hydrophobic tag technologies for targeted protein degradation
inferred← citeshttps://doi.org/10.1016/j.bej.2023.109063openalex-snapshot
Incorporating a β-hairpin sequence motif to increase intracellular stability of a peptide-based PROTAC
inferred← citeshttps://doi.org/10.1016/j.bmc.2025.118297openalex-snapshot
Advances in DNA-based proteolysis-targeting chimeras technology: Novel strategies for targeting previously undruggable proteins in cancer therapy
inferred← citeshttps://doi.org/10.1016/j.ejmech.2023.115384openalex-snapshot
Bifunctional robots inducing targeted protein degradation
inferred← citeshttps://doi.org/10.1016/j.ejmech.2023.116041openalex-snapshot
Journey of Von Hippel-Lindau (VHL) E3 ligase in PROTACs design: From VHL ligands to VHL-based degraders
inferred← citeshttps://doi.org/10.1016/j.ejmech.2024.116184openalex-snapshot
Fluorescence theranostic PROTACs for real-time visualization of ERα degradation
inferred← citeshttps://doi.org/10.1016/j.ejmech.2024.116978openalex-snapshot
Targeting oncogenic transcriptional factor c-myc by oligonucleotide PROTAC for the treatment of hepatocellular carcinoma
inferred← citeshttps://doi.org/10.1016/j.ejps.2024.106793openalex-snapshot
PROTAC: Novel degradable approach for different targets to treat breast cancer
inferred← citeshttps://doi.org/10.1016/j.pharmthera.2024.108725openalex-snapshot
Powering up targeted protein degradation through active and passive tumour-targeting strategies: Current and future scopes
inferred← citeshttps://doi.org/10.1016/j.tips.2025.05.003openalex-snapshot
Emerging approaches for antagonizing the aryl hydrocarbon receptor
inferred← citeshttps://doi.org/10.1021/acs.jmedchem.5c00490openalex-snapshot
Rational Design of Methylene Blue–Raloxifene Conjugates for Efficient Breast Tumor Elimination Triggered by ERα Degradation
inferred← citeshttps://doi.org/10.1021/acsami.3c14640openalex-snapshot
Conjugated Polyelectrolyte/Single Strand DNA Hybrid Polyplexes for Efficient Nucleic Acid Delivery and Targeted Protein Degradation
inferred← citeshttps://doi.org/10.1021/acsnano.2c10379openalex-snapshot
Aptamer-Based Targeted Protein Degradation
inferred← citeshttps://doi.org/10.1021/acsptsci.4c00469openalex-snapshot
Aptamer Proteolysis-Targeting Chimeras (PROTACs): A Novel Strategy to Combat Drug Resistance in Estrogen Receptor α-Positive Breast Cancer
inferred← citeshttps://doi.org/10.1038/s41392-023-01651-wopenalex-snapshot
Transcriptional co-activators: emerging roles in signaling pathways and potential therapeutic targets for diseases
inferred← citeshttps://doi.org/10.1038/s41434-026-00622-4openalex-snapshot
DOCTER: a genetically encoded switchable protein module for ERα-mediated transcriptional regulation
inferred← citeshttps://doi.org/10.1039/d4md00961dopenalex-snapshot
Development of PROTACs targeting estrogen receptor: an emerging technique for combating endocrine resistance
inferred← citeshttps://doi.org/10.1042/bst20220338openalex-snapshot
Interactions governing transcriptional activity of nuclear receptors
inferred← citeshttps://doi.org/10.1097/cm9.0000000000004327openalex-snapshot
ESR1 alterations in breast cancer: Mechanisms, detection, and therapeutic implications
inferred← citeshttps://doi.org/10.1101/2024.04.25.591105openalex-snapshot
Estrogen Receptor α/14-3-3 molecular glues as alternative treatment strategy for endocrine resistant breast cancer
inferred← citeshttps://doi.org/10.21203/rs.3.rs-4283954/v1openalex-snapshot
Evaluation of cereblon expression in gastrointestinal tract tumors
inferred← citeshttps://doi.org/10.3389/fonc.2025.1513225openalex-snapshot
Decoding estrogen receptor and GPER biology: structural insights and therapeutic advances in ERα−positive breast cancer
inferred← citeshttps://doi.org/10.3390/biomedicines14040835openalex-snapshot
Research Progress of PROTACs in Breast Cancer: Subtype-Oriented Target Landscape, Clinical Stratification Evidence, and Engineering Strategies for Translation
inferred← citeshttps://doi.org/10.3390/cancers17111871openalex-snapshot
Targeting the Undruggable: Recent Progress in PROTAC-Induced Transcription Factor Degradation
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