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Diversification of the Three-Component Coupling of 2-Aminoheterocycles, Aldehydes, and Isonitriles: Efficient Parallel Synthesis of a Diverse and Druglike Library of Imidazo- and Tetrahydroimidazo[1,2-a] Heterocycles

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What this work says

Outgoing claims: the papers this work cites, builds on, or argues with.

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Multicomponent Reactions with Isocyanides

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An Easy and Fast Conversion of N2‐[(tert‐Butoxy)carbonyl]‐ L ‐amino Acids to Corresponding Amino‐aldehydes

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Mannich reactions of heterocycles with dimethyl(methylene) ammonium chloride: A high yield, one‐step conversion of estazolam to adinazolam

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Pyrrolization processes of vinyl substituted imidazo[1,2‐a]pyridine, pyrimidine and 1,8‐naphthyridine

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N-methoxy-N-methylamides (Weinreb amides) in modern organic synthesis

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Use of a convertible isocyanide for generation of Ugi reaction derivatives on solid support: Synthesis of α-acylaminoesters and pyrroles

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Characterization of the physico-chemical properties of the imidazopyridine derivative Alpidem. Comparison with Zolpidem

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Integrating cheminformatic analysis in combinatorial chemistry

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A novel dealkylation affording 3-aminoimidazo[1,2-a]pyridines: access to new substitution patterns by solid-phase synthesis

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Y(OTf)3-catalyzed novel Mannich reaction of N-alkoxycarbonylpyrroles, formaldehyde and primary amine hydrochlorides

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N-methoxy-n-methylamides as effective acylating agents

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Parallel synthesis of 3-aminoimidazo[1,2-a]pyridines and pyrazines by a new three-component condensation

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Remarkable three-step-one-pot solution phase preparation of novel imidazolines utilizing a UDC (Ugi/de-Boc/cyclize) strategy

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Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings

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Synthesis and antiviral activity of imidazo[1,2-a]pyridines

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Multiple-Component Condensation Strategies for Combinatorial Library Synthesis

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Polymer-Supported Tetrafluorophenol: A New Activated Resin for Chemical Library Synthesis

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UPS on Weinreb Resin: A Facile Solid-Phase Route to Aldehyde and Ketone Derivatives of “Unnatural” Amino Acids and Peptides

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Domino Reactions in Organic Synthesis

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Synthesis and hypoglycemic activity of substituted 8-(1-piperazinyl)imidazo[1,2-a]pyrazines

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Antiulcer agents. 5. Inhibition of gastric H+/K+-ATPase by substituted imidazo[1,2-a]pyridines and related analogs and its implication in modeling the high affinity potassium ion binding site of the gastric proton pump enzyme

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Angiotensin-converting enzyme inhibitors: synthesis and biological activity of acyltripeptide analogs of enalapril

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2-Amino-3-substituted-6-[(E)-1-phenyl-2-(N-methylcarbamoyl)vinyl]imidazo[1,2-a]pyridines as a Novel Class of Inhibitors of Human Rhinovirus: Stereospecific Synthesis and Antiviral Activity

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2-Amino-4-benzyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridines: Novel Selective β3-Adrenoceptor Agonists

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Novel 2-Phenylimidazo[1,2-a]pyridine Derivatives as Potent and Selective Ligands for Peripheral Benzodiazepine Receptors: Synthesis, Binding Affinity, and in Vivo Studies

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Redox-photosensitized reactions. 10. Formation of a novel type of adduct between an NADH model and carbonyl compounds by photosensitization using Ru(bpy)32+

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Selective reductions. XVIII. Fast reaction of primary, secondary, and tertiary amides with diborane. Simple, convenient procedure for the conversion of amides to the corresponding amines

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Preparation and New Reactions of Imidazo[1,2-a]pyridines

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A Mild and Efficient Alternative to the Classical Swern Oxidation

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Stereocontrolled Synthesis of 5-Acyl-3,4-dihydro-2H-pyrroles and Related Heterocycles via Intramolecular 2-Propylidene-1,3-bis(silane)−Acylnitrilium Ion Cyclizations

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Reduction of Ethanethiol Esters to Aldehydes

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Substituent Effects on Fluorescent Properties of Imidazo[1,2- a ]pyridine-Based Compounds

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Examination of the Computed Molecular Properties of Compounds Selected for Clinical Development

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Incoming claims: where this work appears in other papers’ reference lists and arguments.

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