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Application of Quantitative Structure–Activity Relationship Models of 5-HT1A Receptor Binding to Virtual Screening Identifies Novel and Potent 5-HT1A Ligands

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Outgoing claims: the papers this work cites, builds on, or argues with.

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Aripiprazole, a novel antipsychotic drug, preferentially increases dopamine release in the prefrontal cortex and hippocampus in rat brain
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Beware of q2!
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Novel Variable Selection Quantitative Structure−Property Relationship Approach Based on the k -Nearest-Neighbor Principle
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Quantitative Structure−Activity Relationship Modeling of Dopamine D1Antagonists Using Comparative Molecular Field Analysis, Genetic Algorithms−Partial Least-Squares, and K Nearest Neighbor Methods
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Random Forests
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Predictive QSAR modeling based on diversity sampling of experimental datasets for the training and test set selection
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Predictive QSAR modeling based on diversity sampling of experimental datasets for the training and test set selection
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Rational selection of training and test sets for the development of validated QSAR models
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Predicting new molecular targets for known drugs
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H1-Histamine Receptor Affinity Predicts Short-Term Weight Gain for Typical and Atypical Antipsychotic Drugs
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Aripiprazole, A Novel Atypical Antipsychotic Drug with a Unique and Robust Pharmacology
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Chemoinformatics Approaches to Virtual Screening
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Salvinorin A: A potent naturally occurring nonnitrogenous κ opioid selective agonist
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Human serotonin 1D receptor is encoded by a subfamily of two distinct genes: 5-HT1D alpha and 5-HT1D beta.
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Systematic study of substance P analogs
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An immunohistochemical study of the serotonin 1A receptor in the hippocampus of subjects with Alzheimer's disease
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LIBSVM
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The 5-HT1A receptor in schizophrenia: a promising target for novel atypical neuroleptics?
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A case study evaluating the use of clozapine in depression with psychotic features
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Identification of the Descriptor Pharmacophores Using Variable Selection QSAR Applications to Database Mining
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The Potential Utility of 5-HT1A Receptor Antagonists in the Treatment of Cognitive Dysfunction Associated with Alzheimers Disease
inferredcites →https://doi.org/10.2174/138161207782794257openalex-snapshot
Predictive QSAR Modeling Workflow, Model Applicability Domains, and Virtual Screening
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Long-Term Antidepressant Efficacy and Safety of Olanzapine/Fluoxetine Combination
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Aripiprazole Augmentation of Antidepressants for the Treatment of Partially Responding and Nonresponding Patients With Major Depressive Disorder

What points at this work

Incoming claims: where this work appears in other papers’ reference lists and arguments.

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Additional file 1 of Quantitative prediction model for affinity of drug–target interactions based on molecular vibrations and overall system of ligand-receptor
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Additional file 2 of Quantitative prediction model for affinity of drug–target interactions based on molecular vibrations and overall system of ligand-receptor
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Additional file 3 of Quantitative prediction model for affinity of drug–target interactions based on molecular vibrations and overall system of ligand-receptor
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