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Nanomolar E-Selectin Antagonists with Prolonged Half-Lives by a Fragment-Based Approach

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Outgoing claims: the papers this work cites, builds on, or argues with.

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The Conformation of the Sialyl Lewis X Ligand Changes upon Binding to E-Selectin
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Glycomimetic Ligands for the Human Asialoglycoprotein Receptor
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Conformation of sLex Tetrasaccharide, Free in Solution and Bound to E-, P-, and L-Selectin,
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One-Dimensional Relaxation- and Diffusion-Edited NMR Methods for Screening Compounds That Bind to Macromolecules
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Fragment-Based Lead Discovery Using X-ray Crystallography
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Affinity, Kinetics, and Thermodynamics of E-selectin Binding to E-selectin Ligand-1
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ELAM-1 Mediates Cell Adhesion by Recognition of a Carbohydrate Ligand, Sialyl-Le x
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Recognition by Elam-1 of the Sialyl-Le x Determinant on Myeloid and Tumor Cells
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Discovering High-Affinity Ligands for Proteins: SAR by NMR
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GMI-1070, a novel pan-selectin antagonist, reverses acute vascular occlusions in sickle cell mice
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SPR-based Fragment Screening: Advantages and Applications

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Incoming claims: where this work appears in other papers’ reference lists and arguments.

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