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In Vitro Antimalarial Activity of Chalcones and Their Derivatives
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Outgoing claims: the papers this work cites, builds on, or argues with.
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Characterization of a hemoglobin-degrading, low molecular weight protease from Plasmodium falciparum
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Anti-malarial drug development using models of enzyme structure
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Synthesis and Activity of Some Antimalarial Bisquinolines
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Antimalarial Activity of New Dihydroartemisinin Derivatives. 6. .alpha.-Alkylbenzylic Ethers
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Synthesis and antimalarial activity of some 9-substituted artemisinin derivatives
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Bisquinolines. 1. N,N-bis(7-chloroquinolin-4-yl)alkanediamines with potential against chloroquine-resistant malaria
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Antimalarial drugs. 64. Synthesis and antimalarial properties of 1-imino derivatives of 7-chloro-3-substituted-3,4-dihydro-1,9(2H,10H)-acridinediones and related structures
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Malarial haemozoin/β-haematin supports haem polymerization in the absence of protein
inferredcites →https://doi.org/10.1073/pnas.90.8.3583openalex-snapshot
Structure-based inhibitor design by using protein models for the development of antiparasitic agents.
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Plasmodium falciparum: Differential Sensitivity In Vitro to E‐64 (Cysteine Protease Inhibitor) and Pepstatin A (Aspartyl Protease Inhibitor)
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Disease Problems in the Third World
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Researchers Fret Over Neglect Of 600 Million Patients
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Structure-Based Strategies for Drug Design and Discovery
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Quantitative assessment of antimalarial activity in vitro by a semiautomated microdilution technique
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In vitro activities of and mechanisms of resistance to antifol antimalarial drugs
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Licochalcone A, a new antimalarial agent, inhibits in vitro growth of the human malaria parasite Plasmodium falciparum and protects mice from P. yoelii infection
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THE PROTEASES AND PATHOGENICITY OF PARASITIC PROTOZOA
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A malarial cysteine proteinase is necessary for hemoglobin degradation by Plasmodium falciparum.
What points at this work
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inferred← citeshttps://doi.org/10.1002/ptr.701openalex-snapshot
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Structural assignment of chalcones and differentiation of their isomeric derivatives by electron ionization induced fragmentation
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Claisen‐Schmidt Condensation using Green Catalytic Processes: A Critical Review
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Leishmania major:Molecular Modeling of Cysteine Proteases and Prediction of New Nonpeptide Inhibitors
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Trypanosoma brucei: Killing of Bloodstream Formsin Vitroandin Vivoby the Cysteine Proteinase Inhibitor Z-Phe-Ala-CHN2
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Parasite Proteases as Targets for Therapy
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1-(2,3,4-trimethoxyphenyl)-3-(3-(2-chloroquinolinyl))-2-propen-1-one, a chalcone derivative with analgesic, anti-inflammatory and immunomodulatory properties
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inferred← citeshttps://doi.org/10.1016/b978-0-12-373891-2.00075-4openalex-snapshot
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inferred← citeshttps://doi.org/10.1016/b978-0-12-409547-2.14640-2openalex-snapshot
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inferred← citeshttps://doi.org/10.1016/j.bmc.2013.01.026openalex-snapshot
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Prenylated chalcones isolated from Crotalaria genus inhibits in vitro growth of the human malaria parasite Plasmodium falciparum
inferred← citeshttps://doi.org/10.1016/j.bmcl.2005.03.121openalex-snapshot
Synthesis and biological evaluation of chalcones and their derived pyrazoles as potential cytotoxic agents
inferred← citeshttps://doi.org/10.1016/j.bmcl.2005.07.012openalex-snapshot
Conformationally restricted anti-plasmodial chalcones
inferred← citeshttps://doi.org/10.1016/j.bmcl.2005.08.087openalex-snapshot
Sulfonamide chalcone as a new class of α-glucosidase inhibitors
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In vitro and in vivo efficacy and in vitro metabolism of 1-phenyl-3-aryl-2-propen-1-ones against Plasmodium falciparum
inferred← citeshttps://doi.org/10.1016/j.bmcl.2006.08.065openalex-snapshot
Effects of α-substitutions on structure and biological activity of anticancer chalcones
inferred← citeshttps://doi.org/10.1016/j.bmcl.2007.08.021openalex-snapshot
Synthesis and antimicrobial evaluation of new chalcones containing piperazine or 2,5-dichlorothiophene moiety
inferred← citeshttps://doi.org/10.1016/j.bmcl.2008.01.099openalex-snapshot
Synthesis and biological evaluation of chalcones as inhibitors of the voltage-gated potassium channel Kv1.3
inferred← citeshttps://doi.org/10.1016/j.bmcl.2009.12.062openalex-snapshot
Synthesis, antimalarial and antitubercular activity of acetylenic chalcones
inferred← citeshttps://doi.org/10.1016/j.bmcl.2010.01.113openalex-snapshot
The synthesis and Angiotensin Converting Enzyme (ACE) inhibitory activity of chalcones and their pyrazole derivatives
inferred← citeshttps://doi.org/10.1016/j.bmcl.2010.05.069openalex-snapshot
Synthesis of novel α-pyranochalcones and pyrazoline derivatives as Plasmodium falciparum growth inhibitors
inferred← citeshttps://doi.org/10.1016/j.bmcl.2010.07.128openalex-snapshot
Fluorinated 2′-hydroxychalcones as garcinol analogs with enhanced antioxidant and anticancer activities
inferred← citeshttps://doi.org/10.1016/j.bmcl.2010.10.038openalex-snapshot
Synthesis and biological evaluation of retinoid-chalcones as inhibitors of colon cancer cell growth
inferred← citeshttps://doi.org/10.1016/j.bmcl.2010.11.099openalex-snapshot
In vitro efficacy of 7-benzylamino-1-isoquinolinamines against Plasmodium falciparum related to the efficacy of chalcones
inferred← citeshttps://doi.org/10.1016/j.bmcl.2012.07.028openalex-snapshot
Synthesis and in vitro evaluation of new chloroquine-chalcone hybrids against chloroquine-resistant strain of Plasmodium falciparum
inferred← citeshttps://doi.org/10.1016/j.catcom.2006.02.021openalex-snapshot
Solvent-free synthesis of flavanones over aminopropyl-functionalized SBA-15
inferred← citeshttps://doi.org/10.1016/j.cdc.2021.100664openalex-snapshot
Preparation, spectral characterization and single crystal analysis of bromo derivative of 2-acetyl-1-naphthol
inferred← citeshttps://doi.org/10.1016/j.crci.2015.10.014openalex-snapshot
Composés á structure imidazopyridinyl-arylpropénone, nouveaux agents anti-infectieux potentiels
inferred← citeshttps://doi.org/10.1016/j.drudis.2007.04.009openalex-snapshot
New developments in synthetic peroxidic drugs as artemisinin mimics
inferred← citeshttps://doi.org/10.1016/j.ejmech.2004.05.009openalex-snapshot
3D QSAR studies on antimalarial alkoxylated and hydroxylated chalcones by CoMFA and CoMSIA
inferred← citeshttps://doi.org/10.1016/j.ejmech.2005.03.013openalex-snapshot
Synthesis and antimalarial activity of E-2-quinolinylbenzocycloalcanones
inferred← citeshttps://doi.org/10.1016/j.ejmech.2006.09.019openalex-snapshot
A review of anti-infective and anti-inflammatory chalcones
inferred← citeshttps://doi.org/10.1016/j.ejmech.2007.01.001openalex-snapshot
Synthesis and evaluation of sulfonylurea derivatives as novel antimalarials
inferred← citeshttps://doi.org/10.1016/j.ejmech.2007.09.014openalex-snapshot
Synthesis of novel substituted 1,3-diaryl propenone derivatives and their antimalarial activity in vitro
inferred← citeshttps://doi.org/10.1016/j.ejmech.2008.09.044openalex-snapshot
Synthesis of chlorovinyl sulfones as structural analogs of chalcones and their antiplasmodial activities
inferred← citeshttps://doi.org/10.1016/j.ejmech.2009.02.008openalex-snapshot
Antimalarial pharmacodynamics of chalcone derivatives in combination with artemisinin against Plasmodium falciparum in vitro
inferred← citeshttps://doi.org/10.1016/j.ejmech.2009.10.037openalex-snapshot
Synthesis of some new S-triazine based chalcones and their derivatives as potent antimicrobial agents
inferred← citeshttps://doi.org/10.1016/j.ejmech.2009.11.022openalex-snapshot
Synthesis of new chalcone derivatives containing acridinyl moiety with potential antimalarial activity
inferred← citeshttps://doi.org/10.1016/j.ejmech.2010.08.049openalex-snapshot
Reinvestigation of structure–activity relationship of methoxylated chalcones as antimalarials: Synthesis and evaluation of 2,4,5-trimethoxy substituted patterns as lead candidates derived from abundantly available natural β-asarone
inferred← citeshttps://doi.org/10.1016/j.ejmech.2011.07.019openalex-snapshot
Quinolinyl and quinolinyl N-oxide chalcones: Synthesis, antifungal and cytotoxic activities
inferred← citeshttps://doi.org/10.1016/j.ejmech.2012.05.041openalex-snapshot
Design and synthesis of new (E)-cinnamic N-acylhydrazones as potent antitrypanosomal agents
inferred← citeshttps://doi.org/10.1016/j.ejmech.2012.08.039openalex-snapshot
Synthesis of novel quinoline-2-one based chalcones of potential anti-tumor activity
inferred← citeshttps://doi.org/10.1016/j.ejmech.2013.01.027openalex-snapshot
Synthesis, structure activity relationship and mode of action of 3-substitutedphenyl-1-(2,2,8,8-tetramethyl-3,4,9,10-tetrahydro-2 H ,8 H -pyrano[2,3- f ]chromen-6-yl)-propenones as novel anticancer agents in human leukaemia HL-60 cells
inferred← citeshttps://doi.org/10.1016/j.ejmech.2014.03.079openalex-snapshot
Design, economical synthesis and antiplasmodial evaluation of vanillin derived allylated chalcones and their marked synergism with artemisinin against chloroquine resistant strains of Plasmodium falciparum
inferred← citeshttps://doi.org/10.1016/j.ejmech.2014.05.077openalex-snapshot
Design, synthesis and biological evaluation of hybrid bioisoster derivatives of N-acylhydrazone and furoxan groups with potential and selective anti-Trypanosoma cruzi activity
inferred← citeshttps://doi.org/10.1016/j.ejmech.2014.07.087openalex-snapshot
Synthesis, biological evaluation and molecular docking of novel chalcone–coumarin hybrids as anticancer and antimalarial agents
inferred← citeshttps://doi.org/10.1016/j.ejmech.2015.06.052openalex-snapshot
Chalcone scaffolds as anti-infective agents: Structural and molecular target perspectives
inferred← citeshttps://doi.org/10.1016/j.ejmech.2016.08.042openalex-snapshot
Sulfonamide chalcones: Synthesis and in vitro exploration for therapeutic potential against Brugia malayi
inferred← citeshttps://doi.org/10.1016/j.ejmech.2016.09.044openalex-snapshot
4-Aminoquinoline-ferrocenyl-chalcone conjugates: Synthesis and anti-plasmodial evaluation
inferred← citeshttps://doi.org/10.1016/j.ejmech.2017.11.045openalex-snapshot
Cytotoxicity, molecular modeling, cell cycle arrest, and apoptotic induction induced by novel tetrahydro-[1,2,4]triazolo[3,4-a]isoquinoline chalcones
inferred← citeshttps://doi.org/10.1016/j.ejmech.2018.08.012openalex-snapshot
An update on small molecule strategies targeting leishmaniasis
inferred← citeshttps://doi.org/10.1016/j.ejmech.2020.112215openalex-snapshot
Chalcone hybrids as privileged scaffolds in antimalarial drug discovery: A key review
inferred← citeshttps://doi.org/10.1016/j.ejps.2005.09.007openalex-snapshot
Antiplasmodial activity of ferrocenyl chalcones: Investigations into the role of ferrocene
inferred← citeshttps://doi.org/10.1016/j.ejps.2013.09.019openalex-snapshot
Binary classification of chalcone derivatives with LDA or KNN based on their antileishmanial activity and molecular descriptors selected using the Successive Projections Algorithm feature-selection technique
inferred← citeshttps://doi.org/10.1016/j.ejps.2013.12.018openalex-snapshot
Design, synthesis and docking studies of bischalcones based quinazoline-2(1H)-ones and quinazoline-2(1H)-thiones derivatives as novel inhibitors of cathepsin B and cathepsin H
inferred← citeshttps://doi.org/10.1016/j.exppara.2009.12.007openalex-snapshot
Plasmodium falciparum: In vitro interaction of quassin and neo-quassin with artesunate, a hemisuccinate derivative of artemisinin
inferred← citeshttps://doi.org/10.1016/j.exppara.2017.02.006openalex-snapshot
Design, in silico and in vitro evaluation of curcumin analogues against Plasmodium falciparum
inferred← citeshttps://doi.org/10.1016/j.farmac.2005.01.005openalex-snapshot
Synthesis and antimalarial activity of sulfonamide chalcone derivatives
inferred← citeshttps://doi.org/10.1016/j.fct.2010.04.030openalex-snapshot
Xanthohumol feeding does not impair organ function and homoeostasis in mice
inferred← citeshttps://doi.org/10.1016/j.heliyon.2022.e08939openalex-snapshot
Coumaro-chalcones synthesized under solvent-free conditions as potential agents against malaria, leishmania and trypanosomiasis
inferred← citeshttps://doi.org/10.1016/j.ijbiomac.2015.07.029openalex-snapshot
Chalcones, semicarbazones and pyrazolines as inhibitors of cathepsins B, H and L
inferred← citeshttps://doi.org/10.1016/j.ijbiomac.2025.142817openalex-snapshot
Falcipain-2: A review on structurally diverse non-peptide inhibitors
inferred← citeshttps://doi.org/10.1016/j.ijpara.2004.10.003openalex-snapshot
Cysteine proteases of malaria parasites
inferred← citeshttps://doi.org/10.1016/j.jcat.2003.09.012openalex-snapshot
Activated hydrotalcites as catalysts for the synthesis of chalcones of pharmaceutical interest
inferred← citeshttps://doi.org/10.1016/j.jcat.2005.04.007openalex-snapshot
Catalytic applications of aminopropylated mesoporous silica prepared by a template-free route in flavanones synthesis
inferred← citeshttps://doi.org/10.1016/j.jics.2021.100028openalex-snapshot
Overview on cumulative synthetic approaches for chalcone based functionalized scaffolds
inferred← citeshttps://doi.org/10.1016/j.jtbi.2016.05.019openalex-snapshot
Comparative molecular field analysis and molecular docking studies on novel aryl chalcone derivatives against an important drug target cysteine protease in Plasmodium falciparum
inferred← citeshttps://doi.org/10.1016/j.matpr.2023.06.088openalex-snapshot
Synthesis, characterization and antimicrobial property of novel series of 3-(4-substituted phenyl)-1-(4-((4-morpholino-6-((4-nitrophenyl)amino)-1,3,5-triazin-2-yl)amino)phenyl) prop −2-en-1-one conjugates
inferred← citeshttps://doi.org/10.1016/j.mimet.2014.06.014openalex-snapshot
The 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyl tetrazolium bromide (MTT) assay is a rapid, cheap, screening test for the in vitro anti-tuberculous activity of chalcones
inferred← citeshttps://doi.org/10.1016/j.molcata.2005.08.039openalex-snapshot
LiOH·H2O as a novel dual activation catalyst for highly efficient and easy synthesis of 1,3-diaryl-2-propenones by Claisen–Schmidt condensation under mild conditions
inferred← citeshttps://doi.org/10.1016/j.molcata.2007.04.040openalex-snapshot
Sulfonic acid functionalized mesoporous silicas and organosilicas: Synthesis, characterization and catalytic applications
inferred← citeshttps://doi.org/10.1016/j.molcata.2007.10.021openalex-snapshot
Brønsted acidic ionic liquids as dual catalyst and solvent for environmentally friendly synthesis of chalcone
inferred← citeshttps://doi.org/10.1016/j.molstruc.2013.01.013openalex-snapshot
Studies on molecular weaker interactions, spectroscopic analysis and chemical reactivity of synthesized ethyl 3,5-dimethyl-4-[3-(2-nitro-phenyl)-acryloyl]-1H-pyrrole-2-carboxylate through experimental and quantum chemical approaches
inferred← citeshttps://doi.org/10.1016/j.molstruc.2014.12.062openalex-snapshot
Spectroscopic and quantum chemical correlation for structural evaluation, chemical reactivity and non-linear optical property investigation of two chalcone having pyrrole moiety: A comparative study
inferred← citeshttps://doi.org/10.1016/j.molstruc.2023.135530openalex-snapshot
Synthesis, biological evaluation and molecular docking study of oxindole based chalcone analogues as potent anti-Alzheimer agents
inferred← citeshttps://doi.org/10.1016/j.molstruc.2025.144910openalex-snapshot
Host-guest chemistry: Novel macrocyclic crown chalcone- ether hybrids; Design, synthesis, characterization, biological evaluations, molecular docking and color removal application
inferred← citeshttps://doi.org/10.1016/j.molstruc.2026.146315openalex-snapshot
Cytotoxicity, anti-proliferative, anti-inflammatory, anti-metastatic, and oxidative stress activities of novel cyanochalcones: Induction of apoptosis in HCT-116 cells
inferred← citeshttps://doi.org/10.1016/j.mycmed.2016.03.002openalex-snapshot
Antimicrobial effects of Piper hispidum extract, fractions and chalcones against Candida albicans and Staphylococcus aureus
inferred← citeshttps://doi.org/10.1016/j.optlastec.2012.07.023openalex-snapshot
Optical properties and inclusion of an organic fluorophore in organized media of micellar solutions and beta-cyclodextrin
inferred← citeshttps://doi.org/10.1016/j.optmat.2018.07.036openalex-snapshot
Theoretical and experimental approach to the investigation of hyperpolarizability and charge transfer characteristics of NLO active 2′,3,4,4′,5-pentamethoxy chalcone with silver atoms adsorbed
inferred← citeshttps://doi.org/10.1016/j.phytol.2009.01.002openalex-snapshot
Antiplasmodial β-hydroxydihydrochalcone from seedpods of Tephrosia elata
inferred← citeshttps://doi.org/10.1016/j.plantsci.2024.112015openalex-snapshot
PbWRKY18 promotes resistance against black spot disease by activation of the chalcone synthase gene PbCHS3 in pear
inferred← citeshttps://doi.org/10.1016/j.rechem.2022.100456openalex-snapshot
Recent advances on analytical methodologies for screening and detection of biophenols and their challenges: A brief review
inferred← citeshttps://doi.org/10.1016/j.saa.2009.09.048openalex-snapshot
Some fluorescence properties of dimethylaminochalcone and its novel cyclic analogues
inferred← citeshttps://doi.org/10.1016/j.sciaf.2026.e03393openalex-snapshot
Optimizing antimalarial discovery: A robust machine learning framework for chalcone bioactivity prediction using ensemble classifiers and oversampling strategies
inferred← citeshttps://doi.org/10.1016/j.tet.2021.132472openalex-snapshot
Manganese(I) catalyzed cross-coupling of secondary allylic alcohols and primary alcohols
inferred← citeshttps://doi.org/10.1016/j.tetlet.2007.03.054openalex-snapshot
A simple and highly efficient method for the synthesis of chalcones by using borontrifluoride-etherate
inferred← citeshttps://doi.org/10.1016/j.tetlet.2011.08.120openalex-snapshot
A new chemical access for 3′-acetyl-4′-hydroxychalcones using borontrifluoride–etherate via a regioselective Claisen-Schmidt condensation and its application in the synthesis of chalcone hybrids
inferred← citeshttps://doi.org/10.1016/s0031-9422(03)00373-xopenalex-snapshot
Anti-plasmodial activities and X-ray crystal structures of rotenoids from Millettia usaramensis subspecies usaramensis
inferred← citeshttps://doi.org/10.1016/s0039-9140(98)00120-9openalex-snapshot
News analytical reagents for europium(III)
inferred← citeshttps://doi.org/10.1016/s0065-308x(08)60242-0openalex-snapshot
Proteases of Protozoan Parasites
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