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Discovery of Nonpeptidic Small-Molecule AP-1 Inhibitors: Lead Hopping Based on a Three-Dimensional Pharmacophore Model
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What this work says
Outgoing claims: the papers this work cites, builds on, or argues with.
inferredcites →https://doi.org/10.1002/anie.199416991openalex-snapshot
Peptidomimetics—Tailored Enzyme Inhibitors
inferredcites →https://doi.org/10.1016/s0040-4039(00)99616-3openalex-snapshot
New coupling reagents in peptide chemistry
inferredcites →https://doi.org/10.1016/s0304-3835(97)00543-0openalex-snapshot
Inhibition of fos–jun–DNA complex formation by dihydroguaiaretic acid and in vitro cytotoxic effects on cancer cells
inferredcites →https://doi.org/10.1016/s1359-6446(01)02091-8openalex-snapshot
Virtual screening and fast automated docking methods
inferredcites →https://doi.org/10.1016/s1359-6446(02)02289-4openalex-snapshot
Genome annotation techniques: new approaches and challenges
inferredcites →https://doi.org/10.1021/ja00359a015openalex-snapshot
Resonance Raman spectra of rubredoxin, desulforedoxin, and the synthetic analog Fe(S2-o-xyl)2: conformational effects
inferredcites →https://doi.org/10.1021/ja00439a041openalex-snapshot
tert-Butoxycarbonylaminoacyl-4-(oxymethyl)phenylacetamidomethyl-resin, a more acid-resistant support for solid-phase peptide synthesis
inferredcites →https://doi.org/10.1021/ja00439a042openalex-snapshot
Reaction of hydroxylamine with ethyl acetoacetate. Details of the addition and cyclization steps studied by flow nuclear magnetic resonance
inferredcites →https://doi.org/10.1021/ja01336a041openalex-snapshot
Studies on the Rearrangement of Tertiary-butylmethylcarbinol (Pinacolyl Alcohol). II.1 Dehydration
inferredcites →https://doi.org/10.1021/jm00073a001openalex-snapshot
Concepts and progress in the development of peptide mimetics
inferredcites →https://doi.org/10.1021/jm049501bopenalex-snapshot
“Lead Hopping”. Validation of Topomer Similarity as a Superior Predictor of Similar Biological Activities
inferredcites →https://doi.org/10.1021/jm049890+openalex-snapshot
Design, Synthesis, and Biological Evaluation of New Cyclic Disulfide Decapeptides That Inhibit the Binding of AP-1 to DNA
inferredcites →https://doi.org/10.1021/jo00354a037openalex-snapshot
Selective oxidation of aldehydes to carboxylic acids with sodium chlorite-hydrogen peroxide
inferredcites →https://doi.org/10.1021/jo00354a038openalex-snapshot
Synthesis of novel 6H-1,3-oxazine derivatives with perfluoroalkyl substituents
inferredcites →https://doi.org/10.1021/jo00386a014openalex-snapshot
Total synthesis of isoflavones: jamaicin, calopogonium isoflavone-B, pseudobaptigenin, and maxima substance-B. Friedel-Crafts acylation reactions with acid-sensitive substrates
inferredcites →https://doi.org/10.1021/jo00386a015openalex-snapshot
Synthesis of ring-expanded cytidine: homocytidine
inferredcites →https://doi.org/10.1038/373261a0openalex-snapshot
F-actin binding site masked by the intramolecular association of vinculin head and tail domains
inferredcites →https://doi.org/10.1038/nrd1799openalex-snapshot
Computer-based de novo design of drug-like molecules
inferredcites →https://doi.org/10.1107/s0567740874002615openalex-snapshot
The crystal structure of bis(pyrazine-2-carboxamide)copper(II) perchlorate. Errata
inferredcites →https://doi.org/10.1172/jci119277openalex-snapshot
Studies on the contribution of c-fos/AP-1 to arthritic joint destruction.
inferredcites →https://doi.org/10.2174/0929867003374499openalex-snapshot
Conformational and Topographical Considerations in Designing Agonist Peptidomimetics from Peptide Leads
inferredcites →https://doi.org/10.7164/antibiotics.51.539openalex-snapshot
K1115 A, a New Anthraquinone Derivative that Inhibits the Binding of Activator Protein-1(AP-1) to its Recognition Sites. I. Biological Activities.
What points at this work
Incoming claims: where this work appears in other papers’ reference lists and arguments.
inferred← citeshttps://doi.org/10.2139/ssrn.4803185openalex-extracted
Novel Arylidene Thiobarbiturate Derivatives as Selective Acetylcholinesterase, Α-Glucosidase, and Nonclassical Human Carbonic Anhydrase Inhibitors: Biological Activity and Molecular Modeling Study
inferred← citeshttps://doi.org/10.1002/advs.202205161openalex-snapshot
Blockade of Activin Receptor IIB Protects Arthritis Pathogenesis by Non‐Amplification of Activin A‐ACVR2B‐NOX4 Axis Pathway
inferred← citeshttps://doi.org/10.1002/cmdc.200800355openalex-snapshot
SHOP: A Method For Structure‐Based Fragment and Scaffold Hopping
inferred← citeshttps://doi.org/10.1002/jcb.30543openalex-snapshot
AP‐1/C‐FOS and AP‐1/FRA2 differentially regulate early and late adipogenic differentiation of mesenchymal stem cells
inferred← citeshttps://doi.org/10.1007/978-3-7091-1428-5_7openalex-snapshot
Insights into Roles of Immediate-Early Genes in Angiogenesis
inferred← citeshttps://doi.org/10.1007/s10529-012-1022-4openalex-snapshot
T-5224, a selective inhibitor of c-Fos/activator protein-1, attenuates lipopolysaccharide-induced liver injury in mice
inferred← citeshttps://doi.org/10.1016/j.bbalip.2019.03.002openalex-snapshot
Sustained phospholipase C stimulation of H9c2 cardiomyoblasts by vasopressin induces an increase in CDP-diacylglycerol synthase 1 (CDS1) through protein kinase C and cFos
inferred← citeshttps://doi.org/10.1016/j.bbrc.2018.02.147openalex-snapshot
A selective c-Fos/AP-1 inhibitor prevents cartilage destruction and subsequent osteophyte formation
inferred← citeshttps://doi.org/10.1016/j.bbrep.2017.09.006openalex-snapshot
Activation of TPA-response element present in human Lemur Tyrosine Kinase 2 ( lmtk2 ) gene increases its expression
inferred← citeshttps://doi.org/10.1016/j.bioorg.2024.107613openalex-snapshot
Novel PROTAC probes targeting FOSL1 degradation to eliminate head and neck squamous cell carcinoma cancer stem cells
inferred← citeshttps://doi.org/10.1016/j.bmc.2014.01.009openalex-snapshot
Chemical constituents of Plectranthus amboinicus and the synthetic analogs possessing anti-inflammatory activity
inferred← citeshttps://doi.org/10.1016/j.ejmech.2008.12.006openalex-snapshot
3D-QSAR studies on the inhibitors of AP-1 and NF-κB mediated transcriptional activation
inferred← citeshttps://doi.org/10.1016/j.ijbiomac.2024.138649openalex-snapshot
Long non-coding RNA MMTP mediates necroptosis in alveolar macrophages during Mycoplasma hyopneumoniae infection by enhancing TNF-α transcription
inferred← citeshttps://doi.org/10.1016/j.neurot.2025.e00807openalex-snapshot
Uncovering the role of c-Fos in the bidirectional relationship between depression/anxiety behaviors and α-synuclein propagation in Parkinson’s disease
inferred← citeshttps://doi.org/10.1016/j.phytochem.2009.03.015openalex-snapshot
Fungal transformation of isosteviol lactone and its biological evaluation for inhibiting the AP-1 transcription factor
inferred← citeshttps://doi.org/10.1021/cr400713ropenalex-snapshot
Pathological Unfoldomics of Uncontrolled Chaos: Intrinsically Disordered Proteins and Human Diseases
inferred← citeshttps://doi.org/10.1021/jm070568jopenalex-snapshot
Probing Binding Requirements of Type I and Type II Isoforms of Inosine Monophosphate Dehydrogenase with Adenine-Modified Nicotinamide Adenine Dinucleotide Analogues
inferred← citeshttps://doi.org/10.1021/jm5004733openalex-snapshot
Small Molecule Inhibitors Targeting Activator Protein 1 (AP-1)
inferred← citeshttps://doi.org/10.1021/ol702403ropenalex-snapshot
Synthesis and Cytotoxicity of a New Class of Potent Decapeptide Macrocycles
inferred← citeshttps://doi.org/10.1038/nbt1412openalex-snapshot
Treatment of arthritis with a selective inhibitor of c-Fos/activator protein-1
inferred← citeshttps://doi.org/10.1038/s41467-021-25918-4openalex-snapshot
Determinants of renal cell carcinoma invasion and metastatic competence
inferred← citeshttps://doi.org/10.1038/s41586-026-10258-4openalex-snapshot
Epigenetic memory of colitis promotes tumour growth
inferred← citeshttps://doi.org/10.1038/s41598-017-17289-yopenalex-snapshot
A selective inhibition of c-Fos/activator protein-1 as a potential therapeutic target for intervertebral disc degeneration and associated pain
inferred← citeshttps://doi.org/10.1038/sj.bjp.0707306openalex-snapshot
In silicopharmacology for drug discovery: applications to targets and beyond
inferred← citeshttps://doi.org/10.1039/c2md00289bopenalex-snapshot
Small-molecule inhibitors of dimeric transcription factors: Antagonism of protein–protein and protein–DNA interactions
inferred← citeshttps://doi.org/10.1039/c5ra10831dopenalex-snapshot
Probing the binding mechanism of novel dual NF-κB/AP-1 inhibitors by 3D-QSAR, docking and molecular dynamics simulations
inferred← citeshttps://doi.org/10.1093/eurheartj/ehad679openalex-snapshot
On target inhibition of vascular smooth muscle cell phenotypic transition underpins TNF–OXPHOS–AP-1 as a promising avenue for anti-remodelling interventions in aortic dissection and rupture
inferred← citeshttps://doi.org/10.1101/2025.02.13.638099openalex-snapshot
Clonal memory of colitis accumulates and promotes tumor growth
inferred← citeshttps://doi.org/10.1124/dmd.110.037952openalex-snapshot
Metabolism of the c-Fos/Activator Protein-1 Inhibitor T-5224 by Multiple Human UDP-Glucuronosyltransferase Isoforms
inferred← citeshttps://doi.org/10.1161/atvbaha.120.315622openalex-snapshot
ODC (Ornithine Decarboxylase)-Dependent Putrescine Synthesis Maintains MerTK (MER Tyrosine-Protein Kinase) Expression to Drive Resolution
inferred← citeshttps://doi.org/10.1186/s12890-021-01801-2openalex-snapshot
c-Fos is a mechanosensor that regulates inflammatory responses and lung barrier dysfunction during ventilator-induced acute lung injury
inferred← citeshttps://doi.org/10.1186/s12916-026-04757-4openalex-snapshot
Identification of cryosensitive niches and a targetable FOS/AP‑1 program in the human ovarian cortex by single‑cell and spatial transcriptomics
inferred← citeshttps://doi.org/10.1186/s12967-024-04933-1openalex-snapshot
The siRNA-mediated knockdown of AP-1 restores the function of the pulmonary artery and the right ventricle by reducing perivascular and interstitial fibrosis and key molecular players in cardiopulmonary disease
inferred← citeshttps://doi.org/10.1186/s40560-015-0115-2openalex-snapshot
T-5224, a selective inhibitor of c-Fos/activator protein-1, improves survival by inhibiting serum high mobility group box-1 in lethal lipopolysaccharide-induced acute kidney injury model
inferred← citeshttps://doi.org/10.1517/17460441.2.4.453openalex-snapshot
Conotoxin therapeutics: a pipeline for success?
inferred← citeshttps://doi.org/10.18632/oncotarget.25781openalex-snapshot
Chromatin-associated APC regulates gene expression in collaboration with canonical WNT signaling and AP-1
inferred← citeshttps://doi.org/10.21203/rs.3.rs-6312954/v1openalex-snapshot
Spatiotemporal Dynamics of Human Ovarian Cortex Transcriptome Following Vitrification and Thawing: Insights into the FOS/AP-1 Pathway
inferred← citeshttps://doi.org/10.2741/3001openalex-snapshot
Transcription factors in autoimmune diseases
inferred← citeshttps://doi.org/10.3923/ijp.2013.176.181openalex-snapshot
The Pros and Cons of the In-silico Pharmaco-toxicology in Drug Discovery and Development
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