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ERβ Ligands. 3. Exploiting Two Binding Orientations of the 2-Phenylnaphthalene Scaffold To Achieve ERβ Selectivity
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What this work says
Outgoing claims: the papers this work cites, builds on, or argues with.
inferredcites →https://doi.org/10.1016/0014-5793(96)00782-xopenalex-snapshot
ERβ: Identification and characterization of a novel human estrogen receptor
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In vitro characterization of trimegestone: a new potent and selective progestin
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The ligand binding profiles of estrogen receptors α and β are species dependent
inferredcites →https://doi.org/10.1016/s0039-128x(96)00242-5openalex-snapshot
The estradiol pharmacophore: Ligand structure-estrogen receptor binding affinity relationships and a model for the receptor binding site
inferredcites →https://doi.org/10.1016/s0076-6879(97)76067-1openalex-snapshot
[21] Data collection strategy
inferredcites →https://doi.org/10.1016/s0968-0896(03)00303-1openalex-snapshot
ERβ Ligands. Part 1: The discovery of ERβ selective ligands which embrace the 4-hydroxy-biphenyl template
inferredcites →https://doi.org/10.1021/ja047633oopenalex-snapshot
Structure-Based Design of Estrogen Receptor-β Selective Ligands
inferredcites →https://doi.org/10.1021/jm010254aopenalex-snapshot
Estrogen Receptor-β Potency-Selective Ligands: Structure−Activity Relationship Studies of Diarylpropionitriles and Their Acetylene and Polar Analogues
inferredcites →https://doi.org/10.1021/jm015577lopenalex-snapshot
Toward Selective ERβ Agonists for Central Nervous System Disorders: Synthesis and Characterization of Aryl Benzthiophenes
inferredcites →https://doi.org/10.1021/jm020291hopenalex-snapshot
A New Series of Estrogen Receptor Modulators That Display Selectivity for Estrogen Receptor β
inferredcites →https://doi.org/10.1021/jm049719yopenalex-snapshot
Design and Synthesis of Aryl Diphenolic Azoles as Potent and Selective Estrogen Receptor-β Ligands
inferredcites →https://doi.org/10.1021/jm981064bopenalex-snapshot
Flavonoid-Related Modulators of Multidrug Resistance: Synthesis, Pharmacological Activity, and Structure−Activity Relationships
inferredcites →https://doi.org/10.1021/jm990101bopenalex-snapshot
Estrogen Receptor Subtype-Selective Ligands: Asymmetric Synthesis and Biological Evaluation of cis- and trans-5,11-Dialkyl- 5,6,11,12-tetrahydrochrysenes
inferredcites →https://doi.org/10.1021/tx000208yopenalex-snapshot
Structure−Activity Relationships for a Large Diverse Set of Natural, Synthetic, and Environmental Estrogens
inferredcites →https://doi.org/10.1023/a:1007907728892openalex-snapshot
QXP: Powerful, rapid computer algorithms for structure-based drug design
inferredcites →https://doi.org/10.1038/39645openalex-snapshot
Molecular basis of agonism and antagonism in the oestrogen receptor
inferredcites →https://doi.org/10.1038/39651openalex-snapshot
Structure at 1.65 Å of RhoA and its GTPase-activating protein in complex with a transition-state analogue
inferredcites →https://doi.org/10.1039/b305991jopenalex-snapshot
Solution and solid state 13 C NMR and X-ray studies of genistein complexes with amines. Potential biological function of the C-7, C-5, and C-4′-OH groups
inferredcites →https://doi.org/10.1073/pnas.95.11.5998openalex-snapshot
Crystallographic comparison of the estrogen and progesterone receptor’s ligand binding domains
inferredcites →https://doi.org/10.1074/jbc.m009404200openalex-snapshot
Core LXXLL Motif Sequences in CREB-binding Protein, SRC1, and RIP140 Define Affinity and Selectivity for Steroid and Retinoid Receptors
inferredcites →https://doi.org/10.1074/jbc.m200764200openalex-snapshot
Interaction of Transcriptional Intermediary Factor 2 Nuclear Receptor Box Peptides with the Coactivator Binding Site of Estrogen Receptor α
inferredcites →https://doi.org/10.1107/s0021889892009282openalex-snapshot
The FROG PC series: programs for electron-density and model investigations for proteins
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Structure of trypanothione reductase from Crithidia fasciculata at 2.6 Å resolution; enzyme–NADP interactions at 2.8 Å resolution
inferredcites →https://doi.org/10.1210/endo.138.11.5496openalex-snapshot
Tissue Distribution and Quantitative Analysis of Estrogen Receptor-α (ERα) and Estrogen Receptor-β (ERβ) Messenger Ribonucleic Acid in the Wild-Type and ERα-Knockout Mouse
inferredcites →https://doi.org/10.1210/endo.139.10.6216openalex-snapshot
Interaction of Estrogenic Chemicals and Phytoestrogens with Estrogen Receptor β
inferredcites →https://doi.org/10.2133/dmpk.17.221openalex-snapshot
Sulfation of Environmental Estrogens by Cytosolic Human Sulfotransferases
inferredcites →https://doi.org/10.2174/1568026033451727openalex-snapshot
Estrogen Receptor Modulators: Relationships of Ligand Structure, Receptor Affinity and Functional Activity
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Selective direct C–H polyfluoroarylation of electron-deficient N-heterocyclic compounds
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inferred← citeshttps://doi.org/10.1039/d1ob01619aopenalex-snapshot
MeOTf/KI-catalyzed efficient synthesis of 2-arylnaphthalenes via cyclodimerization of styrene oxides
inferred← citeshttps://doi.org/10.1055/s-0042-1751376openalex-snapshot
Lewis Acid Promoted Homodimerization of Styrene Diols: An Efficient Approach toward 2-Phenylnaphthalenes
inferred← citeshttps://doi.org/10.1073/pnas.1603486113openalex-snapshot
Mutant cycle analysis with modified saxitoxins reveals specific interactions critical to attaining high-affinity inhibition of hNa V 1.7
inferred← citeshttps://doi.org/10.1073/pnas.1702211114openalex-snapshot
Estrogen receptor β, a regulator of androgen receptor signaling in the mouse ventral prostate
inferred← citeshttps://doi.org/10.1074/jbc.m513684200openalex-snapshot
Identification of Ligands with Bicyclic Scaffolds Provides Insights into Mechanisms of Estrogen Receptor Subtype Selectivity
inferred← citeshttps://doi.org/10.1080/10629360701698811openalex-snapshot
Quantitative structure-activity relationships for a series of selective estrogen receptor-beta modulators
inferred← citeshttps://doi.org/10.1080/14756360701503232openalex-snapshot
Benzothiepin-derived molecular scaffolds for estrogen receptor modulators: synthesis and antagonistic effects in breast cancer cells
inferred← citeshttps://doi.org/10.1086/651276openalex-snapshot
Estrogen Receptor β Agonism Increases Survival in Experimentally Induced Sepsis and Ameliorates the Genomic Sepsis Signature: A Pharmacogenomic Study
inferred← citeshttps://doi.org/10.1097/01.ccm.0000227173.13497.56openalex-snapshot
WAY-202196, a selective estrogen receptor-beta agonist, protects against death in experimental septic shock
inferred← citeshttps://doi.org/10.1101/2025.08.14.670313openalex-snapshot
Estrogen Receptor Beta Activation Coordinates Liver Lipid Remodeling and Metabolic Fluxes, Preventing Lipotoxicity
inferred← citeshttps://doi.org/10.1111/j.1747-0285.2011.01119.xopenalex-snapshot
Multiple‐Targeting and Conformational Selection in the Estrogen Receptor: Computation and Experiment
inferred← citeshttps://doi.org/10.1126/science.aan1568openalex-snapshot
Snap deconvolution: An informatics approach to high-throughput discovery of catalytic reactions
inferred← citeshttps://doi.org/10.1142/9781848169586_0006openalex-snapshot
CLUES ABOUT ESTROGEN AND ANTIESTROGEN ACTION FROM X-RAY CRYSTALLOGRAPHY
inferred← citeshttps://doi.org/10.1142/9781848169586_0013openalex-snapshot
NOVEL SELECTIVE ESTROGEN RECEPTOR MODULATORS
inferred← citeshttps://doi.org/10.1152/physrev.00026.2006openalex-snapshot
Estrogen Receptors: How Do They Signal and What Are Their Targets
inferred← citeshttps://doi.org/10.1210/me.2005-0459openalex-snapshot
Estrogen Receptor-β: Recent Lessons from in Vivo Studies
inferred← citeshttps://doi.org/10.1210/me.2009-0288openalex-snapshot
Minireview: Estrogen Receptor-β: Mechanistic Insights from Recent Studies
inferred← citeshttps://doi.org/10.1371/journal.pone.0094209openalex-snapshot
The Role of Estrogen Signaling in a Mouse Model of Inflammatory Bowel Disease: A Helicobacter Hepaticus Model
inferred← citeshttps://doi.org/10.1371/journal.pone.0141184openalex-snapshot
Structure-Activity Relationship of Synthetic 2-Phenylnaphthalenes with Hydroxyl Groups that Inhibit Proliferation and Induce Apoptosis of MCF-7 Cancer Cells
inferred← citeshttps://doi.org/10.1517/13543771003657164openalex-snapshot
Estrogen receptor β selective nonsteroidal estrogens: seeking clinical indications
inferred← citeshttps://doi.org/10.1517/13543776.16.5.559openalex-snapshot
Estrogen receptor modulator review
inferred← citeshttps://doi.org/10.1621/nrs.04012openalex-snapshot
The Unexpected Science of Estrogen Receptor-β Selective Agonists: A New Class of Anti-Inflammatory Agents?
inferred← citeshttps://doi.org/10.1677/erc-07-0281openalex-snapshot
Implications of the binding of tamoxifen to the coactivator recognition site of the estrogen receptor
inferred← citeshttps://doi.org/10.18632/oncotarget.18313openalex-snapshot
Estrogen and estrogen receptors in the modulation of gastrointestinal epithelial secretion
inferred← citeshttps://doi.org/10.21007/etd.cghs.2011.0285openalex-snapshot
"Synthesis and Computational Studies on Hiv-1 Integrase Inhibitors"
inferred← citeshttps://doi.org/10.2174/1568026615666150413154841openalex-snapshot
Structural and Functional Diversity of Estrogen Receptor Ligands
inferred← citeshttps://doi.org/10.2174/157018011795514230openalex-snapshot
Synthesis and Biological Evaluation of Spiro-δ-lactones as Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 2 (17β-HSD2)
inferred← citeshttps://doi.org/10.22028/d291-22367openalex-snapshot
Design, Synthese und biologische Evaluierung von nichtsteroidalen, potenten und selektiven Inhibitoren der 17beta-Hydroxysteroid Dehydrogenase Typ 1 (17beta-HSD1)
inferred← citeshttps://doi.org/10.2478/s11532-010-0050-yopenalex-snapshot
Modeling the activity of 2-phenylnaphthalene inhibitors using self-training artificial neural networks
inferred← citeshttps://doi.org/10.2967/jnumed.116.180158openalex-snapshot
Synthesis and Evaluation of the Estrogen Receptor β–Selective Radioligand 2-18F-Fluoro-6-(6-Hydroxynaphthalen-2-yl)Pyridin-3-ol: Comparison with 16α-18F-Fluoro-17β-Estradiol
inferred← citeshttps://doi.org/10.3109/14756366.2014.959946openalex-snapshot
Receptor-based virtual screening evaluation for the identification of estrogen receptorβligands
inferred← citeshttps://doi.org/10.3389/fphar.2021.695712openalex-snapshot
IIIM-941, a Stilbene Derivative Inhibits NLRP3 Inflammasome Activation by Inducing Autophagy
inferred← citeshttps://doi.org/10.3390/ijerph110908709openalex-snapshot
Versatility or Promiscuity: The Estrogen Receptors, Control of Ligand Selectivity and an Update on Subtype Selective Ligands
inferred← citeshttps://doi.org/10.3390/ijms11093434openalex-snapshot
In Silico Prediction of Estrogen Receptor Subtype Binding Affinity and Selectivity Using Statistical Methods and Molecular Docking with 2-Arylnaphthalenes and 2-Arylquinolines
inferred← citeshttps://doi.org/10.3390/ijms25116238openalex-snapshot
TATA-Binding Protein-Based Virtual Screening of FDA Drugs Identified New Anti-Giardiasis Agents
inferred← citeshttps://doi.org/10.3390/ijms27010463openalex-snapshot
Multicomplex Pharmacophore Modeling of Estrogen Receptors Suggests the Probable Repurposing of Procaterol as an Antiproliferative Agent Against Breast Cancer Cells
inferred← citeshttps://doi.org/10.3390/molecules26092605openalex-snapshot
Predicting Accurate Lead Structures for Screening Molecular Libraries: A Quantum Crystallographic Approach
inferred← citeshttps://doi.org/10.3762/bjoc.12.79openalex-snapshot
Syntheses of dibenzo[d,d']benzo[2,1-b:3,4-b']difuran derivatives and their application to organic field-effect transistors
inferred← citeshttps://doi.org/10.3762/bjoc.6.48openalex-snapshot
Synthesis of fluorinated δ-lactams via cycloisomerization of gem-difluoropropargyl amides
inferred← citeshttps://doi.org/10.3892/ijo.2012.1615openalex-snapshot
The novel resveratrol analogue HS-1793 induces apoptosis via the mitochondrial pathway in murine breast cancer cells
inferred← citeshttps://doi.org/10.4049/jimmunol.180.1.630openalex-snapshot
Selective Estrogen Receptor-β Agonists Repress Transcription of Proinflammatory Genes
inferred← citeshttps://doi.org/10.70675/6d4b3bb2zc7adz43f3z857ez8de3c447fcfbopenalex-snapshot
La 7β-hydroxy-épiandrostérone dans des modèles in vitro de cancer du sein : effets anti-estrogéniques et rôle des récepteurs des estrogènes
inferred← citeshttps://doi.org/10.7717/peerj.11716openalex-snapshot
ERpred: a web server for the prediction of subtype-specific estrogen receptor antagonists
Editorial review for independent work. ICSAC — the Institute for Complexity
Science and Advanced Computing — runs a structured editorial panel for researchers
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