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Macrocycles Are Great Cycles: Applications, Opportunities, and Challenges of Synthetic Macrocycles in Drug Discovery
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Synthesis of small cyclic peptides via intramolecular Heck reactions
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Efficient approach for the diversity-oriented synthesis of macro-heterocycles on solid-support
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Rapid and efficient solid phase syntheses of cyclic peptides with endocyclic biaryl ether bonds
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Peptide-based inhibitors of the hepatitis C virus serine protease
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Macrocyclic hydroxamate inhibitors of matrix metalloproteinases and TNF-α production
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On-resin macrocyclization of peptides via intramolecular SnAr reactions
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Drug-like properties and the causes of poor solubility and poor permeability
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Product Inhibition of the Hepatitis C Virus NS3 Protease
inferredcites →https://doi.org/10.1021/bi990174xopenalex-snapshot
Molecular Recognition of Macrocyclic Peptidomimetic Inhibitors by HIV-1 Protease,
inferredcites →https://doi.org/10.1021/cc020076mopenalex-snapshot
Macrolactones in Diversity-Oriented Synthesis: Preparation of a Pilot Library and Exploration of Factors Controlling Macrocyclization
inferredcites →https://doi.org/10.1021/cc050064bopenalex-snapshot
Synthesis of a Library of Complex Macrodiolides Employing Cyclodimerization of Hydroxy Esters
inferredcites →https://doi.org/10.1021/cc060166hopenalex-snapshot
Diversity-Oriented Asymmetric Synthesis of Hapalosin: Construction of Three Small C9/C4/C3-Modified Hapalosin Analogue Libraries
inferredcites →https://doi.org/10.1021/cc800089mopenalex-snapshot
Combinatorial Synthesis of RGD Model Cyclic Peptides Utilizing a Palladium-Catalyzed Carbonylative Macrolactamization on a Polymer Support
inferredcites →https://doi.org/10.1021/cr0301402openalex-snapshot
Macrolactonizations in the Total Synthesis of Natural Products
inferredcites →https://doi.org/10.1021/cr040669eopenalex-snapshot
Proteases Universally Recognize Beta Strands In Their Active Sites
inferredcites →https://doi.org/10.1021/cr800278zopenalex-snapshot
Mitsunobu and Related Reactions: Advances and Applications
inferredcites →https://doi.org/10.1021/cr8003407openalex-snapshot
Multiple Multicomponent Macrocyclizations (MiBs): A Strategic Development Toward Macrocycle Diversity
inferredcites →https://doi.org/10.1021/cr900357eopenalex-snapshot
s -Tetrazines as Building Blocks for New Functional Molecules and Molecular Materials
inferredcites →https://doi.org/10.1021/cr900368aopenalex-snapshot
Update 1 of: Proteases Universally Recognize Beta Strands In Their Active Sites
inferredcites →https://doi.org/10.1021/ja00087a007openalex-snapshot
Template-Constrained Cyclic Peptides: Design of High-Affinity Ligands for GPIIb/IIIa
inferredcites →https://doi.org/10.1021/ja00147a026openalex-snapshot
Synthesis of peptidyl ruthenium .pi.-arene complexes: application to the synthesis of cyclic biphenyl ether peptides.
inferredcites →https://doi.org/10.1021/ja00151a029openalex-snapshot
Palladium-Mediated Macrocyclization on Solid Support and Its Applications to Combinatorial Synthesis
inferredcites →https://doi.org/10.1021/ja003673qopenalex-snapshot
Conformational Restriction of Flexible Ligands Guided by the Transferred NOE Experiment: Potent Macrocyclic Inhibitors of Farnesyltransferase
inferredcites →https://doi.org/10.1021/ja0256461openalex-snapshot
Conformationally Constrained Macrocycles That Mimic Tripeptide β-Strands in Water and Aprotic Solvents
inferredcites →https://doi.org/10.1021/ja0352202openalex-snapshot
Chemoenzymatic Route to Macrocyclic Hybrid Peptide/Polyketide-like Molecules
inferredcites →https://doi.org/10.1021/ja0455300openalex-snapshot
Structural Mimicry of Two Cytochromeb562Interhelical Loops Using Macrocycles Constrained by Oxazoles and Thiazoles
inferredcites →https://doi.org/10.1021/ja048170popenalex-snapshot
Relationship of Stereochemical and Skeletal Diversity of Small Molecules to Cellular Measurement Space
inferredcites →https://doi.org/10.1021/ja060720ropenalex-snapshot
Supramolecular Compounds from Multiple Ugi Multicomponent Macrocyclizations: Peptoid-based Cryptands, Cages, and Cryptophanes
inferredcites →https://doi.org/10.1021/ja102304popenalex-snapshot
Total Synthesis of Complestatin: Development of a Pd(0)-Mediated Indole Annulation for Macrocyclization
inferredcites →https://doi.org/10.1021/ja1047363openalex-snapshot
Development of a General, Sequential, Ring-Closing Metathesis/Intramolecular Cross-Coupling Reaction for the Synthesis of Polyunsaturated Macrolactones
inferredcites →https://doi.org/10.1021/ja104903xopenalex-snapshot
In Vitro Selection of a DNA-Templated Small-Molecule Library Reveals a Class of Macrocyclic Kinase Inhibitors
inferredcites →https://doi.org/10.1021/ja711120ropenalex-snapshot
Molecular Modeling Based Approach to Potent P2−P4 Macrocyclic Inhibitors of Hepatitis C NS3/4A Protease
inferredcites →https://doi.org/10.1021/ja803299hopenalex-snapshot
Acid Promoted Cinnamyl Ion Mobility within Peptide Derived Macrocycles
inferredcites →https://doi.org/10.1021/ja805097sopenalex-snapshot
Total Synthesis of (+)-Cassaine via Transannular Diels−Alder Reaction
inferredcites →https://doi.org/10.1021/ja805187popenalex-snapshot
Formal Synthesis of (−)-Kendomycin Featuring a Prins-Cyclization To Construct the Macrocycle
inferredcites →https://doi.org/10.1021/ja805649fopenalex-snapshot
Translation of DNA into a Library of 13 000 Synthetic Small-Molecule Macrocycles Suitable for in Vitro Selection
inferredcites →https://doi.org/10.1021/ja809005kopenalex-snapshot
Architectural Chemistry: Synthesis of Topologically Diverse Macromulticycles by Sequential Multiple Multicomponent Macrocyclizations
inferredcites →https://doi.org/10.1021/ja961626lopenalex-snapshot
Application of Ring-Closing Metathesis to the Synthesis of Rigidified Amino Acids and Peptides
inferredcites →https://doi.org/10.1021/ja963495uopenalex-snapshot
Novel Cyclic Biphenyl Ether Peptide β-Strand Mimetics and HIV-Protease Inhibitors
inferredcites →https://doi.org/10.1021/ja983859dopenalex-snapshot
Lactone and Lactam Library Synthesis by Silver Ion-Assisted Orthogonal Cyclization of Unprotected Peptides
inferredcites →https://doi.org/10.1021/ja992658mopenalex-snapshot
A Strategy for Macrocyclic Ring Closure and Functionalization Aimed toward Split-Pool Syntheses
inferredcites →https://doi.org/10.1021/jm00019a017openalex-snapshot
Quantitative structural activity relationship study of bis-tetraazacyclic compounds. A novel series of HIV-1 and HIV-2 inhibitors
inferredcites →https://doi.org/10.1021/jm00048a004openalex-snapshot
Design, Synthesis, and Conformational Analysis of a Novel Macrocyclic HIV-Protease Inhibitor
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Highly potent, orally active diester macrocyclic human renin inhibitors
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Hydrolysis of Iminium Ethers Derived from the Reaction of Ketones with Hydroxy Azides: Synthesis of Macrocyclic Lactams and Lactones
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What points at this work
Incoming claims: where this work appears in other papers’ reference lists and arguments.
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Macrocycles from Multicomponent Reactions
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Highly Substrate‐Selective Macrocyclic Ring Closing Metathesis
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Macrocyclic Protease Inhibitors with Reduced Peptide Character
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Two‐Step Synthesis of Complex Artificial Macrocyclic Compounds
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Peptid‐Diversifizierung durch positionsselektive C‐H‐Aktivierung im späten Synthesestadium
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Internal Nucleophilic Catalyst Mediated Cyclisation/Ring Expansion Cascades for the Synthesis of Medium‐Sized Lactones and Lactams
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Makrozyklische FKBP51‐Liganden enthüllen einen transienten Bindungsmodus mit erhöhter Selektivität
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Macrolactonization Reactions Driven by a Pentafluorobenzoyl Group**
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Synthesis of 20‐Membered Macrocyclic Pseudo‐Natural Products Yields Inducers of LC3 Lipidation
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Ring Expansion Strategies for the Synthesis of Medium Sized Ring and Macrocyclic Sulfonamides
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Non‐Dilute Synthesis of Macrodiolides and Macrotetrolides Enabled by Confinement Catalysis
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Macrocyclization of ω‐Isocyano Aldehydes
inferred← citeshttps://doi.org/10.1002/anie.201200110openalex-snapshot
Structure‐Based Macrocyclization Yields Hepatitis C Virus NS5B Inhibitors with Improved Binding Affinities and Pharmacokinetic Properties
inferred← citeshttps://doi.org/10.1002/anie.201404301openalex-snapshot
Macrocyclic Protease Inhibitors with Reduced Peptide Character
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Atom‐Economical Dimerization Strategy by the Rhodium‐Catalyzed Addition of Carboxylic Acids to Allenes: Protecting‐Group‐Free Synthesis of Clavosolide A and Late‐Stage Modification
inferred← citeshttps://doi.org/10.1002/anie.201508818openalex-snapshot
Scaffold Diversity Synthesis and Its Application in Probe and Drug Discovery
inferred← citeshttps://doi.org/10.1002/anie.201509153openalex-snapshot
The Synthesis of Structurally Diverse Macrocycles By Successive Ring Expansion
inferred← citeshttps://doi.org/10.1002/anie.201509240openalex-snapshot
Conformational Studies and Atropisomerism Kinetics of the ALK Clinical Candidate Lorlatinib (PF‐06463922) and Desmethyl Congeners
inferred← citeshttps://doi.org/10.1002/anie.201607188openalex-snapshot
Butelase‐Mediated Macrocyclization of d ‐Amino‐Acid‐Containing Peptides
inferred← citeshttps://doi.org/10.1002/anie.201610801openalex-snapshot
One‐Pot Assembly of Amino Acid Bridged Hybrid Macromulticyclic Cages through Multiple Multicomponent Macrocyclizations
inferred← citeshttps://doi.org/10.1002/anie.201611685openalex-snapshot
Diversity‐Oriented Synthesis of Cyclic Azapeptides by A3‐Macrocyclization Provides High‐Affinity CD36‐Modulating Peptidomimetics
inferred← citeshttps://doi.org/10.1002/anie.201704426openalex-snapshot
Two‐Step Synthesis of Complex Artificial Macrocyclic Compounds
inferred← citeshttps://doi.org/10.1002/anie.201803369openalex-snapshot
Enantioselective Rhodium‐Catalyzed Dimerization of ω‐Allenyl Carboxylic Acids: Straightforward Synthesis of C2‐Symmetric Macrodiolides
inferred← citeshttps://doi.org/10.1002/anie.201806250openalex-snapshot
Late‐Stage Peptide Diversification by Position‐Selective C−H Activation
inferred← citeshttps://doi.org/10.1002/anie.201811668openalex-snapshot
Late‐Stage Peptide Diversification through Cobalt‐Catalyzed C−H Activation: Sequential Multicatalysis for Stapled Peptides
inferred← citeshttps://doi.org/10.1002/anie.201907206openalex-snapshot
Internal Nucleophilic Catalyst Mediated Cyclisation/Ring Expansion Cascades for the Synthesis of Medium‐Sized Lactones and Lactams
inferred← citeshttps://doi.org/10.1002/anie.202017352openalex-snapshot
Macrocyclic FKBP51 Ligands Define a Transient Binding Mode with Enhanced Selectivity
inferred← citeshttps://doi.org/10.1002/anie.202105882openalex-snapshot
Macrolactonization Reactions Driven by a Pentafluorobenzoyl Group**
inferred← citeshttps://doi.org/10.1002/anie.202114328openalex-snapshot
Synthesis of 20‐Membered Macrocyclic Pseudo‐Natural Products Yields Inducers of LC3 Lipidation
inferred← citeshttps://doi.org/10.1002/anie.202216029openalex-snapshot
Cycling a Tether into Multiple Rings: Pt‐Bridged Macrocycles for Differentiated Guest Recognition, Pseudorotaxane Transformations, and Guest Capture and Release
inferred← citeshttps://doi.org/10.1002/anie.202217178openalex-snapshot
Ring Expansion Strategies for the Synthesis of Medium Sized Ring and Macrocyclic Sulfonamides
inferred← citeshttps://doi.org/10.1002/anie.202320045openalex-snapshot
A Tag‐Free Platform for Synthesis and Screening of Cyclic Peptide Libraries
inferred← citeshttps://doi.org/10.1002/anie.202418057openalex-snapshot
Diastereoselective Anomeric C(sp 3 )−H Cyclization Towards the Design of New Cyclophane‐Braced Glycopeptides
inferred← citeshttps://doi.org/10.1002/anie.202518622openalex-snapshot
Modular Synthesis of Pyritide‐Inspired Macrocycles Featuring Bipyridine Motifs
inferred← citeshttps://doi.org/10.1002/anie.6206059openalex-snapshot
Non‐Dilute Synthesis of Macrodiolides and Macrotetrolides Enabled by Confinement Catalysis
inferred← citeshttps://doi.org/10.1002/anie.6516584openalex-snapshot
Macrocyclization of ω‐Isocyano Aldehydes
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Understanding and designing head‐to‐tail cyclic peptides
inferred← citeshttps://doi.org/10.1002/bkcs.12604openalex-snapshot
Studies toward the total synthesis of (+)‐neopeltolide using N ‐heterocyclic carbene‐catalyzed oxo‐acyloxylation/reductive oxa‐Michael addition strategy
inferred← citeshttps://doi.org/10.1002/cbic.201200579openalex-snapshot
Macrocyclization of Organo‐Peptide Hybrids through a Dual Bio‐orthogonal Ligation: Insights from Structure–Reactivity Studies
inferred← citeshttps://doi.org/10.1002/cbic.201500179openalex-snapshot
Ribosomal Synthesis of Natural‐Product‐Like Bicyclic Peptides in Escherichia coli
inferred← citeshttps://doi.org/10.1002/cbic.201500441openalex-snapshot
Flexibility versus Rigidity for Orally Bioavailable Cyclic Hexapeptides
inferred← citeshttps://doi.org/10.1002/cbic.201700586openalex-snapshot
Enhanced Permeability and Binding Activity of Isobutylene‐Grafted Peptides
inferred← citeshttps://doi.org/10.1002/cbic.201800475openalex-snapshot
Synthesis of Macrocycles Derived from Substituted Triazines
inferred← citeshttps://doi.org/10.1002/cbic.201800751openalex-snapshot
Smart Design of Small‐Molecule Libraries: When Organic Synthesis Meets Cheminformatics
inferred← citeshttps://doi.org/10.1002/cbic.202200415openalex-snapshot
Harnessing the Therapeutic Potential and Biological Activity of Antiviral Peptides
inferred← citeshttps://doi.org/10.1002/cbic.202500188openalex-snapshot
Probing Thrombosis Initiation with Lasso Peptide Variants as Inhibitors to the von Willebrand Protein–Collagen Interaction
inferred← citeshttps://doi.org/10.1002/cbic.202500375openalex-snapshot
Enhancing Peptide Cyclization: Unveiling the Key Roles of Coupling Reagents and Heat for Optimal Results
inferred← citeshttps://doi.org/10.1002/cctc.202000111openalex-snapshot
Protection of Ruthenium Olefin Metathesis Catalysts by Encapsulation in a Self‐assembled Resorcinarene Capsule
inferred← citeshttps://doi.org/10.1002/chem.201202182openalex-snapshot
Tuning Chloride Binding, Encapsulation, and Transport by Peripheral Substitution of Pseudopeptidic Tripodal Small Cages
inferred← citeshttps://doi.org/10.1002/chem.201203266openalex-snapshot
Bending Rigid Molecular Rods: Formation of Oligoproline Macrocycles
inferred← citeshttps://doi.org/10.1002/chem.201203433openalex-snapshot
Exploiting Aggregation To Achieve Phase Separation in Macrocyclization
inferred← citeshttps://doi.org/10.1002/chem.201204260openalex-snapshot
Synthesis and Extended Activity of Triazole‐Containing Macrocyclic Protease Inhibitors
inferred← citeshttps://doi.org/10.1002/chem.201300664openalex-snapshot
Concise Synthesis and Biological Assessment of (+)‐Neopeltolide and a 16‐Member Stereoisomer Library of 8,9‐Dehydroneopeltolide: Identification of Pharmacophoric Elements
inferred← citeshttps://doi.org/10.1002/chem.201303453openalex-snapshot
Exocyclic Control of Turn Induction in Macrocyclic Peptide Scaffolds
inferred← citeshttps://doi.org/10.1002/chem.201303841openalex-snapshot
Synthesis and Conformational Analysis of Cyclic Homooligomers from Pyranoid ε‐Sugar Amino Acids
inferred← citeshttps://doi.org/10.1002/chem.201403117openalex-snapshot
Peptides Come Round: Using SICLOPPS Libraries for Early Stage Drug Discovery
inferred← citeshttps://doi.org/10.1002/chem.201404202openalex-snapshot
Macrocyclic Olefin Metathesis at High Concentrations by Using a Phase‐Separation Strategy
inferred← citeshttps://doi.org/10.1002/chem.201500068openalex-snapshot
Solid‐Phase Parallel Synthesis of Functionalised Medium‐to‐Large Cyclic Peptidomimetics through Three‐Component Coupling Driven by Aziridine Aldehyde Dimers
inferred← citeshttps://doi.org/10.1002/chem.201500368openalex-snapshot
Divergent Solid‐Phase Synthesis of Natural Product‐Inspired Bipartite Cyclodepsipeptides: Total Synthesis of Seragamide A
inferred← citeshttps://doi.org/10.1002/chem.201503171openalex-snapshot
Microwave‐Assisted Organocatalyzed Rearrangement of Propargyl Vinyl Ethers to Salicylaldehyde Derivatives: An Experimental and Theoretical Study
inferred← citeshttps://doi.org/10.1002/chem.201504684openalex-snapshot
Rules of Macrocycle Topology: A [13]‐Macrodilactone Case Study
inferred← citeshttps://doi.org/10.1002/chem.201504832openalex-snapshot
One‐Pot Approach to Organo‐Phosphorus–Chalcogen Macrocycles Incorporating Double OP(S)SCn or OP(Se)SeCn Scaffolds: A Synthetic and Structural Study
inferred← citeshttps://doi.org/10.1002/chem.201601004openalex-snapshot
Modular Synthesis of Novel Macrocycles Bearing α,β‐Unsaturated Chemotypes through a Series of One‐Pot, Sequential Protocols
inferred← citeshttps://doi.org/10.1002/chem.201602332openalex-snapshot
Harnessing C−H Activation of Benzhydroxamates as a Macrocyclization Strategy: Synthesis of Structurally Diverse Macrocyclic Isoquinolones
inferred← citeshttps://doi.org/10.1002/chem.201605246openalex-snapshot
Design of Organic Macrocycle‐Modified Iron Oxide Nanoparticles for Drug Delivery
inferred← citeshttps://doi.org/10.1002/chem.201605615openalex-snapshot
Ring‐Expansion Approach to Medium‐Sized Lactams and Analysis of Their Medicinal Lead‐Like Properties
inferred← citeshttps://doi.org/10.1002/chem.201700467openalex-snapshot
Ring‐Expansion Reactions in the Synthesis of Macrocycles and Medium‐Sized Rings
inferred← citeshttps://doi.org/10.1002/chem.201701183openalex-snapshot
Leptolyngbyolides, Cytotoxic Macrolides from the Marine Cyanobacterium Leptolyngbya sp.: Isolation, Biological Activity, and Catalytic Asymmetric Total Synthesis
inferred← citeshttps://doi.org/10.1002/chem.201701232openalex-snapshot
Photocontrol over Molecular Shape: Synthesis and Photochemical Evaluation of Glycoazobenzene Macrocycles
inferred← citeshttps://doi.org/10.1002/chem.201703209openalex-snapshot
MacroEvoLution: A New Method for the Rapid Generation of Novel Scaffold‐Diverse Macrocyclic Libraries
inferred← citeshttps://doi.org/10.1002/chem.201703316openalex-snapshot
Synthesis of Cyclic Peptide Mimetics by the Successive Ring Expansion of Lactams
inferred← citeshttps://doi.org/10.1002/chem.201802250openalex-snapshot
Chemoenzymatic Route to Oxyfunctionalized Cembranoids Facilitated by Substrate and Protein Engineering
inferred← citeshttps://doi.org/10.1002/chem.201803064openalex-snapshot
Iterative Assembly of Macrocyclic Lactones using Successive Ring Expansion Reactions
inferred← citeshttps://doi.org/10.1002/chem.201804440openalex-snapshot
Synthesis of Diverse α‐Fluoroalkoxyaryl Derivatives and Their Use for the Generation of Fluorinated Macrocycles
inferred← citeshttps://doi.org/10.1002/chem.201900813openalex-snapshot
Total Synthesis, Stereochemical Revision, and Biological Assessment of Iriomoteolide‐2a
inferred← citeshttps://doi.org/10.1002/chem.201902596openalex-snapshot
Domino Transformations of Ene/Yne Tethered Salicylaldehyde Derivatives: Pluripotent Platforms for the Construction of High sp3 Content and Privileged Architectures
inferred← citeshttps://doi.org/10.1002/chem.201904564openalex-snapshot
A Comparative Synthetic Strategy Perspective on α‐Amino Acid‐ and Non‐Amino Acid‐Derived Synthons towards Total Syntheses of Selected Natural Macrolides
inferred← citeshttps://doi.org/10.1002/chem.202001140openalex-snapshot
A Versatile Approach to Dynamic Amide Bond Formation with Imine Nucleophiles
inferred← citeshttps://doi.org/10.1002/chem.202002164openalex-snapshot
Evaluating the Viability of Successive Ring‐Expansions Based on Amino Acid and Hydroxyacid Side‐Chain Insertion
inferred← citeshttps://doi.org/10.1002/chem.202003655openalex-snapshot
Synthesis and Diversification of Macrocyclic Alkynediyl Sulfide Peptides
inferred← citeshttps://doi.org/10.1002/chem.202203717openalex-snapshot
Triple Thorpe–Ingold Effect in the Synthesis of 18‐Membered C3 Symmetric Lactams Stacking as Endless Supramolecular Tubes
inferred← citeshttps://doi.org/10.1002/chem.202303270openalex-snapshot
Divergent Cascade Ring‐Expansion Reactions of Acryloyl Imides
inferred← citeshttps://doi.org/10.1002/chem.202304176openalex-snapshot
In2Q2: A New Entry of 16‐Membered Tetraazamacrocycle Concatenating Indole and Quinoline Units
inferred← citeshttps://doi.org/10.1002/chem.202304319openalex-snapshot
Continuous Synthesis of a Macrocyclic Sulfite of Polyethylene Glycol by Cascaded Continuous Stirred Tank Reactors (CSTRs)
inferred← citeshttps://doi.org/10.1002/chem.202400308openalex-snapshot
Synthesis and Functionalization of Azetidine‐Containing Small Macrocyclic Peptides
inferred← citeshttps://doi.org/10.1002/chem.202502887openalex-snapshot
Modular Assembly of Macrocyclic Sulfonamides via Consecutive Cascade Ring Expansion Reactions
inferred← citeshttps://doi.org/10.1002/cjoc.201900316openalex-snapshot
Design and Synthesis of a Series of Novel Macrocycle Janus Kinase 2 Inhibitors
inferred← citeshttps://doi.org/10.1002/cmdc.201300387openalex-snapshot
A Template‐Based Approach to Inhibitors of Calpain 2, 20S Proteasome, and HIV‐1 Protease
inferred← citeshttps://doi.org/10.1002/cmdc.201500572openalex-snapshot
Hitting a Moving Target: How Does an N‐Methyl Group Impact Biological Activity?
inferred← citeshttps://doi.org/10.1002/cmdc.201600082openalex-snapshot
Design and Development of a Cyclic Decapeptide Scaffold with Suitable Properties for Bioavailability and Oral Exposure
inferred← citeshttps://doi.org/10.1002/cmdc.201700048openalex-snapshot
Pyrrole‐Based Macrocyclic Small‐Molecule Inhibitors That Target Oocyte Maturation
inferred← citeshttps://doi.org/10.1002/cmdc.201700478openalex-snapshot
Computational Macrocyclization: From de novo Macrocycle Generation to Binding Affinity Estimation
inferred← citeshttps://doi.org/10.1002/cmdc.201700522openalex-snapshot
Head‐to‐Tail Cyclic Peptide Inhibitors of the Interaction between Human von Willebrand Factor and Collagen
inferred← citeshttps://doi.org/10.1002/cmdc.70457openalex-snapshot
The Coalescence of a “Happy Accident” and an In Vitro Structure–Activity Panel: Increasing the Potency of a Cyclic Peptide Inhibitor to Thrombosis Initiation
inferred← citeshttps://doi.org/10.1002/cphc.201700995openalex-snapshot
Interconversion Rates between Conformational States as Rationale for the Membrane Permeability of Cyclosporines
inferred← citeshttps://doi.org/10.1002/cssc.202300200openalex-snapshot
Mizoroki‐Heck Macrocyclization Reactions at 1 M Concentration Catalyzed by Sub‐nanometric Palladium Clusters
inferred← citeshttps://doi.org/10.1002/ejoc.201101406openalex-snapshot
Convenient Synthesis of a Galacturonic Acid Based Macrocycle with Potential Copper‐Complexation Ability
inferred← citeshttps://doi.org/10.1002/ejoc.201300953openalex-snapshot
Synthesis and Properties of Carbohydrate‐Based BODIPY‐Functionalised Fluorescent Macrocycles
inferred← citeshttps://doi.org/10.1002/ejoc.201501445openalex-snapshot
Observations on the Influence of Precursor Conformations on Macrocyclization Reactions
inferred← citeshttps://doi.org/10.1002/ejoc.201601384openalex-snapshot
4,5‐Disubstituted N‐Methylimidazoles as Versatile Building Blocks for Defined Side‐Chain Introduction
inferred← citeshttps://doi.org/10.1002/ejoc.201800314openalex-snapshot
Awkwardly‐Shaped Dimers, Capsules and Tetramers: Molecular and Supramolecular Motifs in C5‐Arylated Chiral Calixsalens
inferred← citeshttps://doi.org/10.1002/ejoc.201801714openalex-snapshot
Syntheses of Bis‐Triazole Linked Carbohydrate Based Macrocycles and Their Applications for Accelerating Copper Sulfate Mediated Click Reaction
inferred← citeshttps://doi.org/10.1002/ejoc.201801839openalex-snapshot
Ceramide‐Templated Macrolactams: Total Synthesis and Biological Evaluation of Macrocyclic α‐Galactosylceramide Analogues and their Aglycons
inferred← citeshttps://doi.org/10.1002/ejoc.202300028openalex-snapshot
Synthesis and Applications of Peptides and Peptidomimetics in Drug Discovery
inferred← citeshttps://doi.org/10.1002/ejoc.202300939openalex-snapshot
Synthesis of 13–16‐Membered Cyclotetrapeptide Mimics by Ugi Reactions with Diacids and Diisonitriles
inferred← citeshttps://doi.org/10.1002/jhet.1968openalex-snapshot
Synthesis of New Macrocyclic Schiff Bases Containing Pyrazole and Triazole as Subcyclic Units
inferred← citeshttps://doi.org/10.1002/jhet.3922openalex-snapshot
Synthesis, antimicrobial activity, and ion transportation investigation of four new [1 + 1] condensed furan and thiophene‐based cycloheterophane amides
inferred← citeshttps://doi.org/10.1002/jhet.4383openalex-snapshot
Effective synthesis of new benzo‐fused macrocyclic and thiamacrocyclic dilactams and related pyrazolo‐fused macrocycles
inferred← citeshttps://doi.org/10.1002/jms.70058openalex-snapshot
Cyclic Peptide Conformational Landscapes Through the Lens of Mass Spectrometry and Orthogonal Spectroscopy
inferred← citeshttps://doi.org/10.1002/marc.201800748openalex-snapshot
Polymacrocycles Derived via Ugi Multi‐Component Reactions
inferred← citeshttps://doi.org/10.1002/mats.202000076openalex-snapshot
The Presence of a Wall Enhances the Probability for Ring‐Closing Metathesis: Insights from Classical Polymer Theory and Atomistic Simulations
inferred← citeshttps://doi.org/10.1002/med.21503openalex-snapshot
Recent advances in the discovery and development of factor XI/XIa inhibitors
inferred← citeshttps://doi.org/10.1002/med.70081openalex-snapshot
Current Development of Small Molecules Against Influenza A Virus by Targeting Hemagglutinin
inferred← citeshttps://doi.org/10.1002/minf.202300287openalex-snapshot
The macrocycle inhibitor landscape of SLC‐transporter
inferred← citeshttps://doi.org/10.1002/mog2.50openalex-snapshot
Applications of macrocyclic molecules in cancer therapy: Target cancer development or overcome drug resistance
inferred← citeshttps://doi.org/10.1002/mrc.4481openalex-snapshot
The NMR characterization of locked conformations of two stereoisomers of calix[4]tetrahydrofuran
inferred← citeshttps://doi.org/10.1002/pep2.24044openalex-snapshot
Development of a solid‐phase traceless‐Ugi multicomponent reaction for backbone anchoring and cyclic peptide synthesis
inferred← citeshttps://doi.org/10.1002/pep2.24064openalex-snapshot
Apelins, ELABELA, and their derivatives: Peptidic regulators of the cardiovascular system and beyond
inferred← citeshttps://doi.org/10.1002/pep2.24088openalex-snapshot
Cis/trans isomerization of proline peptide bonds in the backbone of cyclic disulfide‐bridged peptides
inferred← citeshttps://doi.org/10.1002/pep2.24161openalex-snapshot
One‐pot peptide cleavage and macrocyclization through direct amidation using triazabicyclodecene
inferred← citeshttps://doi.org/10.1002/prot.25682openalex-snapshot
Putative structural rearrangements associated with the interaction of macrocyclic inhibitors with norovirus 3CL protease
inferred← citeshttps://doi.org/10.1002/psc.3387openalex-snapshot
Current synthetic chemistry towards cyclic antimicrobial peptides
inferred← citeshttps://doi.org/10.1002/psc.3471openalex-snapshot
Opening the amino acid toolbox for peptide‐based NTS2‐selective ligands as promising lead compounds for pain management
inferred← citeshttps://doi.org/10.1002/slct.201801117openalex-snapshot
Natural Product Inspired Topology Directed Synthesis of Hybrid Macrocyclic Compounds: A Simple Approach to Natural Product Analogues
inferred← citeshttps://doi.org/10.1002/slct.201801900openalex-snapshot
Peptidomimicry with C 2 ‐Symmetric Oligourea Derivatives of 1,2‐Diaminocyclohexane and 1,2‐Diphenyl‐1,2‐diaminoethane: Chirality and Chain Length‐Dependent Conformation
inferred← citeshttps://doi.org/10.1002/slct.202100206openalex-snapshot
Applications of Yamaguchi Method to Esterification and Macrolactonization in Total Synthesis of Bioactive Natural Products
inferred← citeshttps://doi.org/10.1002/slct.202102715openalex-snapshot
Facile Synthesis of the Shape‐Persistent 4‐Hydroxybenzaldehyde Based Macrocycles and Exploration of their Key Electronic Properties: An Experimental and DFT Approach
inferred← citeshttps://doi.org/10.1002/slct.73412openalex-snapshot
Recent Advances in Synthesis, Characterization, and Electrochemical Investigations of Manganese Derived Complexes
inferred← citeshttps://doi.org/10.1002/tcr.201800052openalex-snapshot
One‐Step Construction of the Shape Persistent, Chiral But Symmetrical Polyimine Macrocycles
inferred← citeshttps://doi.org/10.1002/tcr.202000128openalex-snapshot
Unmasking Arene Ruthenium Building Blocks
inferred← citeshttps://doi.org/10.1007/7081_2015_163openalex-snapshot
Heterocyclic Extended Peptide Surrogates for β-Strand Stabilization
inferred← citeshttps://doi.org/10.1007/7081_2015_187openalex-snapshot
Synthesis of Peptidomimetics Through the Disrupted Ugi Reaction with Aziridine Aldehyde Dimers
inferred← citeshttps://doi.org/10.1007/978-1-0716-1689-5_14openalex-snapshot
MOrPH-PhD: A Phage Display System for the Functional Selection of Genetically Encoded Macrocyclic Peptides
inferred← citeshttps://doi.org/10.1007/978-1-0716-1689-5_24openalex-snapshot
Cyclization and Self-Assembly of Cyclic Peptides
inferred← citeshttps://doi.org/10.1007/978-1-0716-2285-8_20openalex-snapshot
Discovery of Cyclic Peptide Binders from Chemically Constrained Yeast Display Libraries
inferred← citeshttps://doi.org/10.1007/978-1-4939-2020-4_2openalex-snapshot
Synthesis of Macrocyclic Organo-peptide Hybrids from Ribosomal Polypeptide Precursors via CuAAC-/Hydrazide-Mediated Cyclization
inferred← citeshttps://doi.org/10.1007/978-1-4939-2020-4_5openalex-snapshot
Macrocyclic Templates for Library Synthesis of Peptido-Conjugates
inferred← citeshttps://doi.org/10.1007/978-1-4939-9504-2_9openalex-snapshot
Frontier Between Cyclic Peptides and Macrocycles
inferred← citeshttps://doi.org/10.1007/978-3-030-14632-0_2openalex-snapshot
Resources for Chemical, Biological, and Structural Data on Natural Products
inferred← citeshttps://doi.org/10.1007/978-981-13-0773-7_2openalex-snapshot
High-Throughput Screening in the Discovery of Small-Molecule Inhibitors of Protein-Protein Interactions
inferred← citeshttps://doi.org/10.1007/978-981-99-2423-3_6openalex-snapshot
Drug Design Methods to Regulate Protein–Protein Interactions
inferred← citeshttps://doi.org/10.1007/s00044-018-2268-8openalex-snapshot
Mechanistic studies of the apoptosis induced by the macrocyclic natural product tetrandrine in MGC 803 cells
inferred← citeshttps://doi.org/10.1007/s00044-019-02424-3openalex-snapshot
Macrocyclic effect on inhibitory activity: a modeling study on MerTK inhibitors
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