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Remarkable Potential of the α-Aminophosphonate/Phosphinate Structural Motif in Medicinal Chemistry

https://doi.org/10.1021/jm200587f

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inferredcites →https://doi.org/10.1046/j.1432-1033.2002.03103.xopenalex-snapshot

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inferredcites →https://doi.org/10.1073/pnas.96.8.4330openalex-snapshot

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inferredcites →https://doi.org/10.1074/jbc.c300511200openalex-snapshot

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inferredcites →https://doi.org/10.1074/jbc.m109.060418openalex-snapshot

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Computer-Aided Analysis and Design of Phosphonic and Phosphinic Enzyme Inhibitors as Potential Drugs and Agrochemicals

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What points at this work

Incoming claims: where this work appears in other papers’ reference lists and arguments.

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Metal‐Free Synthesis of Allylic Phosphine Oxides via [2,3]‐Rearrangement/Michael Addition Cascade

inferred← citeshttps://doi.org/10.1002/hc.21086openalex-snapshot

α‐Aminophosphonates and α‐Aminophosphine Oxides by the Microwave‐Assisted Kabachnik–Fields Reactions of 3‐Amino‐6‐methyl‐2 H‐pyran‐2‐ones

inferred← citeshttps://doi.org/10.1002/hc.21126openalex-snapshot

The Synthesis of N,N ‐Bis(dialkoxyphosphinoylmethyl)‐ and N,N ‐Bis(diphenylphosphinoylmethyl)glycine Esters by the Microwave‐Assisted Double Kabachnik–Fields Reaction

inferred← citeshttps://doi.org/10.1002/hc.21130openalex-snapshot

Double Asymmetric Induction in the Synthesis of Enantiomeric α‐Aminophosphonic Acids Mediated by Sulfinimines

inferred← citeshttps://doi.org/10.1002/hc.21192openalex-snapshot

A Critical Overview of the Kabachnik-Fields Reactions Utilizing Trialkyl Phosphites in Water as the Reaction Medium: A Study of the Benzaldehyde-Benzylamine Triethyl Phosphite/Diethyl Phosphite Models

inferred← citeshttps://doi.org/10.1002/hc.21221openalex-snapshot

Synthesis of N,N‐Bis(dialkoxyphosphinoylmethyl)‐ and N,N‐Bis(diphenylphosphinoylmethyl)‐β‐ and γ‐amino acid Derivatives by the Microwave‐Assisted Double Kabachnik–Fields Reaction

inferred← citeshttps://doi.org/10.1002/hc.21251openalex-snapshot

Clean Procedure for the Synthesis of Α-Aminophosphonates Catalyzed by Choline-Based Ionic Liquid

inferred← citeshttps://doi.org/10.1002/hc.21324openalex-snapshot

Synthesis of α‐aminophosphonates from α‐hydroxyphosphonates; a theoretical study

inferred← citeshttps://doi.org/10.1002/hc.21325openalex-snapshot

Phosphosulfonic acid‐catalyzed green synthesis and bioassay of α‐aryl‐α′‐1,3,4‐thiadiazolyl aminophosphonates

inferred← citeshttps://doi.org/10.1002/hc.21343openalex-snapshot

Synthesis of alkyl α‐aminomethyl‐phenylphosphinates and N,N‐bis(alkoxyphenylphosphinylmethyl)amines by the microwave‐assisted Kabachnik–Fields reaction

inferred← citeshttps://doi.org/10.1002/hc.21398openalex-snapshot

First practical synthesis of novel 1‐phosphonylated pyrrolo[1,2‐a]pyrazine derivatives

inferred← citeshttps://doi.org/10.1002/hlca.202100190openalex-snapshot

Visible‐Light Mediated Photooxidative Phosphorylation of Benzylamines: A Novel and Mild Pathway Towards α‐Aminophosphorus Compounds

inferred← citeshttps://doi.org/10.1002/jhet.3593openalex-snapshot

A Straightforward Synthesis of Six‐Membered‐Ring Heterocyclic α‐Aminophosphonic Acids from N‐Acyliminium Ions

inferred← citeshttps://doi.org/10.1002/marc.201900533openalex-snapshot

A Facile Preparation of Mussel‐Inspired Poly(dopamine phosphonate‐co‐PEGMA)s via a One‐Pot Multicomponent Polymerization System

inferred← citeshttps://doi.org/10.1002/pro.70611openalex-snapshot

Phosphinate pseudopeptide enhances binding free energy in HIV ‐1 protease by driving flap closure and suppressing global flexibility

inferred← citeshttps://doi.org/10.1002/ps.4299openalex-snapshot

Phytotoxicity of aminobisphosphonates targeting both δ 1 ‐pyrroline‐5‐carboxylate reductase and glutamine synthetase

inferred← citeshttps://doi.org/10.1002/psc.2841openalex-snapshot

Practical synthesis of novel phosphonopeptides containing AibP

inferred← citeshttps://doi.org/10.1002/rcm.6984openalex-snapshot

Cleavage of phosphorus–carbon (P–C) bonds of α‐amino phosphonates with intramolecular hydrogen migration in the gas phase using electrospray ionization tandem mass spectrometry

inferred← citeshttps://doi.org/10.1002/slct.201600070openalex-snapshot

A Rapid One‐Pot Five Component Sequential Access to Novel Imidazo[2,1‐b]thiazinyl‐α‐aminophosphonates

inferred← citeshttps://doi.org/10.1002/slct.201701715openalex-snapshot

One Step Carbon‐Phosphor Bond Formation and N‐Alkylation of Tetrahydroisoquinolines under Silver Catalysis

inferred← citeshttps://doi.org/10.1002/slct.201800009openalex-snapshot

Open Flask, Clean and Practical Protocol for Diastereoselective Syntheses of Oxindole Containing Phosphinoyl Compounds under Catalyst‐Free and Solvent‐Free Conditions

inferred← citeshttps://doi.org/10.1002/slct.201800700openalex-snapshot

Synthesis of New Heteroaryl α‐Aminophosphonates and Evaluation of Their Cytotoxicity against Human Breast Cancer MCF‐7 Cell Lines

inferred← citeshttps://doi.org/10.1002/slct.201801456openalex-snapshot

Convenient Au(III)‐Catalysed Synthesis of 1‐Alkyl‐3‐diethoxy‐phosphoryl‐1,2,3,4‐tetrahydroisoquinolines

inferred← citeshttps://doi.org/10.1002/slct.201903191openalex-snapshot

rGO‐SO 3 H Catalysed Green Synthesis of Fluoro‐Substituted Aminomethylene Bisphosphonates and their Anticancer, Molecular Docking studies

inferred← citeshttps://doi.org/10.1002/slct.202000486openalex-snapshot

TAPSO** : A Highly Efficient and Ecofriendly Catalyst for the Synthesis of α‐ Aminophosphonates and Tetrahydropyridines **3‐[N‐Tris(hydroxymethyl)methylamino]‐2‐hydroxypropanesulfonic acid

inferred← citeshttps://doi.org/10.1002/slct.202000693openalex-snapshot

An Overview of Microwave‐Assisted Kabachnik‐Fields Reactions

inferred← citeshttps://doi.org/10.1002/slct.202002369openalex-snapshot

Stereochemistry of the Kabachnik‐Fields Condensation of Terpenic Amino Oximes with Aldehydes and Dimethyl Phosphite

inferred← citeshttps://doi.org/10.1002/slct.202003848openalex-snapshot

Experimental Investigation on the Correlation between the Physicochemical Properties and Catalytic Activity of Six DESs in the Kabachnik‐Fields Reaction

inferred← citeshttps://doi.org/10.1002/slct.202104220openalex-snapshot

Highly Efficient One‐pot Aerobic Synthesis of α‐Aminophosphonate from Alcohols: Dual Catalytic Effect of Tetrabutylammonium Tribromide (TBATB)

inferred← citeshttps://doi.org/10.1002/slct.202200568openalex-snapshot

One‐Pot Synthesis of Selected P‐Vinylbenzyls under Solvent‐Free Conditions

inferred← citeshttps://doi.org/10.1002/slct.202202757openalex-snapshot

Catalyst‐ and Solvent‐Free Hydrophosphorylation of Aldimines with Secondary Phosphine Chalcogenides: Synthesis of Tertiary α ‐Aminophosphine Oxides, Sulfides and Selenides

inferred← citeshttps://doi.org/10.1002/slct.202300639openalex-snapshot

A Novel Phosphonates Synthesized from Schiff's Base Indenoquinoxaline Derivatives and its Biological Activity

inferred← citeshttps://doi.org/10.1002/slct.202404258openalex-snapshot

Phosphorus Heterocycles and Their Biological Applications

inferred← citeshttps://doi.org/10.1002/slct.202404579openalex-snapshot

Hydrophosphorylation of 1,1,1,3,3,3‐hexafluorobut‐2‐yne (HFB) with Diethyl Hydrogenphosphonate: Attractive Synthetic Route to Various Types of CF 3 ‐Containing Phosphonates

inferred← citeshttps://doi.org/10.1002/slct.202404882openalex-snapshot

Mechanochemical Synthesis of Phosphoryl Amides and Esters from Diphenylphosphoryl Azides Under Mild Conditions

inferred← citeshttps://doi.org/10.1002/slct.202500015openalex-snapshot

α ‐Aminophosphonates: Antimicrobial, Anti‐Inflammatory, Antioxidant Activities, Molecular Docking, and DFT Studies

inferred← citeshttps://doi.org/10.1002/slct.202501752openalex-snapshot

Efficient and Versatile Synthesis of Tetrasubstituted α‐Amino and α‐Hydroxy Dimethylphosphine Oxides from Carbo‐ and Heterocyclic Ketones

inferred← citeshttps://doi.org/10.1002/slct.202503353openalex-snapshot

Double C─H Phosphorylation of Quinoxalines Under Catalyst‐Free Conditions

inferred← citeshttps://doi.org/10.1002/slct.73924openalex-snapshot

TBAI‐Mediated, One‐Pot Efficient Synthesis of α‐Aminophosphonates From Aryl Azides and Phosphites

inferred← citeshttps://doi.org/10.1002/tcr.201500266openalex-snapshot

Applications of Chiral Squaramides: From Asymmetric Organocatalysis to Biologically Active Compounds

inferred← citeshttps://doi.org/10.1002/tcr.202200026openalex-snapshot

Rational Development of Bacterial Ureases Inhibitors

inferred← citeshttps://doi.org/10.1007/128_2014_566openalex-snapshot

Synthesis and Biological Applications of Phosphinates and Derivatives

inferred← citeshttps://doi.org/10.1007/978-1-0716-0227-0_20openalex-snapshot

Peptide and Pseudopeptide Bond Synthesis in Phosphorus Dipeptide Analogs

inferred← citeshttps://doi.org/10.1007/978-3-319-38878-6_1openalex-snapshot

Electrophilic Amination for the Synthesis of Alkyl and Aryl Amines

inferred← citeshttps://doi.org/10.1007/978-3-319-38878-6_2openalex-snapshot

Selective α-Amination and α-Acylation of Esters and Amides via Dual Reactivity of O-Acylhydroxylamines Toward Zinc Enolates

inferred← citeshttps://doi.org/10.1007/978-3-319-38878-6_3openalex-snapshot

Copper-Catalyzed α-Amination of Phosphonates and Phosphine Oxides: A Direct Approach to α-Amino Phosphonic Acids and Derivatives

inferred← citeshttps://doi.org/10.1007/s00044-013-0899-3openalex-snapshot

Coumarin-containing aminophosphonates bridged with chiral side chain: synthesis and influence of chirality on cytotoxicity and DNA binding

inferred← citeshttps://doi.org/10.1007/s00044-014-1282-8openalex-snapshot

Transition metal complexes of α-aminophosphonates Part I: synthesis, spectroscopic characterization, and in vitro anticancer activity of copper(II) complexes of α-aminophosphonates

inferred← citeshttps://doi.org/10.1007/s00216-013-6938-6openalex-snapshot

Direct high-performance liquid chromatographic enantioseparation of free α-, β- and γ-aminophosphonic acids employing cinchona-based chiral zwitterionic ion exchangers

inferred← citeshttps://doi.org/10.1007/s00706-019-02465-9openalex-snapshot

Recent advances in the applications of Wittig reaction in the total synthesis of natural products containing lactone, pyrone, and lactam as a scaffold

inferred← citeshttps://doi.org/10.1007/s00706-019-2385-1openalex-snapshot

Tungstosulfonic acid-catalyzed green synthesis and bioassay of α-aminophosphonates

inferred← citeshttps://doi.org/10.1007/s00706-020-02551-3openalex-snapshot

Green one-pot synthesis of N-bisphosphonates as antimicrobial and antioxidant agents

inferred← citeshttps://doi.org/10.1007/s00726-019-02774-7openalex-snapshot

The self-disproportionation of enantiomers (SDE) via column chromatography of β-amino-α,α-difluorophosphonic acid derivatives

inferred← citeshttps://doi.org/10.1007/s00726-021-02962-4openalex-snapshot

New approaches towards the synthesis of 1,2,3,4-tetrahydro isoquinoline-3-phosphonic acid (TicP)

inferred← citeshttps://doi.org/10.1007/s10593-020-02697-2openalex-snapshot

One-Pot Synthesis of N-(Phosphorylmethyl)Pyrrolidines via Acid-Catalyzed Cascade Elimination/Cyclization/Friedel–Crafts Reaction

inferred← citeshttps://doi.org/10.1007/s10989-019-10004-7openalex-snapshot

Phosphinic Dehydrodipeptides: Diversification of the P1′ Residue with the Morita–Baylis–Hillman Acetates and Inhibition of Alanyl Aminopeptidases

inferred← citeshttps://doi.org/10.1007/s11094-019-01922-3openalex-snapshot

Polyene Macrolide Antibotic Derivatives: Preparation, Overcoming Drug Resistance, and Prospects for Use in Medical Practice (Review)

inferred← citeshttps://doi.org/10.1007/s11144-022-02329-0openalex-snapshot

Full factorial optimization of α-aminophosphonates synthesis using diphenylphosphinic acid as efficient organocatalyst

inferred← citeshttps://doi.org/10.1007/s11164-017-2890-yopenalex-snapshot

A novel straightforward synthesis of α-aminophosphonates: one-pot three-component condensation of alcohols, amines, and diethylphosphite in the presence of CuO@Fe3O4 nanoparticles as a catalyst

inferred← citeshttps://doi.org/10.1007/s11164-020-04321-6openalex-snapshot

Design, synthesis, cytotoxic evaluation and molecular docking studies of novel thiazolyl α-aminophosphonates

inferred← citeshttps://doi.org/10.1007/s11172-021-3069-7openalex-snapshot

The synthesis of novel aminoalkylphosphoryl derivatives of diarylmethane and dibenzoxanthene based on acetals and phenols

inferred← citeshttps://doi.org/10.1007/s11224-019-01483-xopenalex-snapshot

New crystal structures of fluorinated α-aminophosphonic acid analogues of phenylglycine

inferred← citeshttps://doi.org/10.1007/s11426-025-2935-3openalex-snapshot

Streamlined synthesis of α-keto-, α-hydroxy- and α,α-difluorophosphonates from amides via electrophilic activation with trifluoromethanesulfonic anhydride

inferred← citeshttps://doi.org/10.1007/s12010-014-1356-6openalex-snapshot

Fungal Platform for Direct Chiral Phosphonic Building Blocks Production. Closer Look on Conversion Pathway

inferred← citeshttps://doi.org/10.1007/s13361-012-0556-yopenalex-snapshot

Differentiation of Diastereoisomers of Protected 1,2-Diaminoalkylphosphonic Acids by EI Mass Spectrometry and Density Functional Theory

inferred← citeshttps://doi.org/10.1007/s13738-018-1571-0openalex-snapshot

One-pot facile synthesis of novel 1,2,3-triazole-appended α-aminophosphonates

inferred← citeshttps://doi.org/10.1007/s13738-023-02811-zopenalex-snapshot

Discovery of novel anticancer candidates based on a combination strategy of synthesis, characterization, biological activity evaluation, consensus docking and molecular modeling

inferred← citeshttps://doi.org/10.1007/s41061-024-00456-xopenalex-snapshot

Recent Advances in the Application of P(III)-Nucleophiles to Create New P−C Bonds through Michaelis–Arbuzov-Type Rearrangement

inferred← citeshttps://doi.org/10.1016/b978-0-12-813834-2.00003-2openalex-snapshot

Reactivity of P–H Group of Phosphine Oxides

inferred← citeshttps://doi.org/10.1016/b978-0-12-819540-6.00005-xopenalex-snapshot

Sonochemical protocol for solvent-free organic synthesis

inferred← citeshttps://doi.org/10.1016/b978-0-32-390644-9.00109-8openalex-snapshot

Phosphorus (V) Stereochemistry and Industrial Applications

inferred← citeshttps://doi.org/10.1016/b978-0-443-27482-4.00016-2openalex-snapshot

Advances in ultrasound-driven organic synthesis without the use of solvents: A green chemistry perspective

inferred← citeshttps://doi.org/10.1016/b978-0-443-31482-7.00101-6openalex-snapshot

Functions Containing Two Nitrogens or a Nitrogen and a Phosphorus

inferred← citeshttps://doi.org/10.1016/b978-0-443-31482-7.00104-1openalex-snapshot

Functions Incorporating a Halogen and Another Heteroatom Group Other Than a Chalcogen

inferred← citeshttps://doi.org/10.1016/b978-0-443-33374-3.00002-5openalex-snapshot

Preparation and chemical transformations of α-iminophosphonates

inferred← citeshttps://doi.org/10.1016/b978-0-443-33374-3.00016-5openalex-snapshot

Phosphonates and the brain, from diagnostics to medicines for neurological disorders

inferred← citeshttps://doi.org/10.1016/b978-0-443-33374-3.00023-2openalex-snapshot

Biology of aminophosphonates

inferred← citeshttps://doi.org/10.1016/b978-0-443-33374-3.00040-2openalex-snapshot

Synthesis of phosphonates for pharmaceutical applications

inferred← citeshttps://doi.org/10.1016/bs.aihch.2015.10.004openalex-snapshot

Phosphono- and Phosphinolactones in the Life Sciences

inferred← citeshttps://doi.org/10.1016/j.arabjc.2018.05.002openalex-snapshot

Fluorinated phosphonate analogues of phenylalanine: Synthesis, X-ray and DFT studies

inferred← citeshttps://doi.org/10.1016/j.biochi.2012.10.018openalex-snapshot

An integrated approach to the ligand binding specificity of Neisseria meningitidis M1 alanine aminopeptidase by fluorogenic substrate profiling, inhibitory studies and molecular modeling

inferred← citeshttps://doi.org/10.1016/j.biochi.2018.06.005openalex-snapshot

Substituted phosphonic analogues of phenylglycine as inhibitors of phenylalanine ammonia lyase from potatoes

inferred← citeshttps://doi.org/10.1016/j.bioorg.2012.01.003openalex-snapshot

Synthesis and inhibitory activity of ureidophosphonates, against acetylcholinesterase: Pharmacological assay and molecular modeling

inferred← citeshttps://doi.org/10.1016/j.bioorg.2019.01.047openalex-snapshot

First biological conversion of chiral heterophosphonate derivative – Scaling and paths of conversion discussion

inferred← citeshttps://doi.org/10.1016/j.bioorg.2019.01.064openalex-snapshot

Synthesis, crystal structure and biological evaluation of new phosphoramide derivatives as urease inhibitors using docking, QSAR and kinetic studies

inferred← citeshttps://doi.org/10.1016/j.bioorg.2019.103039openalex-snapshot

Potential chemical transformation of phosphinic acid derivatives and their applications in the synthesis of drugs

inferred← citeshttps://doi.org/10.1016/j.bioorg.2020.104390openalex-snapshot

Discovery of novel sulfonamide-containing aminophosphonate derivatives as selective COX-2 inhibitors and anti-tumor candidates

inferred← citeshttps://doi.org/10.1016/j.bioorg.2021.104718openalex-snapshot

Novel α-Aminophosphonates of imatinib Intermediate: Synthesis, anticancer Activity, human Abl tyrosine kinase Inhibition, ADME and toxicity prediction

inferred← citeshttps://doi.org/10.1016/j.bioorg.2023.106846openalex-snapshot

Discovery of novel 4,5-diphenyl-imidazol-α-aminophosphonate hybrids as promising anti-diabetic agents: Design, synthesis, in vitro, and in silico enzymatic studies

inferred← citeshttps://doi.org/10.1016/j.bioorg.2023.106935openalex-snapshot

Exploring the reactivity of bicyclic α-iminophosphonates to access new imidazoline I2 receptor ligands

inferred← citeshttps://doi.org/10.1016/j.bioorg.2023.107008openalex-snapshot

Green approach to the synthesis of α-aminophosphonate-tetrahydroisoquinoline hybrids and their anti-cholinesterase activity

inferred← citeshttps://doi.org/10.1016/j.bioorg.2024.107930openalex-snapshot

Combretastatin A-4 based compounds as potential anticancer agents: A review

inferred← citeshttps://doi.org/10.1016/j.bmc.2018.12.041openalex-snapshot

000Synthesis of new α-aminophosphonates: Evaluation as anti-inflammatory agents and QSAR studies

inferred← citeshttps://doi.org/10.1016/j.bmc.2023.117512openalex-snapshot

Harvesting phosphorus-containing moieties for their antibacterial effects

inferred← citeshttps://doi.org/10.1016/j.bmcl.2013.08.005openalex-snapshot

Synthesis and antitumor activities of novel α-aminophosphonates dehydroabietic acid derivatives

inferred← citeshttps://doi.org/10.1016/j.bmcl.2013.12.030openalex-snapshot

Synthesis and antitumor activities of novel rhein α-aminophosphonates conjugates

inferred← citeshttps://doi.org/10.1016/j.bmcl.2016.06.062openalex-snapshot

Discovery of potent and selective inhibitors of human aminopeptidases ERAP1 and ERAP2 by screening libraries of phosphorus-containing amino acid and dipeptide analogues

inferred← citeshttps://doi.org/10.1016/j.bmcl.2019.01.026openalex-snapshot

Calixarene-based phosphinic acids as inhibitors of protein tyrosine phosphatases

inferred← citeshttps://doi.org/10.1016/j.bmcl.2019.02.034openalex-snapshot

Recent developments in the synthesis and applications of phosphinic peptide analogs

inferred← citeshttps://doi.org/10.1016/j.bmcl.2021.128000openalex-snapshot

Fiaud’s Acid, a novel organocatalyst for diastereoselective bis α-aminophosphonates synthesis with in-vitro biological evaluation of antifungal, antioxidant and enzymes inhibition potential

inferred← citeshttps://doi.org/10.1016/j.bmcl.2022.128695openalex-snapshot

Natural aloe emodin-hybridized sulfonamide aminophosphates as novel potential membrane-perturbing and DNA-intercalating agents against Enterococcus faecalis

inferred← citeshttps://doi.org/10.1016/j.bmcl.2025.130096openalex-snapshot

Applications of innovative synthetic strategies in anticancer drug discovery: The driving force of new chemical reactions

inferred← citeshttps://doi.org/10.1016/j.bone.2021.116289openalex-snapshot

Bisphosphonates: The role of chemistry in understanding their biological actions and structure-activity relationships, and new directions for their therapeutic use

inferred← citeshttps://doi.org/10.1016/j.cclet.2017.02.012openalex-snapshot

Synthesis and structure-activity relationships study of α -aminophosphonate derivatives containing a quinoline moiety

inferred← citeshttps://doi.org/10.1016/j.cclet.2022.107914openalex-snapshot

Ni-catalyzed regiodivergent hydrophosphorylation of enynes

inferred← citeshttps://doi.org/10.1016/j.cclet.2023.109294openalex-snapshot

Copper(I)-catalyzed diastereodivergent construction of vicinal P-chiral and C-chiral centers facilitated by dual “soft-soft” interaction

inferred← citeshttps://doi.org/10.1016/j.cclet.2026.112432openalex-snapshot

Enantioconvergent hydrophosphination of allylic alcohols to access chiral γ-hydroxyphosphines via multicatalysis

inferred← citeshttps://doi.org/10.1016/j.ccr.2021.214210openalex-snapshot

What blocks more anticancer platinum complexes from experiment to clinic: Major problems and potential strategies from drug design perspectives

inferred← citeshttps://doi.org/10.1016/j.drudis.2018.11.016openalex-snapshot

Phosphinic acids: current status and potential for drug discovery

inferred← citeshttps://doi.org/10.1016/j.ejmech.2013.04.039openalex-snapshot

The development of a new class of inhibitors for betaine-homocysteine S-methyltransferase

inferred← citeshttps://doi.org/10.1016/j.ejmech.2014.02.067openalex-snapshot

Synthesis and antitumor activities of novel α-aminophosphonate derivatives containing an alizarin moiety

inferred← citeshttps://doi.org/10.1016/j.ejmech.2016.04.018openalex-snapshot

A structural insight into the P1 S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases

inferred← citeshttps://doi.org/10.1016/j.ejmech.2017.06.021openalex-snapshot

Mild C(sp)–H functionalization of dihydrosanguinarine and dihydrochelerythrine for development of highly cytotoxic derivatives

inferred← citeshttps://doi.org/10.1016/j.ejmech.2018.02.058openalex-snapshot

Novel topoisomerase I inhibitors. Syntheses and biological evaluation of phosphorus substituted quinoline derivates with antiproliferative activity

inferred← citeshttps://doi.org/10.1016/j.ejmech.2018.09.011openalex-snapshot

Synthesis of novel antiproliferative hybrid bis-(3-indolyl)methane phosphonate derivatives

inferred← citeshttps://doi.org/10.1016/j.ejmech.2018.09.074openalex-snapshot

Structural exploration of cinnamate-based phosphonic acids as inhibitors of bacterial ureases

inferred← citeshttps://doi.org/10.1016/j.ejmech.2018.10.065openalex-snapshot

Antileishmanial activity of new hybrid tetrahydroquinoline and quinoline derivatives with phosphorus substituents

inferred← citeshttps://doi.org/10.1016/j.ejmech.2018.12.002openalex-snapshot

Synthesis and biological evaluation of cyanoaziridine phosphine oxides and phosphonates with antiproliferative activity

inferred← citeshttps://doi.org/10.1016/j.ejmech.2019.07.029openalex-snapshot

Design, synthesis and biological evaluation of novel α-aminophosphonate oxadiazoles via optimized iron triflate catalyzed reaction as apoptotic inducers

inferred← citeshttps://doi.org/10.1016/j.ejmech.2019.111771openalex-snapshot

First synthesis of merged hybrids phosphorylated azirino[2,1-b]benzo[e][1,3]oxazine derivatives as anticancer agents

inferred← citeshttps://doi.org/10.1016/j.ejmech.2022.114439openalex-snapshot

Dual-functional antitumor conjugates improving the anti-metastasis effect of combretastatin A4 by targeting tubulin polymerization and matrix metalloproteinases

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