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Oxadiazoles in Medicinal Chemistry
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What this work says
Outgoing claims: the papers this work cites, builds on, or argues with.
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Infrared spectra of chalcone analogs containing the selenophene nucleus
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Dipole moments and the structure of the molecules of some oxadiazole derivatives
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Pharmacology of terazosin
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Antikinetoplastid activity of 3-aryl-5-thiocyanatomethyl-1,2,4-oxadiazoles
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Development of novel β-amyloid probes based on 3,5-diphenyl-1,2,4-oxadiazole
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Physiochemical drug properties associated with in vivo toxicological outcomes
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inferredcites →https://doi.org/10.1016/j.tetlet.2006.05.051openalex-snapshot
A mild and efficient one pot synthesis of 1,3,4-oxadiazoles from carboxylic acids and acyl hydrazides
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Structural characterization of two oxadiazolic systems used as spacers for potential angiotensin II receptor antagonists
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Bioisosterism: A Rational Approach in Drug Design
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Correlations between the solvent hydrogen bond acceptor parameter .beta. and the calculated molecular electrostatic potential
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What points at this work
Incoming claims: where this work appears in other papers’ reference lists and arguments.
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Triphenylphosphonium Anhydride Trifluoromethanesulfonate
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Triphenylphosphonium Anhydride Trifluoromethanesulfonate
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1,2,4‐ and 1,3,4‐Oxadiazole Synthesis by Palladium‐Catalyzed Carbonylative Assembly of Aryl Bromides with Amidoximes or Hydrazides
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Pd/PTABS: Catalyst for Efficient C−H (Hetero)Arylation of 1,3,4‐Oxadiazoles Using Bromo(Hetero)Arenes
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General α‐Amino 1,3,4‐Oxadiazole Synthesis via Late‐Stage Reductive Functionalization of Tertiary Amides and Lactams**
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Advancing the Drug Discovery and Development Process
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General α‐Amino 1,3,4‐Oxadiazole Synthesis via Late‐Stage Reductive Functionalization of Tertiary Amides and Lactams**
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Oxadiazoles as Privileged Motifs for Promising Anticancer Leads: Recent Advances and Future Prospects
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Some Novel Mannich Bases of 5‐(3,4‐Dichlorophenyl)‐1,3,4‐oxadiazole‐2(3H)‐one and Their Anti‐Inflammatory Activity
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Synthesis of 5‐[(1 H ‐indol‐3‐yl)methyl]‐1,3,4‐oxadiazole‐2(3 H )‐thiones and their protective activity against oxidative stress
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Activity Profiling of Nitro‐Substituted Di(Hetero)Aryl 1,3,4‐ and 1,2,4‐Oxadiazoles: Antimicrobial, Cholinesterase Inhibition and Antioxidant Potential
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inferred← citeshttps://doi.org/10.1002/slct.202500049openalex-snapshot
Synthesis of Quinazoline‐1,3,4‐Oxadiazole Linked 1,2,3‐Triazole Hybrids as Potent EGFR Targeting Antilung Cancer Agents: In Vitro, In Silico, and DFT Studies
inferred← citeshttps://doi.org/10.1002/slct.74274openalex-snapshot
Rational Design and Synthesis of Benzothiophene–Quinoxaline–Oxadiazole Conjugates Targeting Bacterial and Fungal Pathogens
inferred← citeshttps://doi.org/10.1002/slct.74346openalex-snapshot
Facile Synthesis of Trifluoroethyl‐Functionalized Spirooxindole‐Oxadiazoles via Nitrile Oxide–Isatin Ketimine (3+2) Cycloaddition
inferred← citeshttps://doi.org/10.1007/7355_2013_29openalex-snapshot
The Influence of Bioisosteres in Drug Design: Tactical Applications to Address Developability Problems
inferred← citeshttps://doi.org/10.1007/978-3-319-48281-1_181-1openalex-snapshot
Sustainable Advancement to the Synthesis of Oxadiazoles
inferred← citeshttps://doi.org/10.1007/978-3-319-68255-6_181openalex-snapshot
Sustainable Advancement to the Synthesis of Oxadiazoles
inferred← citeshttps://doi.org/10.1007/978-981-19-0832-3_6openalex-snapshot
Various Synthetic Strategies and Therapeutic Potential of Thiadiazole, Oxadiazole, Isoxazole and Isothiazole Derivatives
inferred← citeshttps://doi.org/10.1007/s00044-014-1025-xopenalex-snapshot
Recyclable CuO nanoparticles-catalyzed synthesis of novel-2,5-disubstituted 1,3,4-oxadiazoles as antiproliferative, antibacterial, and antifungal agents
inferred← citeshttps://doi.org/10.1007/s00044-014-1162-2openalex-snapshot
Multistep synthesis of 1-[{(5-alkenyl/hydroxyalkenylsubstituted)-1,3,4-oxadiazol-2-yl}-methyl]-2-methyl-1H-benzimidazole series and in vitro anticancer screening, SAR studies
inferred← citeshttps://doi.org/10.1007/s00044-016-1651-6openalex-snapshot
Synthesis and antimicrobial evaluation of novel urea derivatives from chromene based oxadiazole amines
inferred← citeshttps://doi.org/10.1007/s00044-017-2047-yopenalex-snapshot
Design, synthesis, characterization, and molecular modeling studies of novel oxadiazole derivatives of nipecotic acid as potential anticonvulsant and antidepressant agents
inferred← citeshttps://doi.org/10.1007/s00044-018-2211-zopenalex-snapshot
Synthesis and DNA binding of new adenine derivatives incorporating 5-((Alkylthio)-1,3,4-oxadiazol-2-yl)methyl moiety
inferred← citeshttps://doi.org/10.1007/s00044-019-02475-6openalex-snapshot
Design, synthesis, and in vitro evaluation of novel 1,3,4-oxadiazolecarbamothioate derivatives of Rivastigmine as selective inhibitors of BuChE
inferred← citeshttps://doi.org/10.1007/s00044-022-02943-6openalex-snapshot
Design, synthesis and molecular docking studies of novel benzimidazole-1,3,4-oxadiazole hybrids for their carbonic anhydrase inhibitory and antioxidant effects
inferred← citeshttps://doi.org/10.1007/s00044-023-03035-9openalex-snapshot
The pyridazine heterocycle in molecular recognition and drug discovery
inferred← citeshttps://doi.org/10.1007/s00339-019-2692-8openalex-snapshot
Solvatochromic analysis and DFT computational study of N-(hexyl)-N-(5-(3-hydroxynaphthyl-2-yl)-1,3,4-oxadiazol-2-yl)amine
inferred← citeshttps://doi.org/10.1007/s00706-015-1528-2openalex-snapshot
Molecular properties prediction and synthesis of new oxadiazole derivatives possessing 3-fluoro-4-methoxyphenyl moiety as potent anti-inflammatory and analgesic agents
inferred← citeshttps://doi.org/10.1007/s00706-019-02478-4openalex-snapshot
Synthesis, molecular docking, antimicrobial evaluation, and DNA cleavage assay of new thiadiazole/oxadiazole ciprofloxacin derivatives
inferred← citeshttps://doi.org/10.1007/s00775-023-02037-7openalex-snapshot
Desulfurization of thiosemicarbazones: the role of metal ions and biological implications
inferred← citeshttps://doi.org/10.1007/s00894-024-05843-1openalex-snapshot
How do physicochemical properties contribute to inhibitory activity of promising peptides against Zika Virus NS3 protease?
inferred← citeshttps://doi.org/10.1007/s00894-026-06682-yopenalex-snapshot
Theoretical analysis on structure–property relationships of triazole-oxadiazole nitro derivatives for energetic applications
inferred← citeshttps://doi.org/10.1007/s10593-019-02607-1openalex-snapshot
3-Amino-4-[5-(chloromethyl)-1,2,4-oxadiazol-3-yl]furazan –a multifunctional synthon for the synthesis of 1,2,5-oxadiazole derivatives
inferred← citeshttps://doi.org/10.1007/s10600-022-03662-5openalex-snapshot
Synthesis of New Hybrids of Abietic Acid and 1,3,4-Oxadiazoles
inferred← citeshttps://doi.org/10.1007/s10822-013-9676-0openalex-snapshot
Automated molecule editing in molecular design
inferred← citeshttps://doi.org/10.1007/s10822-026-00925-zopenalex-snapshot
Efficient corrosion inhibition performance of mild steel in hydrochloric acid (1 M HCl) by 5,5’-(1,3-phenylenebis(1,3,4-oxadiazole−5,2-diyl))bis(benzene−1,3-diamine): theoretical and electrochemical study
inferred← citeshttps://doi.org/10.1007/s10854-025-16460-wopenalex-snapshot
Sol–gel synthesis and characterization of 2-phenyl-5-(pyridin-4-yl)-1,3,4-oxadiazole thin films: a structural and optical study
inferred← citeshttps://doi.org/10.1007/s10870-022-00930-8openalex-snapshot
Crystal Structure Characterization, Hirshfeld Surface Analysis, and Non-covalent Interactions of 2,5-Bis(4-chlorophenyl)-1,3,4-Oxadiazole
inferred← citeshttps://doi.org/10.1007/s10895-024-03676-yopenalex-snapshot
Synthesis, Spectral Characterization and Photoluminescence of 3-chloro-6-methoxy-2-(methylsulfanyl)quinoxaline in Different Solvents: An Experimental and Theoretical Investigation Using DFT
inferred← citeshttps://doi.org/10.1007/s10989-026-10858-8openalex-snapshot
Synthesis, Antibacterial and Antifungal Studies of 2-Amino-1,3,4-Oxadiazoles/Thiadiazoles Derived from Nα-Fmoc-Amino Acid Thiosemicarbazides
inferred← citeshttps://doi.org/10.1007/s11030-021-10367-4openalex-snapshot
Oxadiazol-based mTOR inhibitors with potent antiproliferative activities: synthetic and computational modeling
inferred← citeshttps://doi.org/10.1007/s11030-021-10375-4openalex-snapshot
A review on synthetic account of 1,2,4-oxadiazoles as anti-infective agents
inferred← citeshttps://doi.org/10.1007/s11030-022-10422-8openalex-snapshot
Cytotoxic effect, enzyme inhibition, and in silico studies of some novel N-substituted sulfonyl amides incorporating 1,3,4-oxadiazol structural motif
inferred← citeshttps://doi.org/10.1007/s11030-022-10562-xopenalex-snapshot
PEG-mediated synthesis, antibacterial, antifungal and antioxidant studies of some new 1,3,5-trisubstituted 2-pyrazolines
inferred← citeshttps://doi.org/10.1007/s11094-014-1158-8openalex-snapshot
Synthesis and Biological Evaluation of a New Series of Pyrazolines as New Anticandidal Agents
inferred← citeshttps://doi.org/10.1007/s11094-018-1806-5openalex-snapshot
Method Development and Stress Degradation Profile of 5-Benzyl-1,3,4-Oxadiazole-2-Thiol Studied by UV Spectroscopy
inferred← citeshttps://doi.org/10.1007/s11094-019-01969-2openalex-snapshot
Synthesis, Structure Elucidation and Antimicrobial Properties of New Bis-1,3,4-Oxadiazole Derivatives
inferred← citeshttps://doi.org/10.1007/s11164-015-2121-3openalex-snapshot
Synthesis and antioxidant evaluation of some new 2-benzoylamino-5-hetaryl-1,3,4-oxadiazoles
inferred← citeshttps://doi.org/10.1007/s11164-015-2290-0openalex-snapshot
Synthesis and biological activity of 1,3,4-oxa(thia)diazole, 1,2,4-triazole-5-(thio)one and S-substituted derivatives of 3-((2-carboxyethyl)phenylamino)propanoic acid
inferred← citeshttps://doi.org/10.1007/s11164-016-2586-8openalex-snapshot
Construction of 1,3-disubstituted 4-oxo-1,4-dihydroquinolines as a potential antibacterial agents
inferred← citeshttps://doi.org/10.1007/s11172-024-4479-0openalex-snapshot
Synthesis and hypoglycemic properties of new derivatives of 3,12-dioxo-5β-cholan-24-oic acid
inferred← citeshttps://doi.org/10.1007/s11224-015-0703-8openalex-snapshot
Density functional theory study of the regio‐ and stereoselectivity of 1,3-dipolar cycloaddition reactions between 2-ethylthio-4-phenyl-1-azetin and some substituted nitrile oxides
inferred← citeshttps://doi.org/10.1007/s11224-018-1203-4openalex-snapshot
Participation of furoxancarbonitrile oxide in [3+2] cycloaddition reaction toward C–N triple bond: a Molecular Electron Density Theory study of regioselectivity and mechanistic aspect
inferred← citeshttps://doi.org/10.1007/s12039-015-0834-xopenalex-snapshot
T3P as an efficient cyclodehydration reagent for the one-pot synthesis of 2-amino-1,3,4-oxadiazoles
inferred← citeshttps://doi.org/10.1007/s13738-014-0542-3openalex-snapshot
One-pot synthesis of 1,2,4-oxadiazoles from carboxylic acids using 4-(dimethylamino)pyridinium acetate as efficient, regenerable, and green catalyst with ionic liquid character
inferred← citeshttps://doi.org/10.1007/s13738-016-0813-2openalex-snapshot
Synthesis of bifunctional thieno[3,2-c]pyrazole, pyrazolothieno[2,3-d]pyrimidin derivatives and their antimicrobial activities
inferred← citeshttps://doi.org/10.1007/s13738-016-0879-xopenalex-snapshot
Mechanism of 1,3-dipolar cycloaddition reactions of indan-1-one enamines with aryl nitrile oxide: a DFT analysis
inferred← citeshttps://doi.org/10.1007/s13738-021-02335-4openalex-snapshot
Oxadiazoles: moiety to synthesis and utilize
inferred← citeshttps://doi.org/10.1007/s13738-024-03067-xopenalex-snapshot
Synthesis of novel oxadiazole derivatives: DFT calculations, molecular docking studies, and in vitro, in vivo evaluation of antidiabetic activity using Drosophila melanogaster model
inferred← citeshttps://doi.org/10.1007/s40203-024-00261-wopenalex-snapshot
Discovery, lead identification and exploration of potential oxadiazole derivatives in targeting STAT3 as anti-cancer agents
inferred← citeshttps://doi.org/10.1007/s40242-013-2490-3openalex-snapshot
Design and synthesis of hydrazine and oxadiazole-containing derivatives of Sorafenib as antitumor agents
inferred← citeshttps://doi.org/10.1007/s42250-018-00034-xopenalex-snapshot
Synthesis, Cytotoxicity and Antimicrobial Evaluation of Some New 2-Aryl,5-Substituted 1,3,4-Oxadiazoles and 1,3,4-Thiadiazoles
inferred← citeshttps://doi.org/10.1007/s44371-026-00987-wopenalex-snapshot
QSAR modelling and molecular docking studies of 3-(Pyridine-3-yl)-2-oxazolidinone derivatives as potential antibacterial agents against gram-positive pathogens
inferred← citeshttps://doi.org/10.1007/s44442-025-00036-8openalex-snapshot
Oxadiazoles as multi-target therapeutic agents in Alzheimer’s Disease: A review of cholinesterase, MAO, β-Secretase, and Aβ aggregation inhibition
inferred← citeshttps://doi.org/10.1016/b978-0-08-102237-5.00011-0openalex-snapshot
Synthesis and Biological Significance of Six- and Seven-membered Vicinal Diaryl Heterocycles
inferred← citeshttps://doi.org/10.1016/b978-0-12-409547-2.12347-9openalex-snapshot
Matched Molecular Pair Analysis
inferred← citeshttps://doi.org/10.1016/bs.adioch.2019.10.001openalex-snapshot
Antimony and bismuth as antimicrobial agents
inferred← citeshttps://doi.org/10.1016/bs.aihch.2015.05.001openalex-snapshot
Recent Advances in the Chemistry of 1,2,4-OxadiazolesaaDedicated to Professor Nicolò Vivona on the occasion of his 75th birthday.
inferred← citeshttps://doi.org/10.1016/bs.aihch.2016.11.002openalex-snapshot
A Synopsis of the Properties and Applications of Heteroaromatic Rings in Medicinal Chemistry
inferred← citeshttps://doi.org/10.1016/j.arabjc.2013.12.020openalex-snapshot
Synthesis and biological evaluation of newer analogues of 2,5-disubstituted 1,3,4-oxadiazole containing pyrazole moiety as antimicrobial agents
inferred← citeshttps://doi.org/10.1016/j.bioorg.2016.02.007openalex-snapshot
Combretastatin linked 1,3,4-oxadiazole conjugates as a Potent Tubulin Polymerization inhibitors
inferred← citeshttps://doi.org/10.1016/j.bioorg.2016.10.003openalex-snapshot
Design, synthesis, evaluation and molecular modelling studies of some novel 5,6-diphenyl-1,2,4-triazin-3(2H)-ones bearing five-member heterocyclic moieties as potential COX-2 inhibitors: A hybrid pharmacophore approach
inferred← citeshttps://doi.org/10.1016/j.bioorg.2019.01.067openalex-snapshot
Design, synthesis, and cytotoxicity screening of 5-aryl-3-(2-(pyrrolyl) thiophenyl)-1, 2, 4-oxadiazoles as potential antitumor molecules on breast cancer MCF-7 cells
inferred← citeshttps://doi.org/10.1016/j.bioorg.2020.103567openalex-snapshot
Synthesis and evaluation of novel S-benzyl- and S-alkylphthalimide- oxadiazole -benzenesulfonamide hybrids as inhibitors of dengue virus protease
inferred← citeshttps://doi.org/10.1016/j.bioorg.2021.104752openalex-snapshot
Antiproliferative activity, enzymatic inhibition and apoptosis-promoting effects of benzoxazole-based hybrids on human breast cancer cells
inferred← citeshttps://doi.org/10.1016/j.bioorg.2021.105068openalex-snapshot
Investigation of indole functionalized pyrazoles and oxadiazoles as anti-inflammatory agents: Synthesis, in-vivo, in-vitro and in-silico analysis
inferred← citeshttps://doi.org/10.1016/j.bioorg.2021.105176openalex-snapshot
New N-(1,3,4-thiadiazol-2-yl)furan-2-carboxamide derivatives as potential inhibitors of the VEGFR-2
inferred← citeshttps://doi.org/10.1016/j.bioorg.2022.105921openalex-snapshot
Applications of “linkers” in fragment-based drug design
inferred← citeshttps://doi.org/10.1016/j.bioorg.2024.107258openalex-snapshot
Design, synthesis, biological evaluation and docking study of some new aryl and heteroaryl thiomannosides as FimH antagonists
inferred← citeshttps://doi.org/10.1016/j.bioorg.2024.107383openalex-snapshot
Novel 1,3,4-oxadiazole derivatives as highly potent microsomal prostaglandin E2 synthase-1 (mPGES-1) inhibitors
inferred← citeshttps://doi.org/10.1016/j.bioorg.2025.108123openalex-snapshot
Synthesis of bioisosteres of caffeic acid phenethyl ester: 1,3,4-oxadiazole derivatives containing a catechol fragment with anti-inflammatory activities in vitro and in vivo
inferred← citeshttps://doi.org/10.1016/j.bioorg.2025.109353openalex-snapshot
Design and synthesis of new 1,3,4-oxadiazole-1,2,3,4-tetrahydroisoquinoline hybrids as selective COX-2 inhibitors
inferred← citeshttps://doi.org/10.1016/j.bioorg.2026.110578openalex-snapshot
Novel pyrimidine-based N-Acylhydrazones as dual AChE inhibitors and antioxidants targeting Alzheimer's disease
inferred← citeshttps://doi.org/10.1016/j.bioorg.2026.110634openalex-snapshot
5-indole-appended 1,3,4-Oxadiazole/Oxadiazolinethione hybrids: Synthesis, crystal structure, antimicrobial and antibiofilm evaluation
inferred← citeshttps://doi.org/10.1016/j.bmc.2012.08.047openalex-snapshot
Optimization of anti-Trypanosoma cruzi oxadiazoles leads to identification of compounds with efficacy in infected mice
inferred← citeshttps://doi.org/10.1016/j.bmc.2012.10.057openalex-snapshot
Search for α3β2/3γ2 subtype selective ligands that are stable on human liver microsomes
inferred← citeshttps://doi.org/10.1016/j.bmc.2012.10.058openalex-snapshot
Design, synthesis and characterization of novel 1,2-benzisothiazol-3(2H)-one and 1,3,4-oxadiazole hybrid derivatives: Potent inhibitors of Dengue and West Nile virus NS2B/NS3 proteases
inferred← citeshttps://doi.org/10.1016/j.bmc.2014.02.013openalex-snapshot
Synthesis and methemoglobinemia-inducing properties of benzocaine isosteres designed as humane rodenticides
inferred← citeshttps://doi.org/10.1016/j.bmc.2014.10.037openalex-snapshot
New potent antibacterials against Gram-positive multiresistant pathogens: Effects of side chain modification and chirality in linezolid-like 1,2,4-oxadiazoles
inferred← citeshttps://doi.org/10.1016/j.bmc.2017.03.038openalex-snapshot
Discovery of a series of 1,3,4-oxadiazole-2(3H)-thione derivatives containing piperazine skeleton as potential FAK inhibitors
inferred← citeshttps://doi.org/10.1016/j.bmc.2019.02.031openalex-snapshot
Design and development of novel N-(pyrimidin-2-yl)-1,3,4-oxadiazole hybrids to treat cognitive dysfunctions
inferred← citeshttps://doi.org/10.1016/j.bmc.2020.115888openalex-snapshot
Synthetic approaches to unsymmetrical 2,5-disubstituted 1,3,4-oxadiazoles and their MAO-B inhibitory activity. A review
inferred← citeshttps://doi.org/10.1016/j.bmc.2023.117194openalex-snapshot
The most common linkers in bioactive molecules and their bioisosteric replacement network
inferred← citeshttps://doi.org/10.1016/j.bmc.2023.117292openalex-snapshot
Design and synthesis of thiadiazole-oxadiazole-acetamide derivatives: Elastase inhibition, cytotoxicity, kinetic mechanism, and computational studies
inferred← citeshttps://doi.org/10.1016/j.bmcl.2012.03.067openalex-snapshot
Synthesis and SAR of 1,3-thiazolyl thiophene and pyridine derivatives as potent, orally active and S1P3-sparing S1P1 agonists
inferred← citeshttps://doi.org/10.1016/j.bmcl.2012.10.117openalex-snapshot
Inhibitors of HIV-1 attachment. Part 8: The effect of C7-heteroaryl substitution on the potency, and in vitro and in vivo profiles of indole-based inhibitors
inferred← citeshttps://doi.org/10.1016/j.bmcl.2013.05.059openalex-snapshot
Synthesis and structure–activity relationship of 2-arylamino-4-aryl-pyrimidines as potent PAK1 inhibitors
inferred← citeshttps://doi.org/10.1016/j.bmcl.2015.11.046openalex-snapshot
Synthesis and multiparametric evaluation of thiadiazoles and oxadiazoles as diacylglycerol acyltransferase type 1 inhibitors
inferred← citeshttps://doi.org/10.1016/j.bmcl.2016.01.068openalex-snapshot
Syntheses and biological evaluation of 1,2,3-triazole and 1,3,4-oxadiazole derivatives of imatinib
inferred← citeshttps://doi.org/10.1016/j.bmcl.2016.04.058openalex-snapshot
Design and evaluation of novel oxadiazole derivatives as potential prostate cancer agents
inferred← citeshttps://doi.org/10.1016/j.bmcl.2016.08.072openalex-snapshot
Evolution of physicochemical properties of melanin concentrating hormone receptor 1 (MCHr1) antagonists
inferred← citeshttps://doi.org/10.1016/j.bmcl.2016.12.034openalex-snapshot
Synthetic strategy for increasing solubility of potential FLT3 inhibitor thieno[2,3-d]pyrimidine derivatives through structural modifications at the C2 and C6 positions
inferred← citeshttps://doi.org/10.1016/j.bmcl.2017.09.041openalex-snapshot
Improvement in aqueous solubility achieved via small molecular changes
inferred← citeshttps://doi.org/10.1016/j.bmcl.2018.01.011openalex-snapshot
Design and synthesis of novel dasatinib derivatives as inhibitors of leukemia stem cells
inferred← citeshttps://doi.org/10.1016/j.bmcl.2019.06.054openalex-snapshot
Oxadiazole scaffolds in anti-tuberculosis drug discovery
inferred← citeshttps://doi.org/10.1016/j.bmcl.2019.07.033openalex-snapshot
Applications of amide isosteres in medicinal chemistry
inferred← citeshttps://doi.org/10.1016/j.bmcl.2019.126853openalex-snapshot
Design and evaluation of Nrf2 activators with 1,3,4-oxa/thiadiazole core as neuro-protective agents against oxidative stress in PC-12 cells
inferred← citeshttps://doi.org/10.1016/j.bmcl.2020.127136openalex-snapshot
Synthesis of novel of 2, 5-disubstituted 1, 3, 4- oxadiazole derivatives and their in vitro anti-inflammatory, anti-oxidant evaluation, and molecular docking study
inferred← citeshttps://doi.org/10.1016/j.bmcl.2020.127174openalex-snapshot
Discovery and optimization of new oxadiazole substituted thiazole RORγt inverse agonists through a bioisosteric amide replacement approach
inferred← citeshttps://doi.org/10.1016/j.bmcl.2020.127433openalex-snapshot
Optimization of a series of potent, selective and orally bioavailable SYK inhibitors
inferred← citeshttps://doi.org/10.1016/j.bmcl.2020.127612openalex-snapshot
An efficient synthesis tetrazole and oxadiazole analogues of novel 2′-deoxy-C-nucleosides and their antitumor activity
inferred← citeshttps://doi.org/10.1016/j.bmcl.2021.128112openalex-snapshot
Green synthesis of therapeutically active 1,3,4-oxadiazoles as antioxidants, selective COX-2 inhibitors and their in silico studies
inferred← citeshttps://doi.org/10.1016/j.bmcl.2025.130315openalex-snapshot
Design, synthesis, and evaluation of 1,3,4-oxadiazole-based EGFR inhibitors
inferred← citeshttps://doi.org/10.1016/j.cbi.2015.08.018openalex-snapshot
Antioxidant and anti-inflammatory properties of 1,2,4-oxadiazole analogs of resveratrol
inferred← citeshttps://doi.org/10.1016/j.cclet.2013.05.032openalex-snapshot
Electrosynthesis of oxadiazoles from benzoylhydrazines
inferred← citeshttps://doi.org/10.1016/j.ccr.2024.216408openalex-snapshot
Current state of the art of gold complexes as antileishmanial agents
inferred← citeshttps://doi.org/10.1016/j.cdc.2021.100735openalex-snapshot
Synthesis and biological evaluation of 1,2,4-oxadiazole incorporated 1,2,3-triazole-pyrazole derivatives as anticancer agents
inferred← citeshttps://doi.org/10.1016/j.cdc.2023.101031openalex-snapshot
Synthesis, in vitro α-glucosidase and α-amylase activities and molecular docking study of oxadiazole-sulphonamide hybrid analogues
inferred← citeshttps://doi.org/10.1016/j.csbj.2016.12.003openalex-snapshot
Matched Molecular Pair Analysis in Short: Algorithms, Applications and Limitations
inferred← citeshttps://doi.org/10.1016/j.drudis.2013.03.003openalex-snapshot
Matched Molecular Pair Analysis in drug discovery
inferred← citeshttps://doi.org/10.1016/j.ejmcr.2024.100150openalex-snapshot
Synthetic marvels in tuberculosis research: An in-depth review of 1,3,4-oxadiazole derivatives as antitubercular agents
inferred← citeshttps://doi.org/10.1016/j.ejmech.2012.06.006openalex-snapshot
Structure-based optimization of oxadiazole-based GSK-3 inhibitors
inferred← citeshttps://doi.org/10.1016/j.ejmech.2013.01.038openalex-snapshot
Synthesis and antifungal activity of 3-(1,3,4-oxadiazol-5-yl)-indoles and 3-(1,3,4-oxadiazol-5-yl)methyl-indoles
inferred← citeshttps://doi.org/10.1016/j.ejmech.2014.04.045openalex-snapshot
Design and synthesis of novel 2-phenyl-5-(1,3-diphenyl-1H-pyrazol-4-yl)-1,3,4-oxadiazoles as selective COX-2 inhibitors with potent anti-inflammatory activity
inferred← citeshttps://doi.org/10.1016/j.ejmech.2015.08.051openalex-snapshot
Synthesis and SAR of Imidazo[1,5-a]pyridine derivatives as 5-HT4 receptor partial agonists for the treatment of cognitive disorders associated with Alzheimer's disease
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