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Identification of Antitubercular Benzothiazinone Compounds by Ligand-Based Design

https://doi.org/10.1021/jm3008882
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Outgoing claims: the papers this work cites, builds on, or argues with.

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High throughput solubility measurement in drug discovery and development
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A facile procedure for acetalization under aprotic conditions
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Global tuberculosis drug development pipeline: the need and the reality
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Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings
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Comparison of Nephelometric, UV-Spectroscopic, and HPLC Methods for High-Throughput Determination of Aqueous Drug Solubility in Microtiter Plates
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A High-Throughput Screening Method for the Determination of Aqueous Drug Solubility Using Laser Nephelometry in Microtiter Plates
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Estimation of Aqueous Solubility of Chemical Compounds Using E-State Indices
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Benzothiazinones: Prodrugs That Covalently Modify the Decaprenylphosphoryl-β- d -ribose 2′-epimerase DprE1 of Mycobacterium tuberculosis
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Biosynthesis of D ‐arabinose in mycobacteria – a novel bacterial pathway with implications for antimycobacterial therapy
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Benzothiazinones Kill Mycobacterium tuberculosis by Blocking Arabinan Synthesis
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Decaprenylphosphoryl Arabinofuranose, the Donor of the d -Arabinofuranosyl Residues of Mycobacterial Arabinan, Is Formed via a Two-Step Epimerization of Decaprenylphosphoryl Ribose
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Analogous Mechanisms of Resistance to Benzothiazinones and Dinitrobenzamides in Mycobacterium smegmatis

What points at this work

Incoming claims: where this work appears in other papers’ reference lists and arguments.

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Bioevaluation of quinoline‐4‐carbonyl derivatives of piperazinyl‐benzothiazinones as promising antimycobacterial agents
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Molecular Insight into the Discrepancy of Antitubercular Activity between 8‐Nitro and 8‐Cyano Benzothiazinones
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Recent Advancements in Benzothiazinones (BTZ) Analogs as DprE1 Inhibitor for Potent Antitubercular Therapeutics
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Design, synthesis and antimycobacterial activity of novel nitrobenzamide derivatives
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hERG optimizations of IMB1603, discovery of alternative benzothiazinones as new antitubercular agents
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Benzothiozinone derivatives with anti-tubercular Activity−Further side chain investigation
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Replacement of the essential nitro group by electrophilic warheads towards nitro-free antimycobacterial benzothiazinones
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SYNTHESIS AND ANTITUBERCULAR EVALUATION OF FLUORINATED 2-CYCLOALKYLIMINO SUBSTITUTED 1,3-BENZOTHIAZIN-4-ONES
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Modulators targeting protein-protein interactions in Mycobacterium tuberculosis
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Development of Predictive Classification Models for Whole Cell Antimycobacterial Activity of Benzothiazinones
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Fluorescent Benzothiazinone Analogues Efficiently and Selectively Label Dpre1 in Mycobacteria and Actinobacteria
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