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Voltage-Gated Sodium Channels: Structure, Function, Pharmacology, and Clinical Indications
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Outgoing claims: the papers this work cites, builds on, or argues with.
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inferredcites →https://doi.org/10.1002/ejp.567openalex-snapshotA systematic review of therapeutic interventions to reduce acute and chronic post‐surgical pain after amputation, thoracotomy or mastectomy
inferredcites →https://doi.org/10.1002/ijc.28890openalex-snapshotThe sodium channel β1 subunit mediates outgrowth of neurite‐like processes on breast cancer cells and promotes tumour growth and metastasis
inferredcites →https://doi.org/10.1007/s00018-003-2354-xopenalex-snapshotIsolation and characterization of hainantoxin-IV, a novel antagonist of tetrodotoxin-sensitive sodium channels from the Chinese bird spider Selenocosmia hainana
inferredcites →https://doi.org/10.1007/s10989-013-9389-1openalex-snapshotRoles of Individual Disulfide Bridges in the Conformation and Activity of μ-Conotoxin GIIIA, a Peptide Blocker of Muscle Sodium Channels
inferredcites →https://doi.org/10.1016/j.bmc.2012.03.034openalex-snapshotSolution NMR analysis of the binding mechanism of DIVS6 model peptides of voltage-gated sodium channels and the lipid soluble alkaloid veratridine
inferredcites →https://doi.org/10.1016/j.jmb.2013.10.010openalex-snapshotStructure of a Prokaryotic Sodium Channel Pore Reveals Essential Gating Elements and an Outer Ion Binding Site Common to Eukaryotic Channels
inferredcites →https://doi.org/10.1016/j.toxicon.2006.07.032openalex-snapshotSpecies selective resistance of cardiac muscle voltage gated sodium channels: Characterization of brevetoxin and ciguatoxin binding sites in rats and fish
inferredcites →https://doi.org/10.1016/j.toxicon.2013.01.014openalex-snapshotThe venom of the fishing spider Dolomedes sulfurous contains various neurotoxins acting on voltage-activated ion channels in rat dorsal root ganglion neurons
inferredcites →https://doi.org/10.1016/j.toxicon.2013.05.015openalex-snapshotSynthesis and biological characterization of synthetic analogs of Huwentoxin-IV (Mu-theraphotoxin-Hh2a), a neuronal tetrodotoxin-sensitive sodium channel inhibitor
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inferredcites →https://doi.org/10.1021/cb400012kopenalex-snapshotChemical Engineering and Structural and Pharmacological Characterization of the α-Scorpion Toxin OD1
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inferredcites →https://doi.org/10.1021/jm500687uopenalex-snapshotStudies Examining the Relationship between the Chemical Structure of Protoxin II and Its Activity on Voltage Gated Sodium Channels
inferredcites →https://doi.org/10.1021/jo00087a027openalex-snapshotConformational Analysis of the Sodium Channel Modulator, Brevetoxin A, Comparison with Brevetoxin B Conformations, and a Hypothesis about the Common Pharmacophore of the "Site 5" Toxins
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inferredcites →https://doi.org/10.1038/9195openalex-snapshotThe tetrodotoxin-resistant sodium channel SNS has a specialized function in pain pathways
inferredcites →https://doi.org/10.1038/nm.2750openalex-snapshotMethylglyoxal modification of Nav1.8 facilitates nociceptive neuron firing and causes hyperalgesia in diabetic neuropathy
inferredcites →https://doi.org/10.1042/bj20131275openalex-snapshotNedd4-2 (NEDD4L) controls intracellular Na+-mediated activity of voltage-gated sodium channels in primary cortical neurons
inferredcites →https://doi.org/10.1073/pnas.0400368101openalex-snapshotThe structure of zetekitoxin AB, a saxitoxin analog from the Panamanian golden frog Atelopus zeteki : A potent sodium-channel blocker
inferredcites →https://doi.org/10.1073/pnas.1107027108openalex-snapshotμ-Conotoxins that differentially block sodium channels Na V 1.1 through 1.8 identify those responsible for action potentials in sciatic nerve
inferredcites →https://doi.org/10.1073/pnas.1306285110openalex-snapshotDiscovery of a selective Na V 1.7 inhibitor from centipede venom with analgesic efficacy exceeding morphine in rodent pain models
inferredcites →https://doi.org/10.1073/pnas.1309827110openalex-snapshotNonfunctional Na V 1.1 familial hemiplegic migraine mutant transformed into gain of function by partial rescue of folding defects
inferredcites →https://doi.org/10.1073/pnas.75.6.2606openalex-snapshotPurification of the tetrodotoxin-binding component associated with the voltage-sensitive sodium channel from Electrophorus electricus electroplax membranes.
inferredcites →https://doi.org/10.1074/jbc.m309576200openalex-snapshotA δ-Conotoxin from Conus ermineus Venom Inhibits Inactivation in Vertebrate Neuronal Na+ Channels but Not in Skeletal and Cardiac Muscles
inferredcites →https://doi.org/10.1074/jbc.m704616200openalex-snapshotStructure/Function Characterization of μ-Conotoxin KIIIA, an Analgesic, Nearly Irreversible Blocker of Mammalian Neuronal Sodium Channels
inferredcites →https://doi.org/10.1085/jgp.201310984openalex-snapshotInteractions among DIV voltage-sensor movement, fast inactivation, and resurgent Na current induced by the NaVβ4 open-channel blocking peptide
inferredcites →https://doi.org/10.1093/brain/awr143openalex-snapshotDeletion mutation of sodium channel NaV1.7 in inherited erythromelalgia: enhanced slow inactivation modulates dorsal root ganglion neuron hyperexcitability
inferredcites →https://doi.org/10.1111/bph.12051openalex-snapshotCo‐expression of NaVβ subunits alters the kinetics of inhibition of voltage‐gated sodium channels by pore‐blocking μ‐conotoxins
inferredcites →https://doi.org/10.1111/bph.12119openalex-snapshotPharmacological fractionation of tetrodotoxin‐sensitive sodium currents in rat dorsal root ganglion neurons by μ‐conotoxins
inferredcites →https://doi.org/10.1124/pr.57.4.4openalex-snapshotInternational Union of Pharmacology. XLVII. Nomenclature and Structure-Function Relationships of Voltage-Gated Sodium Channels
inferredcites →https://doi.org/10.1172/jci40801openalex-snapshotHuman voltage-gated sodium channel mutations that cause inherited neuronal and muscle channelopathies increase resurgent sodium currents
inferredcites →https://doi.org/10.1186/1744-8069-10-7openalex-snapshotA Comparison of RNA-Seq and Exon Arrays for Whole Genome Transcription Profiling of the L5 Spinal Nerve Transection Model of Neuropathic Pain in the Rat
inferredcites →https://doi.org/10.1289/ehp.1307196openalex-snapshotCiguatera Fish Poisoning and Climate Change: Analysis of National Poison Center Data in the United States, 2001–2011
inferredcites →https://doi.org/10.2183/pjab.90.56openalex-snapshotChemical construction and structural permutation of neurotoxic natural product, antillatoxin: importance of the three-dimensional structure of the bulky side chain
inferredcites →https://doi.org/10.3390/ijms14059779openalex-snapshotEffects of (−)-Gallocatechin-3-Gallate on Tetrodotoxin-Resistant Voltage-Gated Sodium Channels in Rat Dorsal Root Ganglion Neurons
inferredcites →https://doi.org/10.3390/toxins6030816openalex-snapshotCharacterization of a Novel BmαTX47 Toxin Modulating Sodium Channels: The Crucial Role of Expression Vectors in Toxin Pharmacological Activity
inferredcites →https://doi.org/10.3892/ol.2014.2110openalex-snapshotVoltage-gated sodium channels were differentially expressed in human normal prostate, benign prostatic hyperplasia and prostate cancer cells
inferredcites →https://doi.org/10.5740/jaoacint.sgemccallopenalex-snapshotDevelopment and Utilization of a Fluorescence-Based Receptor-Binding Assay for the Site 5 Voltage-Sensitive Sodium Channel Ligands Brevetoxin and Ciguatoxin
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inferred← citeshttps://doi.org/10.1002/wcms.1641openalex-snapshotRecent advances in computational studies on voltage‐gated sodium channels: Drug design and mechanism studies
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