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Application of Quantitative Structure−Activity Relationships to the Modeling of Antitubercular Compounds. 1. The Hydrazide Family

https://doi.org/10.1021/jm701048s
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Outgoing claims: the papers this work cites, builds on, or argues with.

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Crystal Structure of Mycobacterium tuberculosis Catalase-Peroxidase
inferredcites →https://doi.org/10.1074/jbc.m402384200openalex-snapshot
Enzyme-catalyzed Mechanism of Isoniazid Activation in Class I and Class III Peroxidases
inferredcites →https://doi.org/10.1074/jbc.m406374200openalex-snapshot
Catalase-peroxidases (KatG) Exhibit NADH Oxidase Activity
inferredcites →https://doi.org/10.1093/jac/49.2.275openalex-snapshot
Activity of a new class of isonicotinoylhydrazones used alone and in combination with isoniazid, rifampicin, ethambutol, para-aminosalicylic acid and clofazimine against Mycobacterium tuberculosis
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Modification of the NADH of the Isoniazid Target (InhA) from Mycobacterium tuberculosis
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inferredcites →https://doi.org/10.1128/aac.47.2.670-675.2003openalex-snapshot
Isoniazid Activation Defects in Recombinant Mycobacterium tuberculosis Catalase-Peroxidase (KatG) Mutants Evident in InhA Inhibitor Production
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Influential Observations, High Leverage Points, and Outliers in Linear Regression
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What points at this work

Incoming claims: where this work appears in other papers’ reference lists and arguments.

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Computational Models for Tuberculosis Drug Discovery
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The contribution of the hydrogen bond acidity on the lipophilicity of drugs estimated from chromatographic measurements
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