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Structure−Activity Relationships of Selective Estrogen Receptor Modulators: Modifications to the 2-Arylbenzothiophene Core of Raloxifene
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What this work says
Outgoing claims: the papers this work cites, builds on, or argues with.
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A controlled trial of raloxifene (LY139481) HCl: Impact on bone turnover and serum lipid profile in healthy postmenopausal women
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Oestrogen Replacement Therapy and Cardiovascular Disease
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Alternative mechanisms of action of anti-oestrogens
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A kinetic assay for eosinophil peroxidase activity in eosinophils and eosinophil conditioned media
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The specificity of the estrogen receptor of human uterus
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A chemical classification of nonsteroidal antagonists of sex-steroid hormone action
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Non-genomic effects of estrogens and antiestrogens
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Site-directed estrogen receptor antibodies stabilize 4-hydroxytamoxifen ligand, but not estradiol, and indicate ligand-specific differences in the recognition of estrogen response element DNA in vitro
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Effect of estradiol and antiestrogens on cholesterol biosynthesis in hormone-dependent and -independent breast cancer cell lines
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Synthesis, binding affinities and uterotrophic activity of some 2-substituted estradiol and ring-A-fused pyrone derivatives
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Design of novel antiestrogens
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Synthesis and pharmacology of 2-alkyl raloxifene analogs
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The biological evaluation of novel antioestrogens for the treatment of breast cancer
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Selective estrogen receptor modulators: pharmacological profile in the rat uterus.
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Time-dependent changes in biochemical bone markers and serum cholesterol in ovariectomized rats: Effects of raloxifene HCl, tamoxifen, estrogen, and alendronate
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Current concepts in estrogen replacement therapy in the menopause
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Hypocholesterolemic Activity of Raloxifene (LY139481): Pharmacological Characterization as a Selective Estrogen Receptor Modulator
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Longitudinal and cross-sectional analysis of raloxifene effects on tibiae from ovariectomized aged rats.
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Osteoporosis: Etiology, Diagnosis, and Management
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Protection of hydroxyl groups as tert-butyldimethylsilyl derivatives
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Renin inhibitors. Synthesis of transition-state analog inhibitors containing phosphorus acid derivatives at the scissile bond
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4-(Phosphonoalkyl)- and 4-(phosphonoalkenyl)-2-piperidinecarboxylic acids: synthesis, activity at N-methyl-D-aspartic acid receptors and anticonvulsant activity
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Antiestrogens. 2. Structure-activity studies in a series of 3-aroyl-2-arylbenzo[b]thiophene derivatives leading to [6-hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl]-[4-[2-(1-piperidinyl)ethoxy]phenyl]methanone hydrochloride (LY 156758), a remarkably effective estrogen antagonist with only minimal…
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2-(Hydroxyalkyl)estradiols: Synthesis and Biological Evaluation
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The Characterization of Complex Phenols by Nuclear Magnetic Resonance Spectra
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Synthetic Transformations of Vinyl and Aryl Triflates
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Estrogen Resistance Caused by a Mutation in the Estrogen-Receptor Gene in a Man
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The Use of Estrogens and Progestins and the Risk of Breast Cancer in Postmenopausal Women
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An Alternative Procedure for the Aluminum-Mediated Conversion of Esters to Amides
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Influence of incomplete cholesteryl ester hydrolysis on enzymic measurements of cholesterol.
inferredcites →https://doi.org/10.1096/fasebj.10.8.8666168openalex-snapshot
Raloxifene, tamoxifen, nafoxidine, or estrogen effects on reproductive and nonreproductive tissues in ovariectomized rats
inferredcites →https://doi.org/10.1111/j.1476-5381.1993.tb13840.xopenalex-snapshot
A current view of tamoxifen for the treatment and prevention of breast cancer
inferredcites →https://doi.org/10.1111/j.1749-6632.1995.tb31374.xopenalex-snapshot
Cellular Mechanisms Which Distinguish between Hormone‐ and Antihormone‐Activated Estrogen Receptor
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Raloxifene (LY139481 HCI) prevents bone loss and reduces serum cholesterol without causing uterine hypertrophy in ovariectomized rats.
inferredcites →https://doi.org/10.1210/edrv-16-1-35openalex-snapshot
Estrogen Receptors in Human Nontarget Tissues: Biological and Clinical Implications*
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Estrogen and raloxifene stimulate transforming growth factor-beta 3 gene expression in rat bone: a potential mechanism for estrogen- or raloxifene-mediated bone maintenance
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Tripartite steroid hormone receptor pharmacology: interaction with multiple effector sites as a basis for the cell- and promoter-specific action of these hormones
inferredcites →https://doi.org/10.1210/me.9.6.659openalex-snapshot
Analysis of estrogen receptor function in vitro reveals three distinct classes of antiestrogens
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A Mild Selective Monobromination Reagent System for Alkoxybenzenes; N-Bromosuccinimide–Silica Gel
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The Medicinal Chemistry of Nonsteroidal Antiestrogens: A Review
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Antiestrogens as Calmodulin Antagonists
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Pyridine-Substituted Hydroxythiophenes. I. Preparation of o-(2-, 3- and 4-pyridyl)-3-hydroxythiophenes.
What points at this work
Incoming claims: where this work appears in other papers’ reference lists and arguments.
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Effects of Raloxifene on Serum Lipids and Coagulation Factors in Healthy Postmenopausal Women
inferred← citeshttps://doi.org/10.1002/0471266949.bmc054openalex-snapshot
Female Sex Hormones, Contraceptives, And Fertility Drugs
inferred← citeshttps://doi.org/10.1002/0471266949.bmc054.pub2openalex-snapshot
Estrogen Receptor Modulators
inferred← citeshttps://doi.org/10.1002/9780470768594.ch20openalex-snapshot
Raloxifene, Evista: A Selective Estrogen Receptor Modulator (SERM)
inferred← citeshttps://doi.org/10.1002/9781118219683.ch15openalex-snapshot
Raloxifene: A Selective Estrogen Receptor Modulator (SERM)
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Subtype‐Selective Estrogens
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Transition‐Metal‐Free Synthesis of Heterobiaryls through 1,2‐Migration of Boronate Complex
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Structure–Activity Relationships for a Family of Benzothiophene Selective Estrogen Receptor Modulators Including Raloxifene and Arzoxifene
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Tamoxifen and Other Antiestrogens in Prevention and Therapy of Breast Cancer
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Androgen Replacement Therapy of Male Hypogonadism
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Structural Insights into Estrogen Receptors and Antiestrogen Therapies
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Antiestrogens and Partial Agonists
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Structure-Activity Relationships
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Selective Estrogen Receptor Modulators (SERMs)
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LIV-3D-QSAR model for estrogen receptor ligands
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Acylation of 3-acyl-2-methylbenzo[b]thiophene
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Identification of a series of tetrahydroisoquinoline derivatives as potential therapeutic agents for breast cancer
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Structure–activity relationships of SERMs optimized for uterine antagonism and ovarian safety
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A mutant selective anti-estrogen is a pure antagonist on EREs and AP-1 response elements
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3-Phenyl-1H-5-pyrazolylamine-based derivatives as potent and efficacious inhibitors of FMS-like tyrosine kinase-3 (FLT3)
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6′-Methoxy Raloxifene-analog enhances mouse bone properties with reduced estrogen receptor binding
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Benzothiophene nucleus in target-directed anti-cancer drug discovery
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Raloxifene promotes adipocyte differentiation of 3T3-L1 cells
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Pharmacophore mapping of arylbenzothiophene derivatives for MCF cell inhibition using classical and 3D space modeling approaches
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Selective steroid receptor modulators, degraders and PROTACs: Therapeutic strategies in management of endocrine-related cancers
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Selective estrogen receptor modulators (SERMs) and selective estrogen receptor degraders (SERDs) in cancer treatment
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Plant 2-arylobenzofurans demonstrate a selective estrogen receptor modulator profile
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Three-dimensional models of non-steroidal ligands: A comparative molecular field analysis
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Characterization of Bizzy Nut extracts in estrogen-responsive MCF-7 breast cancer cells
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A convenient approach towards 2- and 3-aminobenzo[b]thiophenes
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Efficient synthesis of 3-benzoyl Benzo[b]thiophenes and raloxifene via Mercury(II)-Catalyzed cyclization of 2-alkynylphenyl alkyl sulfoxides
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Efficient synthesis of 3-oxygenated benzothiophene derivatives
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Bromination of 3-substituted benzo[b]thiophenes: access to Raloxifen intermediate
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Characterization of selective estrogen receptor modulator (SERM) activity in two triarylethylene oxybutyric acids
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Basic Guide to the Mechanisms of Antiestrogen Action
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Nucleophilic aromatic substitution on 3-aroyl-2-arylbenzothiophenes. Rapid access to raloxifene and other selective estrogen receptor modulators
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Synergistic methodologies for the synthesis of 3-aroyl-2-arylbenzo[b]thiophene-based selective estrogen receptor modulators. Two concise syntheses of raloxifene
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Chapter 15. Targeting the estrogen receptor with SERMs
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QSAR models in receptor-mediated effects: the nuclear receptor superfamily
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CHEMOPREVENTION OF BREAST CANCER IN THE OLDER PATIENT
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BREAST CANCER CHEMOPREVENTION
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7 Other medical management of uterine fibroids
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Solid-Phase synthesis and investigation of benzofurans as selective estrogen receptor modulators
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Novel nonsteroidal selective estrogen receptor modulators. Carbon and heteroatom replacement of oxygen in the ethoxypiperidine region of raloxifene
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Dibasic benzo[b]thiophene derivatives as a novel class of active site directed thrombin inhibitors: 4. SAR studies on the conformationally restricted C3-side chain of hydroxybenzo[b]thiophenes
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A new anti-tubulin agent containing the benzo[b]thiophene ring system
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The first organometallic antioestrogens and their antiproliferative effects
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Bioanalytical High-Throughput Selected Reaction Monitoring-LC/MS Determination of Selected Estrogen Receptor Modulators in Human Plasma: 2000 Samples/Day
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From Bones to Bugs: Structure-Based Development of Raloxifene-Derived Pathoblockers That Inhibit Pyocyanin Production in Pseudomonas aeruginosa
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Identification of GDC-0810 (ARN-810), an Orally Bioavailable Selective Estrogen Receptor Degrader (SERD) that Demonstrates Robust Activity in Tamoxifen-Resistant Breast Cancer Xenografts
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Selective Human Estrogen Receptor Partial Agonists (ShERPAs) for Tamoxifen-Resistant Breast Cancer
inferred← citeshttps://doi.org/10.1021/acs.jmedchem.7b01682openalex-snapshot
Discovery of LSZ102, a Potent, Orally Bioavailable Selective Estrogen Receptor Degrader (SERD) for the Treatment of Estrogen Receptor Positive Breast Cancer
inferred← citeshttps://doi.org/10.1021/acsmedchemlett.4c00078openalex-snapshot
Synthesis Studies and the Evaluation of C6 Raloxifene Derivatives
inferred← citeshttps://doi.org/10.1021/bi0205092openalex-snapshot
Identification by MALDI-TOF Mass Spectrometry of 17α-Bromoacetamidopropylestradiol Covalent Attachment Sites on Estrogen Receptor α
inferred← citeshttps://doi.org/10.1021/bi9919706openalex-snapshot
The Major Cyclic Trimeric Product of Indole-3-carbinol Is a Strong Agonist of the Estrogen Receptor Signaling Pathway
inferred← citeshttps://doi.org/10.1021/ci2004779openalex-snapshot
Integrating Medicinal Chemistry, Organic/Combinatorial Chemistry, and Computational Chemistry for the Discovery of Selective Estrogen Receptor Modulators with F orecaster , a Novel Platform for Drug Discovery
inferred← citeshttps://doi.org/10.1021/ci200540yopenalex-snapshot
A Scaffold-Independent Subcellular Event-Based Analysis: Characterization of Significant Structural Modifications
inferred← citeshttps://doi.org/10.1021/ci900254bopenalex-snapshot
Pharmacophore Modeling for Qualitative Prediction of Antiestrogenic Activity
inferred← citeshttps://doi.org/10.1021/co100088qopenalex-snapshot
Highly Substituted Lactone/Ester-Containing Furan Library by the Palladium-Catalyzed Carbonylation of Hydroxyl-Substituted 3-Iodofurans
inferred← citeshttps://doi.org/10.1021/co200090popenalex-snapshot
Parallel Synthesis of a Desketoraloxifene Analogue Library via Iodocyclization/Palladium-Catalyzed Coupling
inferred← citeshttps://doi.org/10.1021/cr020101aopenalex-snapshot
Metalated Heterocycles and Their Applications in Synthetic Organic Chemistry
inferred← citeshttps://doi.org/10.1021/cr980018gopenalex-snapshot
Comparative QSAR Analysis of Estrogen Receptor Ligands
inferred← citeshttps://doi.org/10.1021/jm000170mopenalex-snapshot
Pyrazole Ligands: Structure−Affinity/Activity Relationships and Estrogen Receptor-α-Selective Agonists
inferred← citeshttps://doi.org/10.1021/jm010086mopenalex-snapshot
Design, Synthesis, and Preclinical Characterization of Novel, Highly Selective Indole Estrogens
inferred← citeshttps://doi.org/10.1021/jm0101601openalex-snapshot
Photochemical Synthesis of N-Arylbenzophenanthridine Selective Estrogen Receptor Modulators (SERMs)
inferred← citeshttps://doi.org/10.1021/jm020291hopenalex-snapshot
A New Series of Estrogen Receptor Modulators That Display Selectivity for Estrogen Receptor β
inferred← citeshttps://doi.org/10.1021/jm020450xopenalex-snapshot
Antiestrogens and Selective Estrogen Receptor Modulators as Multifunctional Medicines. 2. Clinical Considerations and New Agents
inferred← citeshttps://doi.org/10.1021/jm020536qopenalex-snapshot
De Novo Design, Synthesis, and Evaluation of Novel Nonsteroidal Phenanthrene Ligands for the Estrogen Receptor
inferred← citeshttps://doi.org/10.1021/jm0210562openalex-snapshot
Antiestrogenically Active 1,1,2-Tris(4-hydroxyphenyl)alkenes without Basic Side Chain: Synthesis and Biological Activity
inferred← citeshttps://doi.org/10.1021/jm030086hopenalex-snapshot
Estrogen Receptor Modulators: Identification and Structure−Activity Relationships of Potent ERα-Selective Tetrahydroisoquinoline Ligands
inferred← citeshttps://doi.org/10.1021/jm034243oopenalex-snapshot
Estrogen Receptor Ligands. II. Discovery of Benzoxathiins as Potent, Selective Estrogen Receptor α Modulators
inferred← citeshttps://doi.org/10.1021/jm050723zopenalex-snapshot
A Selective Estrogen Receptor Modulator Designed for the Treatment of Uterine Leiomyoma with Unique Tissue Specificity for Uterus and Ovaries in Rats
inferred← citeshttps://doi.org/10.1021/jm9705521openalex-snapshot
Three-Dimensional Quantitative Structure−Activity Relationship Study of Nonsteroidal Estrogen Receptor Ligands Using the Comparative Molecular Field Analysis/Cross-Validated r2-Guided Region Selection Approach
inferred← citeshttps://doi.org/10.1021/jm970688zopenalex-snapshot
Synthesis and Pharmacology of Conformationally Restricted Raloxifene Analogues: Highly Potent Selective Estrogen Receptor Modulators
inferred← citeshttps://doi.org/10.1021/jm990078uopenalex-snapshot
Carboxylic Acid Analogues of Tamoxifen: (Z)-2-[p-(1,2-Diphenyl-1-butenyl)phenoxy]-N,N-dimethylethylamine. Estrogen Receptor Affinity and Estrogen Antagonist Effects in MCF-7 Cells
inferred← citeshttps://doi.org/10.1021/jo034325kopenalex-snapshot
Synthesis of Constrained Raloxifene Analogues by Complementary Use of Friedel−Crafts and Directed Remote Metalation Reactions
inferred← citeshttps://doi.org/10.1021/jo062141aopenalex-snapshot
One-Pot Synthesis of Substituted 2-Aminobenzo[b]thiophenes
inferred← citeshttps://doi.org/10.1021/jo9711807openalex-snapshot
Parallel Synthesis of Tamoxifen and Derivatives on Solid Support via Resin Capture
inferred← citeshttps://doi.org/10.1021/ml2002532openalex-snapshot
Hydrophobic Interactions Improve Selectivity to ERα for Benzothiophene SERMs
inferred← citeshttps://doi.org/10.1021/ol061859+openalex-snapshot
Synthesis of Polycyclic Heterocycles via a One-Pot Ortho Alkylation/Direct Heteroarylation Sequence
inferred← citeshttps://doi.org/10.1021/ol502381eopenalex-snapshot
Direct Synthesis of Diverse 2-Aminobenzo[b]thiophenes via Palladium-Catalyzed Carbon–Sulfur Bond Formation Using Na2S2O3as the Sulfur Source
inferred← citeshttps://doi.org/10.1021/tx000208yopenalex-snapshot
Structure−Activity Relationships for a Large Diverse Set of Natural, Synthetic, and Environmental Estrogens
inferred← citeshttps://doi.org/10.1021/tx0342722openalex-snapshot
Oxidation of Raloxifene to Quinoids: Potential Toxic Pathways via a Diquinone Methide and o-Quinones
inferred← citeshttps://doi.org/10.1021/tx049776uopenalex-snapshot
Bioactivation of the Selective Estrogen Receptor Modulator Desmethylated Arzoxifene to Quinoids: 4‘-Fluoro Substitution Prevents Quinoid Formation
inferred← citeshttps://doi.org/10.1023/a:1010019410881openalex-snapshot
Mechanism of Action and Preclinical Profile of Raloxifene, a Selective Estrogen Receptor Modulator*
inferred← citeshttps://doi.org/10.1038/39645openalex-snapshot
Molecular basis of agonism and antagonism in the oestrogen receptor
inferred← citeshttps://doi.org/10.1039/b914424bopenalex-snapshot
As many as six tandem reactions in one step! Unprecedented formation of highly functionalized benzothiophenes
inferred← citeshttps://doi.org/10.1039/c5ra02114fopenalex-snapshot
One-pot synthesis of 2,3-substituted benzo[b]thiophenes via Cu( i ) catalysed intramolecular cyclisation from dithioesters
inferred← citeshttps://doi.org/10.1039/c6md00553eopenalex-snapshot
Design and synthesis of novel selective estrogen receptor degradation inducers based on the diphenylheptane skeleton
inferred← citeshttps://doi.org/10.1039/c6ob02461kopenalex-snapshot
A practical synthesis of benzothiophenes via visible-light-promoted cyclization of disulfides and alkynes
inferred← citeshttps://doi.org/10.1039/c7ob01747bopenalex-snapshot
Visible-light-induced tandem cyclization of 2-alkynylanilines with disulfides: a convenient method for accessing benzothiophenes under transition-metal-free and photocatalyst-free conditions
inferred← citeshttps://doi.org/10.1039/c9md00570fopenalex-snapshot
Recent progress in selective estrogen receptor downregulators (SERDs) for the treatment of breast cancer
inferred← citeshttps://doi.org/10.1039/d0gc00917bopenalex-snapshot
Nickel-catalyzed and Li-mediated regiospecific C–H arylation of benzothiophenes
inferred← citeshttps://doi.org/10.1055/a-2500-6460openalex-snapshot
Synthesis of 2-Aminobenzo[b]thiophenes via an Intramolecular Dehydrogenative C–S Bond Formation Effected by Iodine(III) Reagents
inferred← citeshttps://doi.org/10.1073/pnas.142288199openalex-snapshot
Kinetic analysis of estrogen receptor/ligand interactions
inferred← citeshttps://doi.org/10.1073/pnas.94.25.14105openalex-snapshot
Molecular determinants of tissue selectivity in estrogen receptor modulators
inferred← citeshttps://doi.org/10.1080/00397911.2014.943348openalex-snapshot
Piperidine Nucleophilic Substitution Without Solvent: An Efficient Synthesis of Raloxifene
inferred← citeshttps://doi.org/10.1080/01443610310001620305openalex-snapshot
Comparative analysis of oestrogen and raloxifene effects on the phospholipid composition of high density lipoproteins in healthy postmenopausal women
inferred← citeshttps://doi.org/10.1080/01961779908047953openalex-snapshot
Recent Advances in the Synthesis and Applications of Benzo[b]thiophenes
inferred← citeshttps://doi.org/10.1080/08927022.2012.717281openalex-snapshot
Agonist and antagonist recognition studies for oestrogen receptor by molecular dynamics simulation
inferred← citeshttps://doi.org/10.1080/1062936x.2020.1864468openalex-snapshot
Endocrine disruption: the noise in available data adversely impacts the models’ performance
inferred← citeshttps://doi.org/10.1080/14756360802469127openalex-snapshot
β-Lactam type molecular scaffolds for antiproliferative activity: Synthesis and cytotoxic effects in breast cancer cells
inferred← citeshttps://doi.org/10.1080/17415991003721266openalex-snapshot
Recent trends in the chemistry of aminobenzo[b]thiophenes
inferred← citeshttps://doi.org/10.1089/jwh.1999.8.321openalex-snapshot
Selective Estrogen Receptor Modulators: A Controversial Approach for Managing Postmenopausal Health
inferred← citeshttps://doi.org/10.1093/jnci/90.20.1514openalex-snapshot
Cancer Chemoprevention: Progress and Promise
inferred← citeshttps://doi.org/10.1111/cbdd.12239openalex-snapshot
Discovery of Synthetic Leishmania Inhibitors by Screening of a 2‐Arylbenzothiophene Library
inferred← citeshttps://doi.org/10.1111/j.1527-3466.2001.tb00183.xopenalex-snapshot
Cardiovascular Effects of Raloxifene Hydrochloride
inferred← citeshttps://doi.org/10.1134/s1070363218040126openalex-snapshot
A Convenient Approach to 2-Aminobenzo[b]chalcogenophenes Based on Copper-Catalyzed Transformation of 4-(2-Bromophenyl)-1,2,3-chalcogenodiazoles in the Presence of a Base and Amines
inferred← citeshttps://doi.org/10.1134/s107036322011033xopenalex-snapshot
In Vitro Activity of Organochalcogen Compounds: II. Cytotoxic Effect of 2-Aminobenzo[b]thiophenes Against K562 and HeLa Tumor Cell Lines
inferred← citeshttps://doi.org/10.1134/s1070428013040015openalex-snapshot
4-(2-R-Aryl)-1,2,3-chalcogenadiazoles in the synthesis of fused heterocycles
inferred← citeshttps://doi.org/10.1155/2013/743139openalex-snapshot
Computational Study of Estrogen Receptor-Alpha Antagonist with Three-Dimensional Quantitative Structure-Activity Relationship, Support Vector Regression, and Linear Regression Methods
inferred← citeshttps://doi.org/10.1158/1535-7163.mct-14-0319openalex-snapshot
Novel Selective Estrogen Mimics for the Treatment of Tamoxifen-Resistant Breast Cancer
inferred← citeshttps://doi.org/10.1186/s12915-017-0449-4openalex-snapshot
Targeting protein quality control pathways in breast cancer
inferred← citeshttps://doi.org/10.1210/edrv.20.3.0368openalex-snapshot
Tamoxifen, Raloxifene, and the Prevention of Breast Cancer*
inferred← citeshttps://doi.org/10.1248/cpb.52.79openalex-snapshot
A New Series of Estrogen Receptor Modulators: Effect of Alkyl Substituents on Receptor-Binding Affinity
inferred← citeshttps://doi.org/10.1248/cpb.c19-01108openalex-snapshot
Development of Photoswitchable Estrogen Receptor Ligands
inferred← citeshttps://doi.org/10.1289/ehp.00108s5829openalex-snapshot
Influence of Exogenous Estrogen Receptor Ligands on Uterine Leiomyoma: Evidence from an in Vitro/in Vivo Animal Model for Uterine Fibroids
inferred← citeshttps://doi.org/10.1517/13543776.16.5.559openalex-snapshot
Estrogen receptor modulator review
inferred← citeshttps://doi.org/10.1517/13543784.15.3.317openalex-snapshot
Arzoxifene: the development and clinical outcome of an ideal SERM
inferred← citeshttps://doi.org/10.1530/jme-16-0024openalex-snapshot
Antiestrogens: structure-activity relationships and use in breast cancer treatment
inferred← citeshttps://doi.org/10.1586/14737140.4.4.523openalex-snapshot
Raloxifene and its role in breast cancer prevention
inferred← citeshttps://doi.org/10.1590/s0004-27301999000600008openalex-snapshot
Raloxifeno e osteoporose: revisão de um novo modulador seletivo do receptor de estrógeno
inferred← citeshttps://doi.org/10.1787/9789264078857-enopenalex-snapshot
Detailed Background Review of the Uterotrophic Bioassay
inferred← citeshttps://doi.org/10.2147/cia.s3344openalex-snapshot
Managing the risk of invasive breast cancer in women at risk for breast cancer and osteoporosis: the role of raloxifene
inferred← citeshttps://doi.org/10.2165/00002018-200124140-00003openalex-snapshot
Comparative Tolerability of First-Generation Selective Estrogen Receptor Modulators in Breast Cancer Treatment and Prevention
inferred← citeshttps://doi.org/10.2165/00002512-200724050-00002openalex-snapshot
Selective Estrogen Receptor Modulators for Postmenopausal Osteoporosis
inferred← citeshttps://doi.org/10.2165/00003495-200767160-00004openalex-snapshot
Estrogen Receptor Modulators and Down Regulators
inferred← citeshttps://doi.org/10.2174/0929867329666221006110528openalex-snapshot
Effectiveness of Selective Estrogen Receptor Modulators in Breast Cancer Therapy: An Update
inferred← citeshttps://doi.org/10.2174/1574884711308020006openalex-snapshot
The Discovery and Development of Selective Estrogen Receptor Modulators (SERMs) for Clinical Practice
inferred← citeshttps://doi.org/10.2217/17455057.3.2.139openalex-snapshot
Raloxifene: A Selective Estrogen Receptor Modulator for Reducing the Risk of Invasive Breast Cancer in Postmenopausal Women
inferred← citeshttps://doi.org/10.3109/14756366.2011.642374openalex-snapshot
N-Arylbenzamides: extremely simple scaffolds for the development of novel estrogen receptor agonists
inferred← citeshttps://doi.org/10.3390/molecules17067415openalex-snapshot
Application of 4D-QSAR Studies to a Series of Raloxifene Analogs and Design of Potential Selective Estrogen Receptor Modulators
inferred← citeshttps://doi.org/10.4155/fmc.15.181openalex-snapshot
Design and Synthesis of Novel Flexible Ester-Containing Analogs of Tamoxifen and Their Evaluation as Anticancer Agents
inferred← citeshttps://doi.org/10.70675/41b22f7az01dcz48abzaa5ez4d3ae90798c7openalex-snapshot
Comprehensive data analysis and predictive chemoinformatics models for REACH related physicochemical and (eco)toxicity properties
inferred← citeshttps://doi.org/10.7326/0003-4819-130-5-199903020-00015openalex-snapshot
Clinical Effects of Raloxifene Hydrochloride in Women
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