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Inhibition of Cytochrome P450 2D6: Structure−Activity Studies Using a Series of Quinidine and Quinine Analogues

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Outgoing claims: the papers this work cites, builds on, or argues with.

inferredcites →https://doi.org/10.1016/0891-5849(96)83807-xopenalex-snapshot
Cytochrome P450: Structure, mechanism, and biochemistry
inferredcites →https://doi.org/10.1016/s0090-9556(25)07252-6openalex-snapshot
Propranolol hydroxylation and N-desisopropylation by cytochrome P4502D6: studies using the yeast-expressed enzyme and NADPH/O2 and cumene hydroperoxide-supported reactions.
inferredcites →https://doi.org/10.1021/jm00061a004openalex-snapshot
Development of a pharmacophore for inhibition of human liver cytochrome P-450 2D6: molecular modeling and inhibition studies
inferredcites →https://doi.org/10.1021/jo00121a024openalex-snapshot
Steric Effects in SN2 Reactions. Primary Carbon Kinetic Isotope Effects in Menshutkin Reactions
inferredcites →https://doi.org/10.1021/jo9609844openalex-snapshot
SN2 Mechanism for Alcoholysis, Aminolysis, and Hydrolysis of Acetyl Chloride
inferredcites →https://doi.org/10.1021/tx00026a010openalex-snapshot
A predictive model for substrates of cytochrome P450-debrisoquine (2D6)
inferredcites →https://doi.org/10.1042/0264-6021:3450565openalex-snapshot
Evidence that serine 304 is not a key ligand-binding residue in the active site of cytochrome P450 2D6
inferredcites →https://doi.org/10.1042/bj3160647openalex-snapshot
Influence of amino acid residue 374 of cytochrome P-450 2D6 (CYP2D6) on the regio- and enantio-selective metabolism of metoprolol
inferredcites →https://doi.org/10.1042/bj3200531openalex-snapshot
Structure-activity relationships for chemical and glutathione S-transferase-catalysed glutathione conjugation reactions of a series of 2-substituted 1-chloro-4-nitrobenzenes

What points at this work

Incoming claims: where this work appears in other papers’ reference lists and arguments.

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Characterization of Cytochrome P450 Mechanism‐Based Inhibition
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Characterization of Cytochrome P 450 Mechanism‐Based Inhibition
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Stereochemical Elements Associated with Drug Metabolism and Toxicity
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Characterization of Cytochrome P450 Mechanism Based Inhibition
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Diastereoisomer‐Selective Inclusion Complexation of Cinchona Alkaloids with a Modified β‐Cyclodextrin: Fluorescent Behavior Enhanced by Chiral‐Tether Binding. Short Communication
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Ag‐Catalyzed Cyclization‐Intermolecular Sulfinyl Group Transfer Cascade Reactions Enabling Enantioselective Synthesis of 4‐Sulfinylisoquinolines
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Structural evolution of quinine derivatives for enhanced antifungal potency: key modifications and quantitative structure–activity relationship ( QSAR ) analysis
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RETRACTED ARTICLE: Identification of CYP3A4 as the primary cytochrome P450 responsible for the metabolism of tandospirone by human liver microsomes
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Identification of CYP3A4 as the primary cytochrome P450 responsible for the metabolism of tandospirone by human liver microsomes
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Temperature-dependent Time-resolved Fluorescence Study of Cinchonine Alkaloid Dication
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Steady State and Time-Resolved Fluorescence Spectroscopy of Cinchonine Dication in Sodium Dodecylsulphate Micellar System
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Analysis of Species-Selectivity of Human, Mouse and Rat Cytochrome P450 1A and 2B Subfamily Enzymes using Molecular Modeling, Docking and Dynamics Simulations
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Retraction Note to: Identification of CYP3A4 as the primary cytochrome P450 responsible for the metabolism of tandospirone by human liver microsomes
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Insight into the effects of chiral isomers quinidine and quinine on CYP2D6 inhibition
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Cytochrome P450 bio-affinity detection coupled to gradient HPLC: On-line screening of affinities to cytochrome P4501A2 and 2D6
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Human Cytochrome P450 1, 2, 3 Families as Pharmacogenes with Emphases on Their Antimalarial and Antituberculosis Drugs and Prevalent African Alleles
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