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Recent Advances in the Synthesis of Pyrazoles. A Review

https://doi.org/10.1080/00304940903077832

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What this work says

Outgoing claims: the papers this work cites, builds on, or argues with.

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Synthesis of 3-Benzoyl-4-styryl-2-pyrazolines and Their Oxidation to the Corresponding Pyrazoles

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3-Aroyl-5-hydroxyflavones: Synthesis and Transformation into Aroylpyrazoles

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Domino Cu‐Catalyzed CN Coupling/Hydroamidation: A Highly Efficient Synthesis of Nitrogen Heterocycles

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1,3‐Diketones from Acid Chlorides and Ketones: A Rapid and General One‐Pot Synthesis of Pyrazoles.

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Microwave‐Assisted Solution‐Phase Synthesis of 1,4,5‐Trisubstituted Pyrazoles

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Synthesis of Pyrazolyl‐2‐pyrazolines by Treatment of 3‐(3‐Aryl‐3‐oxopropenyl)chromen‐4‐ones with Hydrazine and Their Oxidation to Bis(pyrazoles)

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Synthesis of Pyrazoles by Treatment of 3‐Benzylchromones, 3‐Benzylflavones and Their 4‐Thio Analogues with Hydrazine

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The preparation of N‐carboalkoxypyrazoles and N‐phenylpyrazoles from C(α)‐dianions of carboalkoxyhydrazones and phenylhydrazones

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Synthesis of fluoromethyl, difluoromethyl and trifluoromethyl analogues of pyrazosulfuron‐ethyl as herbicides

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A simple and convenient method for the synthesis of 1‐dialkylaminocarbothioic acid S‐[(2,3‐epithio)propyl] esters

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Solid support synthesis of highly functionalized pyrazoles and isoxazoles; Scaffolds for molecular diversity

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Pyrazoles

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Pyrazoles and their Benzo Derivatives

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In vitro and in vivo profile of 2-(3-di-fluoromethyl-5-phenylpyrazol-1-yl)-5-methanesulfonylpyridine, a potent, selective, and orally active canine COX-2 inhibitor

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Novel potent and selective calcium-release-activated calcium (CRAC) channel inhibitors. Part 1: Synthesis and inhibitory activity of 5-(1-methyl-3-trifluoromethyl-1H-pyrazol-5-yl)-2-thiophenecarboxamides

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Discovery of a potent, selective and orally active canine COX-2 inhibitor, 2-(3-difluoromethyl-5-phenyl-pyrazol-1-yl)-5-methanesulfonyl-pyridine

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Polar substitutions in the benzenesulfonamide ring of celecoxib afford a potent 1,5-diarylpyrazole class of COX-2 inhibitors

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Methanesulfonamide group at position-4 of the C-5-phenyl ring of 1,5-diarylpyrazole affords a potent class of cyclooxygenase-2 (COX-2) inhibitors

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5-Heteroatom substituted pyrazoles as canine COX-2 inhibitors. Part 1: Structure–activity relationship studies of 5-alkylamino pyrazoles and discovery of a potent, selective, and orally active analog

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Synthesis and SAR of heteroaryl-phenyl-substituted pyrazole derivatives as highly selective and potent canine COX-2 inhibitors

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1-[3-Aminobenzisoxazol-5′-yl]-3-trifluoromethyl-6-[2′-(3-(R)-hydroxy-N-pyrrolidinyl)methyl-[1,1′]-biphen-4-yl]-1,4,5,6-tetrahydropyrazolo-[3,4-c]-pyridin-7-one (BMS-740808) a highly potent, selective, efficacious, and orally bioavailable inhibitor of blood coagulation factor Xa

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Synthesis of trifluoromethylated pyrazoles from trifluoromethylenaminones and monosubstituted hydrazines

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Modified reaction conditions to achieve high regioselectivity in the two component synthesis of 1,5-diarylpyrazoles

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Microwave-assisted synthesis utilizing supported reagents: a rapid and versatile synthesis of 1,5-diarylpyrazoles

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One-pot synthesis of pyrazole-5-carboxylates by cyclization of hydrazone 1,4-dianions with diethyl oxalate

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One-pot three-component synthesis of pyrazoles through a tandem coupling-cyclocondensation sequence

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Synthesis of fluorinated pyrazole derivatives from β-alkoxyvinyl trifluoroketones

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Regioselective synthesis of fluorinated pyrazole derivatives from trifluoromethyl-1,3-diketone

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Synthesis of fluorinated heterocycles

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Reaction of hydrazinoquinolines with trifluoromethyl-β-diketones: structural and mechanistic studies

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Haloacetylated enol ethers 10. Condensation of β-alkoxyvinyl trifluoromethyl ketones with thiosemicarbazide. Synthesis of new trifluoromethyl 4,5-dihydro-1H-1-pyrazolethiocarboxyamides

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Formation and dehydration of a series of 5-hydroxy-5-trifluoromethyl-4,5-dihydropyrazoles

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1,4-Dianion of acetophenone n-ethoxycarbonylhydrazone as a synthetic intermediate

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Reaction of α-chloroketones with 1,4-dianion of acetophenone n-ethoxy-carbonylhydrazone

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Difluoromethyl Nitrile Oxide (CF2HCNO): A Neglected Chemical Reagent

inferred← citeshttps://doi.org/10.1002/ejoc.201800286openalex-snapshot

Base‐Promoted Transition‐Metal‐Free Arylation of Imidazo‐Fused Heterocycles with Diaryliodonium Salts

inferred← citeshttps://doi.org/10.1002/ejoc.201900173openalex-snapshot

Gem‐Difluorination of Triazole Alkyl Functionalized Amino Pyrazoles by Selectfluor to Access 4,4‐Difluoro‐pyrazol‐3‐ones/Pyrazol‐3‐imines

inferred← citeshttps://doi.org/10.1002/ejoc.201900494openalex-snapshot

Regioselective Thermal [3+2]‐Dipolar Cycloadditions of α‐Diazoacetates with α‐Sulfenyl/Sulfinyl/Sulfonyl‐β‐Chloroacrylamide Derivatives to Form Densely Functionalised Pyrazoles

inferred← citeshttps://doi.org/10.1002/ejoc.202000467openalex-snapshot

Polyethylene Glycol (PEG‐400) as Methylene Spacer and Green Solvent for the Synthesis of Heterodiarylmethanes under Metal‐Free Conditions

inferred← citeshttps://doi.org/10.1002/ejoc.202000496openalex-snapshot

Iodine‐Catalyzed Ring Opening of 1,1‐Diacylcyclopropanes for Synthesis of Fully Substituted Pyrazole Derivatives

inferred← citeshttps://doi.org/10.1002/hlca.201400032openalex-snapshot

1,3‐Dipolar Cycloadditions of Ethyl 2‐Diazo‐3,3,3‐trifluoropropanoate to Alkynes and [1,5] Sigmatropic Rearrangements of the Resulting 3H‐Pyrazoles: Synthesis of Mono‐, Bis‐ and Tris(trifluoromethyl)‐Substituted Pyrazoles

inferred← citeshttps://doi.org/10.1002/jbt.23704openalex-snapshot

Synthesis, molecular docking analysis, drug‐likeness evaluation, and inhibition potency of new pyrazole‐3,4‐dicarboxamides incorporating sulfonamide moiety as carbonic anhydrase inhibitors

inferred← citeshttps://doi.org/10.1002/jhet.1042openalex-snapshot

A Simple and Efficient Synthesis of Ethyl 1‐Aryl‐4‐formyl‐1H‐pyrazole‐3‐carboxylates

inferred← citeshttps://doi.org/10.1002/jhet.2354openalex-snapshot

One‐Pot Synthesis of Highly Substituted 1H‐Pyrazole‐5‐carboxylates from 4‐Aryl‐2,4‐diketoesters and Arylhydrazines

inferred← citeshttps://doi.org/10.1002/jhet.2710openalex-snapshot

Regioselective Synthesis, Antimicrobial Evaluation and QSAR Studies of Some 3‐Aryl‐1‐heteroarylindeno[1,2‐c]pyrazol‐4(1H)‐ones

inferred← citeshttps://doi.org/10.1002/jhet.3557openalex-snapshot

A Convenient Synthesis of Pyrazole‐imidazoline Derivatives by Microwave Irradiation

inferred← citeshttps://doi.org/10.1002/jhet.3636openalex-snapshot

Et3N‐Prompted Efficient Synthesis of Anthracenyl Pyrazolines and Their Cytotoxicity Evaluation against Cancer Cell Lines

inferred← citeshttps://doi.org/10.1002/jhet.4691openalex-snapshot

Synthesis of anthracene linked polycyclic pyridine derivatives fused with coumarin and pyrazole by one‐pot multicomponent strategy followed by oxidation

inferred← citeshttps://doi.org/10.1002/open.202500024openalex-snapshot

SiO 2 @Benzothiazole‐Cl@Fc as an Efficient Heterogeneous Catalyst for the Synthesis of 1,3,5‐Trisubstituted Pyrazoles by A 3 Coupling

inferred← citeshttps://doi.org/10.1002/slct.201601113openalex-snapshot

Three‐Component Domino HWE Olefination/1,3‐Dipolar Cycloaddition/Oxidation Strategy for the Rapid Synthesis of Trisubstituted Pyrazoles

inferred← citeshttps://doi.org/10.1002/slct.201702384openalex-snapshot

Three‐Component Synthesis of 3,4‐Disubstituted Pyrazoles Using Diazosulfone as a Diazomethane Surrogate

inferred← citeshttps://doi.org/10.1002/slct.202000719openalex-snapshot

Metal‐Free Synthesis of Pyrazoles and Chromenopyrazoles from Hydrazones and Acetylenic Esters

inferred← citeshttps://doi.org/10.1002/slct.202103915openalex-snapshot

Synthesis of Pyrazoles through [3+2] Cyclization of Nitrile Imines with Cinnamaldehydes Followed by Air Oxidation

inferred← citeshttps://doi.org/10.1002/slct.202304010openalex-snapshot

Synthesis, Characterization and Evaluation of Antimicrobial Activity, Phytotoxicity, Molecular Docking & Dynamic Simulations of Benzothiazole Functionalized C−C Linked Pyrazolyl‐Thiazoles

inferred← citeshttps://doi.org/10.1002/tcr.201600141openalex-snapshot

Synthesis of Functionalized Pyrazoles via 1,3‐Dipolar Cycloaddition of α ‐Diazo ‐β ‐ketophosphonates, Sufones and Esters with Electron‐Deficient Alkenes

inferred← citeshttps://doi.org/10.1002/tcr.201600146openalex-snapshot

Synthesis of Imidazo[1,2‐a]pyridines: C‐H Functionalization in the Direction of C‐S Bond Formation

inferred← citeshttps://doi.org/10.1007/128_2012_322openalex-snapshot

Alkene Synthesis Through Transition Metal-Catalyzed Cross-Coupling of N-Tosylhydrazones

inferred← citeshttps://doi.org/10.1007/7081_2012_82openalex-snapshot

Metalation of Pyrazoles and Indazoles

inferred← citeshttps://doi.org/10.1007/978-3-319-04346-3_7openalex-snapshot

Fluorinated Pyrazoles and Indazoles

inferred← citeshttps://doi.org/10.1007/s00044-011-9735-9openalex-snapshot

Antimicrobial, analgesic, DPPH scavenging activities and molecular docking study of some 1,3,5-triaryl-2-pyrazolines

inferred← citeshttps://doi.org/10.1007/s00044-017-2058-8openalex-snapshot

One pot synthesis of thiazolo[2,3-b]dihydropyrimidinone possessing pyrazole moiety and evaluation of their anti-inflammatory and antimicrobial activities

inferred← citeshttps://doi.org/10.1007/s00706-013-0962-2openalex-snapshot

A simple new hydrazine-free synthesis of methyl 1,4,5-trisubstituted 1H-pyrazole-3-carboxylates

inferred← citeshttps://doi.org/10.1007/s00706-014-1293-7openalex-snapshot

Reaction of hydrazones derived from active methylene compounds with Vilsmeier–Haack reagent

inferred← citeshttps://doi.org/10.1007/s00706-014-1371-xopenalex-snapshot

Design, synthesis, and pharmacological evaluation of new pyrazoline derivatives

inferred← citeshttps://doi.org/10.1007/s00706-021-02886-5openalex-snapshot

Structure-based design of novel pyrazolyl–chalcones as anti-cancer and antimicrobial agents: synthesis and in vitro studies

inferred← citeshttps://doi.org/10.1007/s00706-025-03394-6openalex-snapshot

An efficient reaction for the synthesis of functionalized pyrazoles

inferred← citeshttps://doi.org/10.1007/s10562-020-03265-1openalex-snapshot

Copper Iodide Nanoparticles Immobolized Porous Polysulfonamide: An Effective Nanocatalyst for Synthesis of Imidazo [1,2-a] Pyridines

inferred← citeshttps://doi.org/10.1007/s10593-013-1325-yopenalex-snapshot

Synthesis of bis-heterocyclic compounds with a phenylene bridge from 1,4- and 1,3-bis(2-chloro-2-cyanovinyl)benzenes

inferred← citeshttps://doi.org/10.1007/s10593-015-1739-9openalex-snapshot

Synthesis and investigation of isomeric mono- and dinitro derivatives of 3-methyl-4-(pyrazol-3-yl)furazan

inferred← citeshttps://doi.org/10.1007/s10593-015-1760-zopenalex-snapshot

Synthesis of 1-(N-nitropyrazolyl)-1Н-tetrazoles – a new type of heteronuclear N-nitropyrazole derivatives

inferred← citeshttps://doi.org/10.1007/s10593-022-03139-xopenalex-snapshot

A Regioselective Synthesis of 5-chloro-1-vinyl- and 3-alkenyl-5-chloro-1H-pyrazoles

inferred← citeshttps://doi.org/10.1007/s10593-024-03362-8openalex-snapshot

A simple one-pot, two-component synthesis of 1,3,5-trisubstituted pyrazoles using Ce-MMZ catalyst

inferred← citeshttps://doi.org/10.1007/s11030-013-9445-yopenalex-snapshot

Catalyst-free, one-pot, three-component synthesis of 5-amino-1,3-aryl-1 $$H$$ -pyrazole-4-carbonitriles in green media

inferred← citeshttps://doi.org/10.1007/s11030-015-9596-0openalex-snapshot

Transition metal-free one-pot synthesis of nitrogen-containing heterocycles

inferred← citeshttps://doi.org/10.1007/s11030-017-9771-6openalex-snapshot

Synthesis of diverse N-acyl-pyrazoles via cyclocondensation of hydrazides with α-oxeketene dithioacetal

inferred← citeshttps://doi.org/10.1007/s11030-024-10901-0openalex-snapshot

Synthesis, molecular docking and molecular dynamics simulations, drug-likeness studies, ADMET prediction and biological evaluation of novel pyrazole-carboxamides bearing sulfonamide moiety as potent carbonic anhydrase inhibitors

inferred← citeshttps://doi.org/10.1007/s11033-025-11333-1openalex-snapshot

Unlocking the therapeutic potential of N-heterocyclic derivatives as Pim kinase inhibitors

inferred← citeshttps://doi.org/10.1007/s11164-022-04681-1openalex-snapshot

Synthesis, spectroscopic (FT-IR and NMR), DFT and molecular docking studies of ethyl 1-(3-nitrophenyl)-5-phenyl-3-((4-(trifluoromethyl)phenyl)carbamoyl)-1H-pyrazole-4-carboxylate

inferred← citeshttps://doi.org/10.1007/s11224-022-01962-8openalex-snapshot

A theoretical study of the valence tautomerism of 1H-pyrazolium-4-olates (X = O) and related compounds (X = S, Se, NH): relative stabilities, protonation effects, and tautomerization barriers

inferred← citeshttps://doi.org/10.1007/s12039-020-01792-3openalex-snapshot

Design, synthesis and characterization of functionalized pyrazole derivatives bearing amide and sulfonamide moieties from aza-aurones

inferred← citeshttps://doi.org/10.1016/b978-0-12-404598-9.00003-1openalex-snapshot

The Literature of Heterocyclic Chemistry, Part XI, 2008–2009

inferred← citeshttps://doi.org/10.1016/b978-0-12-407777-5.00003-8openalex-snapshot

Recent Advances in the Synthesis of Polysubstituted Heterocycles

inferred← citeshttps://doi.org/10.1016/b978-0-12-812733-9.00016-7openalex-snapshot

Biorelevant fluorine-containing N-heterocycles

inferred← citeshttps://doi.org/10.1016/j.arabjc.2014.12.004openalex-snapshot

Synthesis and evaluation of in vitro bioactivity for polysubstituted N-arylpyrazole derivatives

inferred← citeshttps://doi.org/10.1016/j.biopha.2018.04.061openalex-snapshot

In vitro screening, homology modeling and molecular docking studies of some pyrazole and imidazole derivatives

inferred← citeshttps://doi.org/10.1016/j.carbon.2013.09.008openalex-snapshot

Enhancement in the fluorescence of graphene quantum dots by hydrazine hydrate reduction

inferred← citeshttps://doi.org/10.1016/j.catcom.2013.09.002openalex-snapshot

Iron-catalyzed aerobic oxidative aromatization of 1,3,5-trisubstituted pyrazolines

inferred← citeshttps://doi.org/10.1016/j.catcom.2017.06.051openalex-snapshot

Visible-light-photoredox catalytic C C, C N bond formation: Synthesis of pyrazole derivatives via radical ions

inferred← citeshttps://doi.org/10.1016/j.comptc.2014.01.018openalex-snapshot

The mechanisms of nucleophilic substitution in 1-methyl-3,4,5-trinitropyrazole

inferred← citeshttps://doi.org/10.1016/j.ejmech.2011.09.016openalex-snapshot

Synthesis of functionalized tetrasubstituted pyrazolyl heterocycles – A review

inferred← citeshttps://doi.org/10.1016/j.ejmech.2018.03.037openalex-snapshot

Synthesis and anti-mitotic activity of 2,4- or 2,6-disubstituted- and 2,4,6-trisubstituted-2H-pyrazolo[4,3-c]pyridines

inferred← citeshttps://doi.org/10.1016/j.jfluchem.2012.11.008openalex-snapshot

Synthesis of diversely fluorinated pyrazoles as novel active agrochemical ingredients

inferred← citeshttps://doi.org/10.1016/j.jfluchem.2015.06.003openalex-snapshot

An approach to (4-fluoroalkyl-1-alkyl-1H-pyrazol-3-yl)methylamines

inferred← citeshttps://doi.org/10.1016/j.jfluchem.2018.12.012openalex-snapshot

Synthesis, structure and NMR study of fluorinated isoxazoles derived from hemi-curcuminoids

inferred← citeshttps://doi.org/10.1016/j.jics.2025.101763openalex-snapshot

An overview of pyrazolo[3,4-d]pyrimidine heterocycles: recent synthetic approaches and biological activities

inferred← citeshttps://doi.org/10.1016/j.jorganchem.2026.124114openalex-snapshot

Innovative eco-friendly nanocatalyst: CS-NPs/MWCNT@CuFe2O4@Pd for sustainable A3 coupling in the synthesis of 1,3,5-trisubstituted pyrazoles

inferred← citeshttps://doi.org/10.1016/j.mencom.2014.11.009openalex-snapshot

Synthesis of 1,1,1-trifluorobut-3-yn-2-ones and their reactions with N-nucleophiles

inferred← citeshttps://doi.org/10.1016/j.molliq.2019.111686openalex-snapshot

Small molecule based five-membered heterocycles: A view of liquid crystalline properties beyond the biological applications

inferred← citeshttps://doi.org/10.1016/j.molliq.2021.117136openalex-snapshot

Quantum chemical exploration on the inhibition performance of indole and some of its derivatives against copper corrosion

inferred← citeshttps://doi.org/10.1016/j.molstruc.2019.04.085openalex-snapshot

Synthesis, conformational studies and NBO analysis of (4-chloro-3,5-dimethyl-1H-pyrazol- 1-yl)(p-tolyl)methanone

inferred← citeshttps://doi.org/10.1016/j.molstruc.2019.127633openalex-snapshot

Molecular structure of 1,4-bis(substituted-carbonyl)benzene: A combined experimental and theoretical approach

inferred← citeshttps://doi.org/10.1016/j.molstruc.2020.127692openalex-snapshot

Molecular structure, magnetic properties and catalytic activity in selective ethylene dimerization of nickel (II) complexes with bis(3,5-dimethylpyrazol-1-yl)methane

inferred← citeshttps://doi.org/10.1016/j.molstruc.2022.134790openalex-snapshot

Computational and experimental investigation on biological and photophysical properties of high yielded novel aryl-substituted pyrazolone analogue

inferred← citeshttps://doi.org/10.1016/j.molstruc.2024.137892openalex-snapshot

Carbon quantum dots-based palladium complex: A versatile nano-catalyst for the green synthesis of pyrazoles

inferred← citeshttps://doi.org/10.1016/j.molstruc.2024.139472openalex-snapshot

Synthesis, biological evaluation and molecular docking of novel pyrazole derivatives as multitarget acetylcholinesterase and carbonic anhydrase inhibitors

inferred← citeshttps://doi.org/10.1016/j.molstruc.2024.141002openalex-snapshot

Synthesis, crystal structure and fluorescence properties of some new bis-1H-pyrazoles

inferred← citeshttps://doi.org/10.1016/j.molstruc.2025.143523openalex-snapshot

Pyrazoles a privileged scaffold in drug discovery – Synthetic strategies & exploration of pharmacological potential

inferred← citeshttps://doi.org/10.1016/j.poly.2021.115543openalex-snapshot

Copper complexes from 3,5-disubstituted N-hydroxyethylpyrazole ligands: Cleavage of C N bond as well as formation of second coordination sphere complexes

inferred← citeshttps://doi.org/10.1016/j.tet.2011.04.103openalex-snapshot

A facile approach to polysubstituted pyrazoles from hydrazonyl chlorides and vinyl azides

inferred← citeshttps://doi.org/10.1016/j.tet.2012.11.012openalex-snapshot

‘One-pot’ synthesis of 4-substituted 1,5-diaryl-1H-pyrazole-3-carboxylates via lithium tert-butoxide-mediated sterically hindered Claisen condensation and Knorr reaction

inferred← citeshttps://doi.org/10.1016/j.tet.2012.12.038openalex-snapshot

Efficient one-pot synthesis of substituted pyrazoles

inferred← citeshttps://doi.org/10.1016/j.tet.2013.12.046openalex-snapshot

Cascade regioselective synthesis of pyrazoles from nitroallylic acetates and N-tosyl hydrazine

inferred← citeshttps://doi.org/10.1016/j.tet.2016.11.069openalex-snapshot

Synthesis of dibenzopyranones and pyrazolobenzopyranones through copper(0)/Selectfluor system-catalyzed double CH activation/oxygen insertion of 2-arylbenzaldehydes and 5-arylpyrazole-4-carbaldehydes

inferred← citeshttps://doi.org/10.1016/j.tetlet.2010.07.077openalex-snapshot

One-pot copper-catalyzed synthesis of N-functionalized pyrazoles from boronic acids

inferred← citeshttps://doi.org/10.1016/j.tetlet.2014.02.058openalex-snapshot

N-Alkylhydrazones of aliphatic ketones in the synthesis of 1,3,4-trisubstituted non-symmetric pyrazoles

inferred← citeshttps://doi.org/10.1016/j.tetlet.2014.02.068openalex-snapshot

Synthesis of substituted 2,4,5,6-tetrahydrocyclopenta[c]pyrazoles and 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazoles by intramolecular nitrilimine cycloaddition

inferred← citeshttps://doi.org/10.1016/j.tetlet.2014.09.073openalex-snapshot

Synthesis of dihydropyrazolo[4,3-c]azepines via iodine-mediated intramolecular hydrative cyclization

inferred← citeshttps://doi.org/10.1016/j.tetlet.2018.06.007openalex-snapshot

One-pot synthesis of hydrazine derivatives from aldehydes via radical addition reactions

inferred← citeshttps://doi.org/10.1016/j.tetlet.2018.12.009openalex-snapshot

Visible-light promoted one-pot synthesis of pyrazoles from alkynes and hydrazines

inferred← citeshttps://doi.org/10.1016/j.tetlet.2022.153992openalex-snapshot

Sequential one-pot synthesis and antioxidant evaluation of 5-amino-4-(arylselanyl)-1H-pyrazoles

inferred← citeshttps://doi.org/10.1016/j.tetlet.2023.154752openalex-snapshot

Synthetic diversification of tryptanthrin through its C6-hydrazone

inferred← citeshttps://doi.org/10.1016/j.tgchem.2023.100031openalex-snapshot

Revisiting the role of sulfated oxides for the synthesis of pharmaceutically important heterocycles: Understanding, challenges, and future prospects

inferred← citeshttps://doi.org/10.1021/acs.chemrev.0c01015openalex-snapshot

Fluorinated Pyrazoles: From Synthesis to Applications

inferred← citeshttps://doi.org/10.1021/acs.joc.0c02516openalex-snapshot

α,β-Disubstituted CF3-Enones as a Trifluoromethyl Building Block: Regioselective Preparation of Totally Substituted 3-CF3-Pyrazoles

inferred← citeshttps://doi.org/10.1021/acs.joc.1c00606openalex-snapshot

Direct Preparation of N-Substituted Pyrazoles from Primary Aliphatic or Aromatic Amines

inferred← citeshttps://doi.org/10.1021/acs.joc.2c00727openalex-snapshot

Ring Opening of Pyrrolinium Ions Enabled Regioselective Synthesis of 4-Alkyl N-Arylpyrazoles

inferred← citeshttps://doi.org/10.1021/acs.joc.5c00857openalex-snapshot

Copper-Catalyzed Conjugation between Nitrile Imines and Terminal Alkynes

inferred← citeshttps://doi.org/10.1021/acs.joc.7b00774openalex-snapshot

Selective, Metal-Free Approach to 3- or 5-CF3-Pyrazoles: Solvent Switchable Reaction of CF3-Ynones with Hydrazines

inferred← citeshttps://doi.org/10.1021/acs.joc.8b01228openalex-snapshot

Rh(II)-Catalyzed Ring Expansion of Pyrazoles with Diazocarbonyl Compounds as a Method for the Preparation of 1,2-Dihydropyrimidines

inferred← citeshttps://doi.org/10.1021/acs.joc.9b00819openalex-snapshot

Development of Cyanopyrazoles as Building Blocks to Fungicide Fluxapyroxad and Analogues

inferred← citeshttps://doi.org/10.1021/acs.oprd.0c00300openalex-snapshot

Practical Synthetic Method for Functionalized 1-Methyl-3/5-(trifluoromethyl)-1H-pyrazoles

inferred← citeshttps://doi.org/10.1021/acs.orglett.4c02471openalex-snapshot

Copper-Catalyzed Alkynylation of In Situ-Generated Azoalkenes: An Umpolung Approach to Pyrazoles

inferred← citeshttps://doi.org/10.1021/acs.orglett.5b01127openalex-snapshot

C sp 3 –C sp 3 Bond Cleavage in the Palladium-Catalyzed Aminohydroxylation of Allylic Hydrazones Using Atmospheric Oxygen as the Sole Oxidant

inferred← citeshttps://doi.org/10.1021/acs.orglett.5b01248openalex-snapshot

A Michael Equilibration Model To Control Site Selectivity in the Condensation toward Aminopyrazoles

inferred← citeshttps://doi.org/10.1021/acs.orglett.6b01867openalex-snapshot

Visible-Light Photocatalytic Aerobic Annulation for the Green Synthesis of Pyrazoles

inferred← citeshttps://doi.org/10.1021/acs.orglett.7b03811openalex-snapshot

Synthesis of 5-(Trifluoromethyl)pyrazolines by Formal [4 + 1]-Annulation of Fluorinated Sulfur Ylides and Azoalkenes

inferred← citeshttps://doi.org/10.1021/acs.orglett.8b01854openalex-snapshot

Direct Regioselective [3 + 2] Cycloaddition Reactions of Masked Difluorodiazoethane with Electron-Deficient Alkynes and Alkenes: Synthesis of Difluoromethyl-Substituted Pyrazoles

inferred← citeshttps://doi.org/10.1021/acs.orglett.9b02206openalex-snapshot

One-Pot Highly Regioselective Synthesis of α-Ketoamide N-Arylpyrazoles from Secondary β-Enamino Diketones

inferred← citeshttps://doi.org/10.1021/acscatal.6b02439openalex-snapshot

Copper-Catalyzed Double C–H Alkylation of Aldehyde-Derived N,N-Dialkylhydrazones with Polyhalomethanes: Flexible Access to 4-Functionalized Pyrazoles

inferred← citeshttps://doi.org/10.1021/acscatal.8b03391openalex-snapshot

Catalyst Choice for Highly Enantioselective [3 + 3]-Cycloaddition of Enoldiazocarbonyl Compounds

inferred← citeshttps://doi.org/10.1021/acsomega.6c07653openalex-snapshot

Synthesis, SAR Analysis, and Antifungal Potency against Plant Pathogenic Fungi of New Azidopyrazoles

inferred← citeshttps://doi.org/10.1021/acsomega.8b02304openalex-snapshot

Efficient One-Pot, Two-Component Modular Synthesis of 3,5-Disubstituted Pyrazoles

inferred← citeshttps://doi.org/10.1021/co200147yopenalex-snapshot

Solid Phase Synthesis of 1,5-Diarylpyrazole-4-carboxamides: Discovery of Antagonists of the CB-1 Receptor

inferred← citeshttps://doi.org/10.1021/cr2000459openalex-snapshot

From 2000 to Mid-2010: A Fruitful Decade for the Synthesis of Pyrazoles

inferred← citeshttps://doi.org/10.1021/jacsau.5c00105openalex-snapshot

Bioinspired Synthesis of Bridged Isochromane Fused Pyrazoles by a Silver Catalyzed Cascade Reaction and Its Application for Antibacterial Activity

inferred← citeshttps://doi.org/10.1021/jo2000989openalex-snapshot

Synthesis of 3-Amino-4-fluoropyrazoles

inferred← citeshttps://doi.org/10.1021/jo2009824openalex-snapshot

Microwave-Assisted and Continuous Flow Multistep Synthesis of 4-(Pyrazol-1-yl)carboxanilides

inferred← citeshttps://doi.org/10.1021/jo201119eopenalex-snapshot

Synthesis of Pyrazoles via Electrophilic Cyclization

inferred← citeshttps://doi.org/10.1021/jo201685popenalex-snapshot

Synthesis of Pyrazoles via CuI-Mediated Electrophilic Cyclizations of α,β-Alkynic Hydrazones

inferred← citeshttps://doi.org/10.1021/ol101087jopenalex-snapshot

A Modular Sydnone Cycloaddition/Suzuki−Miyaura Cross-Coupling Strategy to Unsymmetrical 3,5-Bis(hetero)aromatic Pyrazoles

inferred← citeshttps://doi.org/10.1021/ol1019713openalex-snapshot

New Synthesis of Fluorinated Pyrazoles

inferred← citeshttps://doi.org/10.1021/ol201555zopenalex-snapshot

A Novel Synthesis of Fluorinated Pyrazoles via Gold(I)-Catalyzed Tandem Aminofluorination of Alkynes in the Presence of Selectfluor

inferred← citeshttps://doi.org/10.1021/ol2031608openalex-snapshot

Terminal Alkyne Addition to Diazodicarboxylates: Synthesis of Hydrazide Linked Alkynes (Ynehydrazides)

inferred← citeshttps://doi.org/10.1021/ol301655fopenalex-snapshot

Novel Synthesis of 5-Amino-3-bromo-1-(tert-butyl)-1H-pyrazole-4-carbonitrile: A Versatile Intermediate for the Preparation of 5-Amino-3-aryl-1-(tert-butyl)-1H-pyrazole-4-carboxamides

inferred← citeshttps://doi.org/10.1021/ol403447gopenalex-snapshot

Regioselective Synthesis of 1,3,5-Trisubstituted Pyrazoles from N -Alkylated Tosylhydrazones and Terminal Alkynes

inferred← citeshttps://doi.org/10.1021/ol501312sopenalex-snapshot

Dual Roles of Sulfonyl Hydrazides: A Three-Component Reaction To Construct Fully Substituted Pyrazoles Using TBAI/TBHP

inferred← citeshttps://doi.org/10.1021/op500114vopenalex-snapshot

Synthesis of Fluorinated and Nonfluorinated Tebufenpyrad Analogues for the Study of Anti-angiogenesis MOA

inferred← citeshttps://doi.org/10.1039/c1cc15809kopenalex-snapshot

Single-step synthesis of pyrazoles using titanium catalysis

inferred← citeshttps://doi.org/10.1039/c2ra20274copenalex-snapshot

Synthesis of 3,5-disubstituted pyrazoles via cyclocondensation of 1,2-allenic ketones with hydrazines: application to the synthesis of 5-(5-methyl-pyrazol-3-yl)-2′-deoxycytidine

inferred← citeshttps://doi.org/10.1039/c3ob41435copenalex-snapshot

DABCO-promoted synthesis of pyrazoles from tosylhydrazones and nitroalkenes

inferred← citeshttps://doi.org/10.1039/c3ob42102copenalex-snapshot

Effect of configuration of 2-vinyldiazocarbonyl compounds on their reactivity: experimental and computational study

inferred← citeshttps://doi.org/10.1039/c3ra41569dopenalex-snapshot

Molecular iodine catalyzed one-pot multicomponent reactions for the synthesis of dihydrochromeno[4,3-b]pyrazolo[4,3-e]pyridin-6(7H)-ones

inferred← citeshttps://doi.org/10.1039/c4cc02856bopenalex-snapshot

Copper-mediated pyrazole synthesis from 2,3-allenoates or 2-alkynoates, amines and nitriles

inferred← citeshttps://doi.org/10.1039/c4ob02556copenalex-snapshot

Ylide formal [4 + 1] annulation

inferred← citeshttps://doi.org/10.1039/c4ob02670eopenalex-snapshot

Three-component synthesis of fluorinated pyrazoles from fluoroalkylamines, NaNO 2 and electron-deficient alkynes

inferred← citeshttps://doi.org/10.1039/c4ra16439copenalex-snapshot

Metal-free synthesis of 3,5-disubstituted 1H- and 1-aryl-1H-pyrazoles from 1,3-diyne-indole derivatives employing two successive hydroaminations

inferred← citeshttps://doi.org/10.1039/c5cs00805kopenalex-snapshot

Multicomponent syntheses of functional chromophores

inferred← citeshttps://doi.org/10.1039/c5py01218jopenalex-snapshot

Tetraaryl pyrazole polymers: versatile synthesis, aggregation induced emission enhancement and detection of explosives

inferred← citeshttps://doi.org/10.1039/c6cc06935eopenalex-snapshot

Solvent-dependent copper-catalyzed synthesis of pyrazoles under aerobic conditions

inferred← citeshttps://doi.org/10.1039/c6ob01522kopenalex-snapshot

[3 + 2] cycloaddition and subsequent oxidative dehydrogenation between alkenes and diazo compounds: a simple and direct approach to pyrazoles using TBAI/TBHP

inferred← citeshttps://doi.org/10.1039/c6pp00009fopenalex-snapshot

Synthesis, regioselective aerobic Pd(ii)-catalyzed C–H bond alkenylation and the photophysical properties of pyrenylphenylpyrazoles

inferred← citeshttps://doi.org/10.1039/c8ob02352bopenalex-snapshot

Regioselective [3 + 2]-annulation of hydrazonyl chlorides with 1,3-dicarbonyl compounds for assembling of polysubstituted pyrazoles

inferred← citeshttps://doi.org/10.1039/c9cc03363gopenalex-snapshot

Retracted Article: Molybdenum-silver co-catalyzed cycloaddition of alkynes with N -isocyanoiminotriphenylphosphorane (NIITP): an efficient strategy for the synthesis of monosubstituted pyrazoles

inferred← citeshttps://doi.org/10.1039/c9ra09013dopenalex-snapshot

Sulphated alumina tungstic acid (SATA): a highly efficient and novel heterogeneous mesostructured catalyst for the synthesis of pyrazole carbonitrile derivatives and evaluation of green metrics

inferred← citeshttps://doi.org/10.1039/c9tc04309hopenalex-snapshot

B–N coordinated triaryl pyrazole: effect of dimerization, and optical and NLO properties

inferred← citeshttps://doi.org/10.1039/d0nj02215bopenalex-snapshot

Synthesis of 3-oxadiazole-substituted imidazo[1,2- a ]pyridines by nickel immobilized on multifunctional amphiphilic porous polysulfonamide–melamine

inferred← citeshttps://doi.org/10.1039/d0ob01228aopenalex-snapshot

Pyrazoles: ‘one-pot’ synthesis from arenes and carboxylic acids

inferred← citeshttps://doi.org/10.1039/d0ra09778kopenalex-snapshot

Monoallylation and benzylation of dicarbonyl compounds with alcohols catalysed by a cationic cobalt( iii ) compound

inferred← citeshttps://doi.org/10.1039/d2qo01196dopenalex-snapshot

Sustainable synthesis of pyrazoles using alcohols as the primary feedstock by an iron catalyzed tandem C–C and C–N coupling approach

inferred← citeshttps://doi.org/10.1039/d3gc02118aopenalex-snapshot

From screening to the hectogram scale: sustainable electrochemical synthesis of mefenpyr-diethyl

inferred← citeshttps://doi.org/10.1039/d3nj03326kopenalex-snapshot

NIS-mediated regioselective addition of allenamides with pyrazoles: synthesis of iodo-substituted allylic pyrazoles

inferred← citeshttps://doi.org/10.1039/d3ob00671aopenalex-snapshot

Electrochemically enabled oxidative aromatization of pyrazolines

inferred← citeshttps://doi.org/10.1039/d3ob01997gopenalex-snapshot

Iodine/DMSO-mediated one-pot access towards 1-aryl-2-(pyrazol-5-yl)ethane-1,2-diones via a domino reaction from functionalized pent-2-ene-1,5-diones

inferred← citeshttps://doi.org/10.1039/d5ra07282dopenalex-snapshot

Sustainable multicomponent synthesis of C-4 sulfenylated pyrazoles via sodium thiosulfate-promoted tandem cyclocondensation and C–H sulfenylation

inferred← citeshttps://doi.org/10.1055/s-0041-1737395openalex-snapshot

Facile One-Pot Preparation of 5-Substituted 4-Iodo-1-tosylpyrazoles from N-Propargyl-N′-tosylhydrazines through Iodocyclization

inferred← citeshttps://doi.org/10.1080/00304948.2020.1792228openalex-snapshot

Convenient OPC-VH Mediated Synthesis of 4-Functional Pyrazoles

inferred← citeshttps://doi.org/10.1080/00304948.2021.1904750openalex-snapshot

Green Methods for the Synthesis of Pyrazoles: A Review

inferred← citeshttps://doi.org/10.1080/00397911.2013.828757openalex-snapshot

Synthesis of Pyrazole Derivatives Possessing Anticancer Activity: Current Status

inferred← citeshttps://doi.org/10.1080/02678292.2018.1446553openalex-snapshot

Synthesis and mesomorphism behaviour of chalcones and pyrazoles type compounds as photo-luminescent materials

inferred← citeshttps://doi.org/10.1080/10426507.2022.2046575openalex-snapshot

Convenient methods for the synthesis organotellurium compounds derived from pyrazole derivatives: synthesis and antimicrobial evaluation

inferred← citeshttps://doi.org/10.1107/s1600536810026036openalex-snapshot

3,5-Bis(4-fluorophenyl)-1-phenyl-4,5-dihydro-1H-pyrazole

inferred← citeshttps://doi.org/10.1107/s2056989018011477openalex-snapshot

N-(6-Methoxypyridin-2-yl)-1-(pyridin-2-ylmethyl)-1H-pyrazole-3-carboxamide: crystal structure and Hirshfeld surface analysis

inferred← citeshttps://doi.org/10.1107/s205698902401140xopenalex-snapshot

Synthesis, crystal structure and Hirshfeld surface analysis of 5-methyl-1 H -pyrazol-3-yl 4-nitrobenzenesulfonate at 90 K

inferred← citeshttps://doi.org/10.1111/cbdd.12496openalex-snapshot

Identification of Novel Proteasome Inhibitors from an Enaminone Library

inferred← citeshttps://doi.org/10.1134/s1063774518060160openalex-snapshot

Synthesis and Single Crystal X-Ray Structure of 3,5-Diphenyl-1-(phenylacetyl)-4,5-dihydro-1H-pyrazol

inferred← citeshttps://doi.org/10.1134/s1068162023040167openalex-snapshot

Synthesis, Antioxidant, Antifungal and Antibacterial Activities of New Class of Fused Isoxazole-Pyrimidines and Pyrazole-Pyrimidines as Five and Six Membered Heterocyclic Compounds

inferred← citeshttps://doi.org/10.1134/s1070363217090304openalex-snapshot

Features of the reaction of some symmetrically substituted isoindigos with hydrazine hydrate

inferred← citeshttps://doi.org/10.1134/s1070428023060052openalex-snapshot

Synthesis of 5-Chloro-3-styryl-1H-pyrazoles Based on 2,2-Dichlorovinyl Ketones

inferred← citeshttps://doi.org/10.1246/cl.200081openalex-snapshot

Structures and Photoluminescence of Coinage Metal(I) Phenylpyrazolato Trinuclear Complexes [M(3,5-Et2-4-Ph-pz)]3 and Arene Sandwich Complexes {[Ag(3,5-Et2-4-Ph-pz)]3}2(Ar) (Ar = Mesitylene and Toluene)

inferred← citeshttps://doi.org/10.1248/cpb.c12-00725openalex-snapshot

Divergent Synthesis and Evaluation of Inhibitory Activities against Cyclooxygenases-1 and -2 of Natural Withasomnines and Analogues

inferred← citeshttps://doi.org/10.1371/journal.pone.0308036openalex-snapshot

Laccase-mediated chemoselective C-4 arylation of 5-aminopyrazoles

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