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Growing PAINS in Academic Drug Discovery
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What this work says
Outgoing claims: the papers this work cites, builds on, or argues with.
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Promiscuous Aggregate-Based Inhibitors Promote Enzyme Unfolding
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New Substructure Filters for Removal of Pan Assay Interference Compounds (PAINS) from Screening Libraries and for Their Exclusion in Bioassays
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Drug-Like Property Concepts in Pharmaceutical Design
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Observations on Screening-Based Research and Some Concerning Trends in the Literature
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