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Crystal structure, absolute configuration, and phosphodiesterase inhibitory activity of (+)-1-(4-bromobenzyl)-4-[(3-cyclopentyloxy)-4-methoxyphenyl]-2-pyrrolidinone

https://doi.org/10.1021/jm00074a007
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Visible‐Light‐Driven C−H Oxidation of Cyclic Tertiary Amines: Access to Synthetic Strychnos Alkaloids with Antiviral Activity
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Enaminones 9. Further studies on the anticonvulsant activity and potential type IV phosphodiesterase inhibitory activity of substituted vinylic benzamides
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Cesium salts as superior catalysts for solvent-free modifications of biosourced pterolactam
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Selective syntheses of benzoxazoles and N-(2-hydroxyaryl)pyrrolidin-2-ones from the corresponding cyclopropyl amides with PPh3/CX4
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One-pot and regioselective synthesis of functionalized γ-lactams via a metal-free sequential Ugi 4CR/Intramolecular 5-exo-dig cyclization reaction
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Conjugated addition of bis(oxazolinyl)zinc to substituted 2-nitrovinyl benzenes: an alternative synthesis of (±)-Rolipram
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Rhodium-catalyzed asymmetric addition of arylboronic acids to γ-phthalimido-substituted-α,β-unsaturated carboxylic acid esters: an approach to γ-amino acids
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Chapter 8. Emerging Opportunities in the Treatment of Asthma and Allergy
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Chapter 19. Isozyme-Selective Phosphodiesterase Inhibitors as Antiasthmatic Agents
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1 Phosphodiesterase Type IV Inhibitors
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Structure-activity relationships involving the catechol subunit of rolipram
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Deacetylative Amination of Acetyl Arenes and Alkanes with C–C Bond Cleavage
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Multicomponent Approach to a Library of N-Substituted γ-Lactams
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Development of a Catalytic Enantioselective Conjugate Addition of 1,3-Dicarbonyl Compounds to Nitroalkenes for the Synthesis of Endothelin-A Antagonist ABT-546. Scope, Mechanism, and Further Application to the Synthesis of the Antidepressant Rolipram
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Direct β-selectivity of α,β-unsaturated γ-butyrolactam for asymmetric conjugate additions in an organocatalytic manner
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Iodine( iii ) promoted ring-rearrangement reaction of 1-arylamino-2-oxocyclopentane-1-carbonitriles to synthesize N -aryl-δ-valerolactams
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Visible light-driven photocatalytic sulfonative oxidation of benzyl secondary amines
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Enantiomeric HPLC Separations of 4-Substituted-Pyrrolidin-2-Ones using Cellulose Based Chiral Stationary Phases
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Part II: From Dermatologicals to Sensory Organ and Various Drugs
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Inhibitor Binding to Type 4 Phosphodiesterase (PDE4) Assessed Using [3H]Piclamilast and [3H]Rolipram
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Synthesis and Antibacterial Activity of 5-Aryl-4-[hydroxy(4-chlorophenyl)methylene]-1-[2-(1H-indol-3-yl)ethyl]pyrrolidine-2,3-diones
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Synthesis of Pyrrolidine-2,3-dione Derivatives by Reacting Methyl 4-(4-Fluorophenyl)-2,4-dioxobutanoate with Tryptamine and Aromatic Aldehydes
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Effects of dialkoxylphenyl compounds with oxime group on macrophage function and the proliferation of lymphocytes
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Synthesis and Structure-Activity Relationship of N-Arylrolipram Derivatives as Inhibitors of PDE4 Isozymes.
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Overview: Cardiovascular & Renal; Cyclic nucleotide phosphodiesterase inhibitors
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Spiro-Lactams as Novel Antimicrobial Agents
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Synthesis of 5-Aryl-1-[2-(1H-indol-3-yl)ethyl]- 4-(hydroxy-4-methylphenylmethylene)pyrrolidine-2,3-diones by Reaction of Tryptamine with 4-Methylbenzoyltartaric Acid Methyl Ester and Aromatic Aldehydes
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Enantiodivergent Synthesis of (R)- and (S)-Rolipram
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Efficient Synthesis of β-Aryl-γ-lactams and Their Resolution with (S)-Naproxen: Preparation of (R)- and (S)-Baclofen
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Novel Isoxazolidine and γ-Lactam Analogues of Homonucleosides
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Asymmetric Michael Addition in Synthesis of β-Substituted GABA Derivatives
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An Efficient Synthesis of Enantiomerically Pure γ-Aminobutyric Acid (GABA) Derivatives
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An efficient method for the synthesis of substituted N-aryl lactams
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