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Identification of Novel Breast Cancer Resistance Protein (BCRP) Inhibitors by Virtual Screening
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What this work says
Outgoing claims: the papers this work cites, builds on, or argues with.
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Structure activity relationships and quantitative structure activity relationships for the flavonoid-mediated inhibition of breast cancer resistance protein
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Structure–activity relationships of new inhibitors of breast cancer resistance protein (ABCG2)
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Structure–activity relationships of flavonoids as inhibitors of breast cancer resistance protein (BCRP)
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Novel web-based tools combining chemistry informatics, biology and social networks for drug discovery
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Breast cancer resistance protein (BCRP/ABCG2): New inhibitors and QSAR studies by a 3D linear solvation energy approach
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Identification and functional characterization of breast cancer resistance protein in human bronchial epithelial cells (Calu-3)
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Breast Cancer Resistance Protein: Mediating the Trans-placental Transfer of Glyburide across the Human Placenta
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Inhibition of volume-activated I- and taurine efflux from HeLa cells by P-glycoprotein blockers correlates with calmodulin inhibition.
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Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings 1PII of original article: S0169-409X(96)00423-1. The article was originally published in Advanced Drug Delivery Reviews 23 (1997) 3–25. 1
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Computational Models for Drug Inhibition of the Human Apical Sodium-Dependent Bile Acid Transporter
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Machine Learning Methods and Docking for Predicting Human Pregnane X Receptor Activation
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Uptake and Efflux of Quinacrine, a Candidate for the Treatment of Prion Diseases, at the Blood-Brain Barrier
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The sulphonylurea glibenclamide inhibits multidrug resistance protein (MRP1) activity in human lung cancer cells
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A multidrug resistance transporter from human MCF-7 breast cancer cells
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Receiver-operating characteristic (ROC) plots: a fundamental evaluation tool in clinical medicine
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Modulation of human BCRP (ABCG2) activity by anti-HIV drugs
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Pharmacokinetic Interaction of Fluvoxamine and Thioridazine in Schizophrenic Patients
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ABCB1 and Cytochrome P450 Polymorphisms
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Antipsychotic Drugs Inhibit the Function of Breast Cancer Resistance Protein
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Rapid Identification of P-glycoprotein Substrates and Inhibitors
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Breast Cancer Resistance Protein Interacts with Various Compounds in Vitro, but Plays a Minor Role in Substrate Efflux at the Blood-Brain Barrier
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Identification and Validation of Novel Human Pregnane X Receptor Activators among Prescribed Drugs via Ligand-Based Virtual Screening
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Human Breast Cancer Resistance Protein: Interactions with Steroid Drugs, Hormones, the Dietary Carcinogen 2-Amino-1-methyl-6-phenylimidazo(4,5-b)pyridine, and Transport of Cimetidine
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A Global Drug Inhibition Pattern for the Human ATP-Binding Cassette Transporter Breast Cancer Resistance Protein (ABCG2)
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Quantitative Evaluation of the Impact of Active Efflux by P-Glycoprotein and Breast Cancer Resistance Protein at the Blood-Brain Barrier on the Predictability of the Unbound Concentrations of Drugs in the Brain Using Cerebrospinal Fluid Concentration as a Surrogate
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In Silico Prediction of Pregnane X Receptor Activators by Machine Learning Approache
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Using Extended-Connectivity Fingerprints with Laplacian-Modified Bayesian Analysis in High-Throughput Screening Follow-Up
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Increased Oral Bioavailability of Topotecan in Combination With the Breast Cancer Resistance Protein and P-Glycoprotein Inhibitor GF120918
inferredcites →https://doi.org/10.1208/aapsj070112openalex-snapshot
Role of the breast cancer resistance protein (ABCG2) in drug transport
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Drugs Behave as Substrates, Inhibitors and Inducers of Human Cytochrome P450 3A4
inferredcites →https://doi.org/10.3892/mmr.2011.734openalex-snapshot
Differential effects of calcium antagonists on ABCG2/BCRP-mediated drug resistance and transport in SN-38-resistant HeLa cells
inferredcites →https://doi.org/10.7270/q2j104fdopenalex-snapshot
BindingDB Entry 50041981: Reversal of breast cancer resistance protein-mediated drug resistance by estrogen antagonists and agonists.
What points at this work
Incoming claims: where this work appears in other papers’ reference lists and arguments.
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Inhibitory Effects of Alkaloids on BCRP Implicated in Reversing Multidrug Resistance: A Case Example of Enhancing Temozolomide Cytotoxicity
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Topología molecular aplicada al reconocimiento de sustratos de la Proteína de Resistencia del Cáncer de Mama (BCRP)
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