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Synthesis of the NK1 Receptor Antagonist GW597599. Part 3: Development of a Scalable Route to a Key Chirally Pure Arylpiperazine Urea, A Happy End
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Outgoing claims: the papers this work cites, builds on, or argues with.
inferredcites →https://doi.org/10.1002/ejoc.200700325openalex-snapshot
Synthesis of 3‐Phenyl‐4‐piperidones from Acetophenone by Shapiro and Aza‐Michael Reactions and Their Further Derivatization
inferredcites →https://doi.org/10.1016/s0040-4039(00)75977-6openalex-snapshot
Conversion of amines to carbamoyl chlorides using carbon dioxide as a phosgene replacement
inferredcites →https://doi.org/10.1021/ja01475a023openalex-snapshot
Synthesis of a Heptapeptide Sequence Derived from Bovine Insulin1
inferredcites →https://doi.org/10.1021/ja073219nopenalex-snapshot
Molecular Wire Behavior in π-Stacked Donor-Bridge-Acceptor Tertiary Arylureas
inferredcites →https://doi.org/10.1021/jm900023bopenalex-snapshot
Discovery Process and Pharmacological Characterization of 2-(S)-(4-Fluoro-2-methylphenyl)piperazine-1-carboxylic Acid [1-(R)-(3,5-Bis-trifluoromethylphenyl)ethyl]methylamide (Vestipitant) as a Potent, Selective, and Orally Active NK1 Receptor Antagonist
inferredcites →https://doi.org/10.1021/jm960070+openalex-snapshot
3-Phenyl-Substituted Imidazo[1,5-a]quinoxalin-4-ones and Imidazo[1,5-a]quinoxaline Ureas That Have High Affinity at the GABAA/Benzodiazepine Receptor Complex
inferredcites →https://doi.org/10.1021/jm9602571openalex-snapshot
Cyclic HIV Protease Inhibitors: Synthesis, Conformational Analysis, P2/P2‘ Structure−Activity Relationship, and Molecular Recognition of Cyclic Ureas
inferredcites →https://doi.org/10.1021/op800146dopenalex-snapshot
Synthesis of the NK1 Receptor Antagonist GW597599. Part 1: Development of a Scalable Route to a Key Chirally Pure Arylpiperazine
inferredcites →https://doi.org/10.1021/op8002823openalex-snapshot
Synthesis of the NK1 Receptor Antagonist GW597599. Part 2: Development of a Scalable Route to a Key Chirally Pure Arylpiperazine
inferredcites →https://doi.org/10.1055/s-1984-31064openalex-snapshot
Monoprotection of α,ω-Alkanediamines with theN-Benzyloxycarbonyl Group
inferredcites →https://doi.org/10.1055/s-1989-27272openalex-snapshot
A New Convenient Method for the Synthesis of Symmetrical and UnsymmetricalN,N′-Disubstituted Ureas
inferredcites →https://doi.org/10.1111/j.1399-3011.1986.tb01061.xopenalex-snapshot
Use of 10% sulfuric acid/dioxane for removal of N‐α‐tertiary‐butyloxycarbonyl group during solid phase peptide synthesis
What points at this work
Incoming claims: where this work appears in other papers’ reference lists and arguments.
inferred← citeshttps://doi.org/10.2139/ssrn.4765835openalex-extracted
Polyfunctionalized Organoselenides: New Synthetic Approach from Seleno-Containing Cyanohydrins and Anti-Melanoma Activity
inferred← citeshttps://doi.org/10.1002/chem.202500299openalex-snapshot
Efficient and Selective Transformations of α‐Keto Esters into α‐Arylated α‐Hydroxy Esters Using Continuous‐Flow System
inferred← citeshttps://doi.org/10.1002/mrc.2611openalex-snapshot
Application of LC–NMR to the identification of bulk drug impurities in NK1 antagonist GW597599 (vestipitant)
inferred← citeshttps://doi.org/10.1016/j.bmcl.2024.129860openalex-snapshot
Polyfunctionalized organoselenides: New synthetic approach from selenium-containing cyanohydrins and anti-melanoma activity
inferred← citeshttps://doi.org/10.1016/j.tetlet.2010.05.019openalex-snapshot
Dynamic thermodynamic resolution of lithiated N-Boc-N′-alkylpiperazines
inferred← citeshttps://doi.org/10.1021/acs.oprd.5b00283openalex-snapshot
Optimization of the Preparation of (R)-3,5-Bis(trifluoromethyl)-α-methyl-N-methylbenzylamine l -(−)-Malic Acid Salt through Classical Resolution
inferred← citeshttps://doi.org/10.1021/acs.orglett.6b01190openalex-snapshot
Synthesis of Chiral Piperazines via Hydrogenation of Pyrazines Activated by Alkyl Halides
inferred← citeshttps://doi.org/10.1021/jacs.5b11288openalex-snapshot
Synthesis of Enantiopure Piperazines via Asymmetric Lithiation–Trapping of N-Boc Piperazines: Unexpected Role of the Electrophile and Distal N-Substituent
inferred← citeshttps://doi.org/10.1021/op1000622openalex-snapshot
Application of the QbD Principles in the Development of the Casopitant Mesylate Manufacturing Process. Process Research Studies for the Definition of the Control Strategy of some Drug Substance-CQAs for Stages 2a, 2b, and 2c
inferred← citeshttps://doi.org/10.1021/op1000836openalex-snapshot
Development of a Control Strategy for a Defluorinated Analogue in the Manufacturing Process of Casopitant Mesylate
inferred← citeshttps://doi.org/10.1021/op500169mopenalex-snapshot
Design of Experiments (DoE) and Process Optimization. A Review of Recent Publications
inferred← citeshttps://doi.org/10.1039/c2ob25412copenalex-snapshot
Unsymmetrical tetrasubstituted ureas from tertiary carbamoylimidazole: activation by AlMe3
inferred← citeshttps://doi.org/10.1039/c3cc40392kopenalex-snapshot
Reactions of organolithiums with dialkyl oxalates. A flow microreactor approach to synthesis of functionalized α-keto esters
inferred← citeshttps://doi.org/10.2174/0115680266294434240322043536openalex-snapshot
Green Synthesis of Biorelevant Scaffolds through Organocatalytic/ Enzymatic Dynamic Kinetic Resolution
inferred← citeshttps://doi.org/10.3184/174751916x14546711471143openalex-snapshot
A Scalable and Facile Process for the Preparation of N -(Pyridin-4-yl) Piperazine-1-Carboxamide Hydrochloride
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