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Synthesis of 3-trifluoromethylpyrazoles via trifluoromethylation/cyclization of α,β-alkynic hydrazones using a hypervalent iodine reagent
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What this work says
Outgoing claims: the papers this work cites, builds on, or argues with.
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Modern Synthetic Methods for Fluorine‐Substituted Target Molecules
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CF 3 ‐Bearing Aromatic and Heterocyclic Building Blocks
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Zinc‐Mediated Formation of Trifluoromethyl Ethers from Alcohols and Hypervalent Iodine Trifluoromethylation Reagents
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A Ritter‐Type Reaction: Direct Electrophilic Trifluoromethylation at Nitrogen Atoms Using Hypervalent Iodine Reagents
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Copper‐Catalyzed Trifluoromethylation of Unactivated Olefins
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Tamed Arene and Heteroarene Trifluoromethylation
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Direct Electrophilic N‐Trifluoromethylation of Azoles by a Hypervalent Iodine Reagent
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A “Renaissance” in Radical Trifluoromethylation
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Introduction of Fluorine and Fluorine‐Containing Functional Groups
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Silver‐Mediated Cycloaddition of Alkynes with CF3CHN2: Highly Regioselective Synthesis of 3‐Trifluoromethylpyrazoles
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Recent Developments on the Trifluoromethylation of (Hetero)Arenes
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The New Age of Electrophilic Perfluoroalkylation Reactions
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Strategies for nucleophilic, electrophilic, and radical trifluoromethylations
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Reaction of 2-hydroxyethylhydrazine with a trifluoromethyl-β-diketone: Study and structural characterization of a new 5-hydroxy-5-trifluoromethyl-4,5-dihydropyrazole intermediate
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Synthesis of bromodifluoromethyl substituted pyrazoles and isoxazoles
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Preparation of trifluoromethyl-pyrazoles and -pyrazolines by the reaction of 2,2,2-trifluorodiazoethane with carbon-carbon multiple bonds
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Aromatic Trifluoromethylation with Metal Complexes
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From 2000 to Mid-2010: A Fruitful Decade for the Synthesis of Pyrazoles
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Update 1 of: Asymmetric Fluorination, Trifluoromethylation, and Perfluoroalkylation Reactions
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Perfluoroalkylation with Organosilicon Reagents
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Copper-Catalyzed C(sp3)–C(sp3) Bond Formation Using a Hypervalent Iodine Reagent: An Efficient Allylic Trifluoromethylation
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Synthesis and Biological Activities of Novel Pyrazole Oxime Derivatives Containing a 2-Chloro-5-thiazolyl Moiety
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Synthesis and Biological Evaluation of the 1,5-Diarylpyrazole Class of Cyclooxygenase-2 Inhibitors: Identification of 4-[5-(4-Methylphenyl)-3- (trifluoromethyl)-1 H -pyrazol-1-yl]benzenesulfonamide (SC-58635, Celecoxib)
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Electrophilic Trifluoromethylation of S-Hydrogen Phosphorothioates
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Synthesis of Pyrazoles via Electrophilic Cyclization
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Improved Regioselectivity in Pyrazole Formation through the Use of Fluorinated Alcohols as Solvents: Synthesis and Biological Activity of Fluorinated Tebufenpyrad Analogs
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A Novel Synthesis of Fluorinated Pyrazoles via Gold(I)-Catalyzed Tandem Aminofluorination of Alkynes in the Presence of Selectfluor
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The pharmacokinetics of mavacoxib, a long‐acting COX‐2 inhibitor, in young adult laboratory dogs
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Fluorine in Pharmaceuticals: Looking Beyond Intuition
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Shelf-stable electrophilic trifluoromethylating reagents: A brief historical perspective
What points at this work
Incoming claims: where this work appears in other papers’ reference lists and arguments.
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Preparation of New Spiropyrazole, Pyrazole and Hydantoin Derivatives and Investigation of Their Antioxidant and Antibacterial Activities.
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Recent Advances in Trifluoromethylation Reactions with Electrophilic Trifluoromethylating Reagents
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ChemInform Abstract: Synthesis of 3‐Trifluoromethylpyrazoles via Trifluoromethylation/Cyclization of α,β‐Alkynic Hydrazones Using a Hypervalent Iodine Reagent.
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Study on the Degradation of the Highly Reactive Hypervalent Trifluoromethylation Iodine Reagent PhI(OAc)(CF3)
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Et3N‐Prompted Efficient Synthesis of Anthracenyl Pyrazolines and Their Cytotoxicity Evaluation against Cancer Cell Lines
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Assembly of nitrogen-containing heterocycles initiated by the aza-Michael reaction
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Kinetics of the heterocyclization of (E)-1,5-diphenylpent-1-en-4-yn-3-one phenylhydrazone in the presence of 1,8-diazabicyclo[5.4.0]undec-7-ene
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Five-Membered Ring Systems
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Five-Membered Ring Systems
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Development of Electrophilic Trifluoromethylating Reagents
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Silver-catalyzed synthesis of 5-aryl-3-trifluoromethyl pyrazoles
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Advances in Synthetic Applications of Hypervalent Iodine Compounds
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Conjugated Ynones in Organic Synthesis
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Regioselective Synthesis of 5-Trifluoromethylpyrazoles by [3 + 2] Cycloaddition of Nitrile Imines and 2-Bromo-3,3,3-trifluoropropene
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Selective, Metal-Free Approach to 3- or 5-CF3-Pyrazoles: Solvent Switchable Reaction of CF3-Ynones with Hydrazines
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Synthesis of 3-Trifluoromethylpyrazole Derivatives
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