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Construction of the CSIRO Fragment Library

https://doi.org/10.1071/ch13325
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What this work says

Outgoing claims: the papers this work cites, builds on, or argues with.

inferredcites →https://doi.org/10.1002/cber.19731060109openalex-snapshot
Reaktionen mit Dialkylcyanamiden. Umsetzung von Dialkylcyanamiden mit Schwefel‐ bzw. Phosphorhalogeniden; Synthese von substituierten Chlorformamidinen
inferredcites →https://doi.org/10.1002/prac.19883300609openalex-snapshot
Synthese und Strukturermittlung von Sulfamoyl‐guanidinen
inferredcites →https://doi.org/10.1007/bf00811103openalex-snapshot
�ber die Synthese von Dihydro-1,2,3,5-thiatriazol-1,1-dioxiden, 2. Mitt.
inferredcites →https://doi.org/10.1007/s10822-009-9264-5openalex-snapshot
Design of compound libraries for fragment screening
inferredcites →https://doi.org/10.1007/s10822-009-9280-5openalex-snapshot
Lessons for fragment library design: analysis of output from multiple screening campaigns
inferredcites →https://doi.org/10.1007/s10822-011-9521-2openalex-snapshot
The DINGO dataset: a comprehensive set of data for the SAMPL challenge
inferredcites →https://doi.org/10.1016/b978-0-12-381274-2.00020-0openalex-snapshot
Experiences in Fragment-Based Lead Discovery
inferredcites →https://doi.org/10.1016/j.ab.2005.02.027openalex-snapshot
Kinetic studies of small molecule interactions with protein kinases using biosensor technology
inferredcites →https://doi.org/10.1016/j.ab.2005.09.034openalex-snapshot
Analyzing a kinetic titration series using affinity biosensors
inferredcites →https://doi.org/10.1016/j.ab.2006.08.005openalex-snapshot
Exploring “one-shot” kinetics and small molecule analysis using the ProteOn XPR36 array biosensor
inferredcites →https://doi.org/10.1016/j.ab.2006.08.021openalex-snapshot
Comparative analysis of 10 small molecules binding to carbonic anhydrase II by different investigators using Biacore technology
inferredcites →https://doi.org/10.1016/j.ab.2006.08.032openalex-snapshot
High-resolution characterization of antibody fragment/antigen interactions using Biacore T100
inferredcites →https://doi.org/10.1016/j.bmcl.2013.03.028openalex-snapshot
Learning from our mistakes: The ‘unknown knowns’ in fragment screening
inferredcites →https://doi.org/10.1016/j.ddtec.2004.11.007openalex-snapshot
Lead- and drug-like compounds: the rule-of-five revolution
inferredcites →https://doi.org/10.1016/j.ddtec.2010.11.010openalex-snapshot
Fragment library design: efficiently hunting drugs in chemical space
inferredcites →https://doi.org/10.1016/j.drudis.2007.08.005openalex-snapshot
Integration of fragment screening and library design
inferredcites →https://doi.org/10.1016/s0065-2725(08)60184-1openalex-snapshot
Cycloaddition Reactions of Nitrile Oxides with Alkenes
inferredcites →https://doi.org/10.1016/s0169-409x(96)00423-1openalex-snapshot
Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings
inferredcites →https://doi.org/10.1016/s1359-6446(03)02831-9openalex-snapshot
A ‘Rule of Three’ for fragment-based lead discovery?
inferredcites →https://doi.org/10.1016/s1359-6446(05)03730-xopenalex-snapshot
Defining and maintaining a high quality screening collection: the GSK experience
inferredcites →https://doi.org/10.1016/s1359644602025722openalex-snapshot
Nonleadlikeness and leadlikeness in biochemical screening
inferredcites →https://doi.org/10.1021/bi3005126openalex-snapshot
Fragment-Based Approaches in Drug Discovery and Chemical Biology
inferredcites →https://doi.org/10.1021/ci025584yopenalex-snapshot
The Chemistry Development Kit (CDK): An Open-Source Java Library for Chemo- and Bioinformatics
inferredcites →https://doi.org/10.1021/ci049806zopenalex-snapshot
Design and Characterization of Libraries of Molecular Fragments for Use in NMR Screening against Protein Targets
inferredcites →https://doi.org/10.1021/jm020427bopenalex-snapshot
Kinase Inhibitors: Not Just for Kinases Anymore
inferredcites →https://doi.org/10.1021/jm030267jopenalex-snapshot
Characteristic Physical Properties and Structural Fragments of Marketed Oral Drugs
inferredcites →https://doi.org/10.1021/jm100164zopenalex-snapshot
Cheminformatic Tools for Medicinal Chemists
inferredcites →https://doi.org/10.1021/jm1013693openalex-snapshot
Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design
inferredcites →https://doi.org/10.1021/jm400830ropenalex-snapshot
Discovery and Biophysical Characterization of 2-Amino-oxadiazoles as Novel Antagonists of PqsR, an Important Regulator of Pseudomonas aeruginosa Virulence
inferredcites →https://doi.org/10.1021/jm700952vopenalex-snapshot
Surface Plasmon Resonance Based Assay for the Detection and Characterization of Promiscuous Inhibitors
inferredcites →https://doi.org/10.1021/jm9602928openalex-snapshot
The Properties of Known Drugs. 1. Molecular Frameworks
inferredcites →https://doi.org/10.1021/jm9903996openalex-snapshot
Properties of Known Drugs. 2. Side Chains
inferredcites →https://doi.org/10.1021/jo2011818openalex-snapshot
Atropisomerism-Induced Facial Selectivity in Nitrile Oxide Cycloadditions with 5-Methylenehydantoins
inferredcites →https://doi.org/10.1038/nature03194openalex-snapshot
Lessons from natural molecules
inferredcites →https://doi.org/10.1038/nature09454openalex-snapshot
Clinical efficacy of a RAF inhibitor needs broad target blockade in BRAF-mutant melanoma
inferredcites →https://doi.org/10.1038/nrd2220openalex-snapshot
A decade of fragment-based drug design: strategic advances and lessons learned
inferredcites →https://doi.org/10.1039/c2ob25271fopenalex-snapshot
Facial selectivity induced by N-aryl atropisomerism in benzonitrile oxide cycloadditions with 4-methylene-2-oxazolidinones
inferredcites →https://doi.org/10.1071/ch04295openalex-snapshot
N,N-Dialkyl (N'-Chlorosulfonyl)chloroformamidines in Heterocyclic Synthesis. I. The Preparation of [1,2,3,5]Thiatriazole and [1,3,2,4]Oxathiadiazole Derivatives
inferredcites →https://doi.org/10.1071/ch05070openalex-snapshot
N,N-Dialkyl-N'-Chlorosulfonylchloroformamidines in Heterocyclic Synthesis. II. Thiazolo-, Thiadiazolo-, and Oxadiazolo-Fused [1,2,4,6]Thiatriazine Dioxides
inferredcites →https://doi.org/10.1071/ch06367openalex-snapshot
N,N-Dialkyl-N'-Chlorosulfonyl Chloroformamidines in Heterocyclic Synthesis. III. Pyrido- and Pyridazo-Fused [1,2,4,6]Thiatriazine Dioxides
inferredcites →https://doi.org/10.1071/ch06368openalex-snapshot
N,N-Dialkyl-N'-Chlorosulfonyl Chloroformamidines in Heterocyclic Synthesis. IV. 3-Dialkylamino-1,1,8-trioxo-1H-1?6-pyrano[3,4-e][1,4,3]oxathiazines
inferredcites →https://doi.org/10.1071/ch07336openalex-snapshot
N, N-Dialkyl-N'-Chlorosulfonyl Chloroformamidines in Heterocyclic Synthesis. V* The Preparation of some Benzimidazo-Fused [1,2,4,6]Thiatriazine Dioxides
inferredcites →https://doi.org/10.1071/ch08059openalex-snapshot
N,N-Dialkyl-N'-Chlorosulfonyl Chloroformamidines in Heterocyclic Synthesis. VI The Preparation of Some Fused [1,4,2,6]Dithiadiazine Dioxides
inferredcites →https://doi.org/10.1071/ch08111openalex-snapshot
Regioselective 1,3-Dipolar Cycloaddition Reactions of 4-Methylene-2-oxazolidinones with Benzonitrile Oxide
inferredcites →https://doi.org/10.1071/ch08250openalex-snapshot
N,N-Dialkyl-N'-Chlorosulfonyl Chloroformamidines in Heterocyclic Synthesis. Part VII* 4-Dialkylamino[1,2,3,5]Benzoxathiadiazepine Dioxides and 4-Dialkylamino-[2,1,3,5]Benzothiatriazepine Dioxides
inferredcites →https://doi.org/10.1071/ch09479openalex-snapshot
Spiroheterocycles via Regioselective Cycloaddition Reactions of Nitrile Oxides with 5-Methylene-1H-pyrrol-2(5H)-ones
inferredcites →https://doi.org/10.1071/ch09581openalex-snapshot
N,N-Dialkyl-N'-Chlorosulfonyl Chloroformamidines in Heterocyclic Synthesis. Part VIII.* Novel Pyrazolo-Fused Oxathiadiazines and Thiatriazoles
inferredcites →https://doi.org/10.1071/ch09607openalex-snapshot
N,N-Dialkyl-N'-Chlorosulfonyl Chloroformamidines in Heterocyclic Synthesis. Part IX.* Novel Triazolo-Fused Thiatriazoles and Pyrazolo-Fused Oxathiazines
inferredcites →https://doi.org/10.1071/ch13270openalex-snapshot
N-Aryl Atropisomerism Induces Facial Selectivity in Benzonitrile Oxide Cycloadditions with Exocyclic Methylene Benzosultams
inferredcites →https://doi.org/10.1071/ch13302openalex-snapshot
Fragment Screening for the Modelling Community: SPR, ITC, and Crystallography
inferredcites →https://doi.org/10.1071/ch9931401openalex-snapshot
Diastereoselective Propionitrile Oxide Cycloaddition Reactions With Some γ-Substituted α-Methylene-γ-butyrolactones
inferredcites →https://doi.org/10.1073/pnas.0711741105openalex-snapshot
Discovery of a selective inhibitor of oncogenic B-Raf kinase with potent antimelanoma activity
inferredcites →https://doi.org/10.1073/pnas.1015271108openalex-snapshot
Route to three-dimensional fragments using diversity-oriented synthesis
inferredcites →https://doi.org/10.1158/1535-7163.mct-05-0313openalex-snapshot
A c-fms tyrosine kinase inhibitor, Ki20227, suppresses osteoclast differentiation and osteolytic bone destruction in a bone metastasis model
inferredcites →https://doi.org/10.1177/1087057106295507openalex-snapshot
Investigation of 3 Industry-Wide Applied Storage Conditions for Compound Libraries
inferredcites →https://doi.org/10.1177/1087057108326536openalex-snapshot
Stability of Screening Compounds in Wet DMSO
inferredcites →https://doi.org/10.1177/1087057112465979openalex-snapshot
Parallel Screening of Low Molecular Weight Fragment Libraries: Do Differences in Methodology Affect Hit Identification?
inferredcites →https://doi.org/10.1371/journal.pone.0029444openalex-snapshot
Structure of S. aureus HPPK and discovery of a new inhibitor
inferredcites →https://doi.org/10.1371/journal.pone.0040147openalex-snapshot
Small Molecule Inhibitors of the LEDGF Site of Human Immunodeficiency Virus Integrase Identified by Fragment Screening and Structure Based Design
inferredcites →https://doi.org/10.1517/17460441.1.3.225openalex-snapshot
Fragment screening by biochemical assay
inferredcites →https://doi.org/10.2174/092986711796391714openalex-snapshot
Managing the Liabilities Arising from Structural Alerts: A Safe Philosophy for Medicinal Chemists
inferredcites →https://doi.org/10.2174/138527210791616812openalex-snapshot
Spiro Isoxazolines via Nitrile Oxide 1,3-Dipolar Cycloaddition Reactions
inferredcites →https://doi.org/10.2174/1568026054637700openalex-snapshot
Library Design for Fragment Based Screening
inferredcites →https://doi.org/10.3851/imp1716openalex-snapshot
Structural Basis for a New Mechanism of Inhibition of H I V-1 Integrase Identified by Fragment Screening and Structure-Based Design
inferredcites →https://doi.org/10.3987/com-93-s49openalex-snapshot
Asymmetric Synthesis of a Homochiral D2-Isoxazoline Amino Acid Derivative

What points at this work

Incoming claims: where this work appears in other papers’ reference lists and arguments.

inferred← citeshttps://doi.org/10.1002/9783527677047.ch06openalex-snapshot
Fragment‐Based Lead Generation
inferred← citeshttps://doi.org/10.1016/j.bmcl.2023.129391openalex-snapshot
Synthesis and biological evaluation of 2-(Tetrazol-5-yl)sulfonylacetamides as inhibitors of Mycobacterium tuberculosis and Mycobacterium marinum
inferred← citeshttps://doi.org/10.1016/j.comche.2014.02.001openalex-snapshot
Combinatorial Chemistry Online Volume 16, Issue 3, March 2014
inferred← citeshttps://doi.org/10.1016/j.ejmech.2023.115637openalex-snapshot
3-Methoxy-2-phenylimidazo[1,2-b]pyridazines highly active against Mycobacterium tuberculosis and Mycobacterium marinum
inferred← citeshttps://doi.org/10.1016/j.ejmech.2024.116796openalex-snapshot
Discovery of 1,3,4-oxadiazoles with slow-action activity against Plasmodium falciparum malaria parasites
inferred← citeshttps://doi.org/10.1016/j.tetasy.2015.01.011openalex-snapshot
Functionalized α-oximinoketones as building blocks for the construction of imidazoline-based potential chiral auxiliaries
inferred← citeshttps://doi.org/10.1021/acs.jmedchem.5b01940openalex-snapshot
Native State Mass Spectrometry, Surface Plasmon Resonance, and X-ray Crystallography Correlate Strongly as a Fragment Screening Combination
inferred← citeshttps://doi.org/10.1038/s41598-019-52593-9openalex-snapshot
A suicide inhibitor of nematode trehalose-6-phosphate phosphatases
inferred← citeshttps://doi.org/10.1039/9781788018982-00188openalex-snapshot
Fragment-based Ligand Discovery (FBLD)
inferred← citeshttps://doi.org/10.1063/1.5122849openalex-snapshot
Fragment screening for a protein-protein interaction inhibitor to WDR5
inferred← citeshttps://doi.org/10.1071/ch13492openalex-snapshot
Fragment-Based Drug Discovery
inferred← citeshttps://doi.org/10.1071/ch14547openalex-snapshot
N,N-Dialkyl-N′-Chlorosulfonyl Chloroformamidines in Heterocyclic Synthesis. Part XI.* Some Substitution Reactions of Pyrazolo[1,5-b][1,2,4,6]thiatriazine 1,1-Dioxides
inferred← citeshttps://doi.org/10.1071/ch15587openalex-snapshot
Unexpected Isomerisation of a Fragment Analogue During Fragment-Based Screening of HIV Integrase Catalytic Core Domain
inferred← citeshttps://doi.org/10.1101/2023.03.09.531229openalex-snapshot
Discovery of 1,3,4-oxadiazoles with slow-action activity against Plasmodium falciparum malaria parasites
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