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New 2-Phenylthiazoles as Potential Sortase A Inhibitors: Synthesis, Biological Evaluation and Molecular Docking

https://doi.org/10.3390/molecules22111827
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What this work says

Outgoing claims: the papers this work cites, builds on, or argues with.

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Synthesis, biological evaluation and molecular docking of 2-phenyl-benzo[d]oxazole-7-carboxamide derivatives as potential Staphylococcus aureus Sortase A inhibitors
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Chinese herb medicine against Sortase A catalyzed transformations, a key role in gram-positive bacterial infection progress
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Sortase enzymes in Gram‐positive bacteria
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Combined Pharmacophore and 3D‐QSAR Study on A Series of Staphylococcus aureus Sortase A inhibitors
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Structure of the Cell Wall Anchor of Surface Proteins in Staphylococcus aureus
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The Rates of the Reaction of Heterocyclic (Thiophene and Thiazole) Bromoketones with Thioamides
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Antibacterial Activity of New Dibenzoxepinone Oximes with Fluorine and Trifluoromethyl Group Substituents
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Discovery of a New Class of Sortase A Transpeptidase Inhibitors to Tackle Gram-Positive Pathogens: 2-(2-Phenylhydrazinylidene)alkanoic Acids and Related Derivatives
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Structural Analysis of Sortase A Inhibitors

What points at this work

Incoming claims: where this work appears in other papers’ reference lists and arguments.

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Anti-Biofilm Potential and Mechanistic Insight into Sortasea Inhibition by Secondary Metabolites of C. Longa Against Staphylococcus Aureus and Streptococcus Mutans
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Structure‐Based Development of a Covalent Inhibitor Targeting Streptococcus Pyogenes over Staphylococcus Aureus Sortase A
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Asymmetric Disulfanylbenzamides as Irreversible and Selective Inhibitors of Staphylococcus aureus Sortase A
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Structural studies of Staphylococcus aureus Sortase inhibiton via Conus venom peptides
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Ligand-Based Design of Novel Thiazole-Quinazolinone Hybrids with Dual Antimicrobial and Anti-Virulence Activity Targeting Staphylococcal Sortase A
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Structure-Guided Design, Synthesis, and Antivirulence Assessment of Covalent Staphylococcus aureus Sortase A Inhibitors
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Thiazoles, Their Benzofused Systems, and Thiazolidinone Derivatives: Versatile and Promising Tools to Combat Antibiotic Resistance
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Analyses of the Antibiofilm Activity of o-Phenanthroline Monohydrate against Enterococcus faecalis and Staphylococcus aureus and the Mechanisms Underlying These Effects
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Inhibitory effect of a natural phenolic compound, 3- p-trans -coumaroyl-2-hydroxyquinic acid against the attachment phase of biofilm formation of Staphylococcus aureus through targeting sortase A
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Identification and prioritization of promising lead molecules fromSyzygium aromaticumagainst Sortase C fromStreptococcus pyogenes: anin silicoinvestigation
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Orientin mediates protection against MRSA-induced pneumonia by inhibiting Sortase A
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Synthesis, Reaction and Biological Activity of Thiazoles
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Recent Trends in Drug Development for the Treatment of Adenocarcinoma Breast Cancer: Thiazole, Triazole, and Thiosemicarbazone Analogues as Efficient Scaffolds
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ANTI-BIOFILM ACTIVITY EVALUATION AND MOLECULAR DOCKING STUDY OF SOME 2(3-PYRIDYL)-THIAZOLYL-1,3,4-OXADIAZOLINES
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Staphylococcal Biofilms: Challenges and Novel Therapeutic Perspectives
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An Insight into Rational Drug Design: The Development of In-House Azole Compounds with Antimicrobial Activity
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Design and Synthesis of Small Molecules as Potent Staphylococcus aureus Sortase A Inhibitors
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In-Silico Identified New Natural Sortase A Inhibitors Disrupt S. aureus Biofilm Formation
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New N-(oxazolylmethyl)-thiazolidinedione Active against Candida albicans Biofilm: Potential Als Proteins Inhibitors
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Identification of Novel Antistaphylococcal Hit Compounds Targeting Sortase A
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