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Simple Size-Independent Measure of Ligand Efficiency
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What this work says
Outgoing claims: the papers this work cites, builds on, or argues with.
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Group Efficiency: A Guideline for Hits‐to‐Leads Chemistry
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Novel arylsulfonamides possessing sub-picomolar HIV protease activities and potent anti-HIV activity against wild-type and drug-resistant viral strains
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A widely applicable set of descriptors
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Ligand Binding Efficiency: Trends, Physical Basis, and Implications
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Identification of N-(4-Piperidinyl)-4-(2,6-dichlorobenzoylamino)-1H-pyrazole-3-carboxamide (AT7519), a Novel Cyclin Dependent Kinase Inhibitor Using Fragment-Based X-Ray Crystallography and Structure Based Drug Design
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The maximal affinity of ligands
inferredcites →https://doi.org/10.1081/rrs-120037896openalex-snapshot
Thermodynamics of Protein–Ligand Interactions: History, Presence, and Future Aspects
inferredcites →https://doi.org/10.1093/jnci/81.8.577openalex-snapshot
New Soluble-Formazan Assay for HIV-1 Cytopathic Effects: Application to High-Flux Screening of Synthetic and Natural Products for AIDS-Antiviral Activity
inferredcites →https://doi.org/10.1093/nar/gkl999openalex-snapshot
BindingDB: a web-accessible database of experimentally determined protein-ligand binding affinities
What points at this work
Incoming claims: where this work appears in other papers’ reference lists and arguments.
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